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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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ADGRL2
adhesion G protein-coupled receptor L2
Chromosome 1 · 1p31.1
NCBI Gene: 23266Ensembl: ENSG00000117114.21HGNC: HGNC:18582UniProt: A0A6I8PIV6
66PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Highly ConstrainedReceptor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
G protein-coupled receptor activitypostsynaptic membraneG protein-coupled receptor signaling pathwayexcitatory synapse assemblycataractankylosing spondylitisovarian neoplasmbladder exstrophy
✦AI Summary

ADGRL2 (latrophilin-2) is an adhesion G protein-coupled receptor that functions as a mechanosensor and cell-adhesion mediator with diverse physiological roles 1. In the nervous system, ADGRL2 localizes to postsynaptic spines of excitatory synapses and mediates synapse specificity by interacting with presynaptic teneurins to promote synapse formation 1. Beyond synaptic function, ADGRL2 serves as a force-sensitive mechanoreceptor: it is essential for equilibrioception in vestibular hair cells, where it converts mechanical force stimuli into increased channel opening of TMC1, enabling mechanotransduction and balance maintenance 2. In endothelial cells, ADGRL2 mediates fluid shear stress mechanotransduction at cell-cell junctions, activating Gαi2 and Gαq/11 signaling upstream of the PECAM-1 complex to regulate flow-dependent angiogenesis and artery remodeling; human genetic variants in ADGRL2 correlate with cardiovascular disease 3. ADGRL2 also provides cytoprotection against septic endothelial dysfunction by preserving eNOS activity and enhancing antioxidative NRF2 responses 4. In epithelial tissues, ADGRL2 specifically activates Gα13 to enable epidermal differentiation 5. In cancer, ADGRL2 polymorphisms associate with severe malaria risk 6, and ADGRL2 promotes breast cancer cell migration, adhesion, and invasion through ROCK and PKA signaling 7. These findings establish ADGRL2 as a multifunctional mechanoreceptor critical for neuronal, vascular, and epithelial homeostasis.

Sources cited
1
ADGRL2 nomenclature and classification as adhesion GPCR; synaptic localization and interaction with teneurins
PMID: 25713288
2
ADGRL2 is essential for equilibrioception; functions as force-sensitive mechanoreceptor converting force into TMC1 channel opening in vestibular hair cells
PMID: 39966628
3
ADGRL2 mediates fluid shear stress mechanotransduction in endothelial cells; required for flow-dependent angiogenesis and artery remodeling; ADGRL2 variants correlate with cardiovascular disease
PMID: 38886581
4
ADGRL2 protects endothelial cells from LPS-induced dysfunction by preserving eNOS activity and enhancing NRF2-mediated antioxidative responses
PMID: 39594576
5
ADGRL2 selectively activates Gα13 to enable epidermal differentiation; critical interaction between ADGRL2 intracellular loop 3 and Gα13 QQQ glutamine triplet
PMID: 41252157
6
ADGRL2 promotes breast cancer cell migration, adhesion, and invasion through C-terminal fragment activation of ROCK and PKA signaling via Gα12/13 and Gαs coupling
PMID: 40545252
7
LPHN2/ADGRL2 polymorphisms associate with risk of severe Plasmodium falciparum malaria in children
PMID: 30033078
Disease Associationsⓘ20
cataractOpen Targets
0.35Weak
ankylosing spondylitisOpen Targets
0.34Weak
ovarian neoplasmOpen Targets
0.32Weak
bladder exstrophyOpen Targets
0.31Weak
self-injurious ideationOpen Targets
0.31Weak
ulcerative colitisOpen Targets
0.31Weak
systemic lupus erythematosusOpen Targets
0.30Weak
type 1 diabetes mellitusOpen Targets
0.30Weak
autoimmune diseaseOpen Targets
0.30Weak
autoimmune thyroid diseaseOpen Targets
0.30Weak
juvenile idiopathic arthritisOpen Targets
0.30Weak
Crohn's diseaseOpen Targets
0.30Weak
common variable immunodeficiencyOpen Targets
0.30Weak
celiac diseaseOpen Targets
0.30Weak
psoriasisOpen Targets
0.30Weak
obesityOpen Targets
0.29Weak
ovarian dysfunctionOpen Targets
0.28Weak
type 2 diabetes mellitusOpen Targets
0.26Weak
cardiac arrestOpen Targets
0.25Weak
obsessive-compulsive disorderOpen Targets
0.21Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
TENM4Protein interaction99%TENM1Protein interaction99%TENM3Protein interaction98%UNC5DProtein interaction98%GNAT3Protein interaction98%UNC5CLProtein interaction97%
Tissue Expression6 tissues
Heart
100%
Lung
73%
Ovary
60%
Liver
49%
Brain
15%
Bone Marrow
1%
Gene Interaction Network
Click a node to explore
ADGRL2TENM4TENM1TENM3UNC5DGNAT3UNC5CL
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt O95490
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.30Highly Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.22 [0.16–0.30]
RankingsWhere ADGRL2 stands among ~20K protein-coding genes
  • #7,033of 20,598
    Most Researched66
  • #1,158of 17,882
    Most Constrained (LOEUF)0.30 · top 10%
Genes detectedADGRL2
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
International Union of Basic and Clinical Pharmacology. XCIV. Adhesion G protein-coupled receptors.
PMID: 25713288
Pharmacol Rev · 2015
1.00
2
A force-sensitive adhesion GPCR is required for equilibrioception.
PMID: 39966628
Cell Res · 2025
0.90
3
Latrophilin-2 mediates fluid shear stress mechanotransduction at endothelial junctions.
PMID: 38886581
EMBO J · 2024
0.80
4
The Adhesion GPCR ADGRL2/LPHN2 Can Protect Against Cellular and Organismal Dysfunction.
PMID: 39594576
Cells · 2024
0.70
5
A correlation study of adhesion G protein-coupled receptors as potential therapeutic targets in Uterine Corpus Endometrial cancer.
PMID: 35413679
Int Immunopharmacol · 2022
0.60