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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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ARHGAP18
Rho GTPase activating protein 18
Chromosome 6 · 6q22.33
NCBI Gene: 93663Ensembl: ENSG00000146376.12HGNC: HGNC:21035UniProt: Q8N392
46PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
GTPase activator activitycadherin bindingrufflecytoplasmic microtubuleaortic diseaseimmune system diseaseobesityprostatitis
✦AI Summary

ARHGAP18 (Rho GTPase activating protein 18) functions as a negative regulator of Rho GTPases, particularly RhoA and RhoC, by enhancing their GTP hydrolysis and converting them to an inactive GDP-bound state 1. The protein plays critical roles in endothelial cell biology, where it is essential for flow-dependent endothelial cell alignment in the direction of blood flow, a protective response against atherosclerosis 23. ARHGAP18 deficiency leads to loss of endothelial alignment, disrupted cell junctions, and promotes pro-inflammatory phenotypes 2. The protein regulates cellular processes through multiple pathways, including the YAP signaling cascade, where ARHGAP18 acts upstream of YAP and controls its nuclear localization 3. In cancer contexts, ARHGAP18 exhibits complex, context-dependent roles. In hepatocellular carcinoma, it is upregulated by transcription factor GATA1 and promotes proliferation and invasion 4. In triple-negative breast cancer, ARHGAP18 overexpression paradoxically enhances metastasis by reducing RhoA activation 5. The protein also regulates endothelial permeability and inflammatory responses, with advanced glycosylation end products decreasing ARHGAP18 expression in diabetic complications 1. Additionally, ARHGAP18 appears protective in COPD, where miR-613-mediated upregulation inhibits cigarette smoke-induced apoptosis and epithelial-mesenchymal transition 6.

Sources cited
1
ARHGAP18 negatively regulates RhoA by enhancing GTP hydrolysis and converting to inactive GDP-bound state
PMID: 32016689
2
ARHGAP18 is essential for flow-dependent endothelial cell alignment and protects against atherosclerosis
PMID: 30630384
3
ARHGAP18 acts upstream of YAP signaling and is required for endothelial cell alignment under flow
PMID: 32013974
4
ARHGAP18 is upregulated by GATA1 and promotes proliferation and invasion in hepatocellular carcinoma
PMID: 37171759
5
ARHGAP18 overexpression enhances metastasis in triple-negative breast cancer by reducing RhoA activation
PMID: 28619708
6
miR-613-mediated ARHGAP18 upregulation protects against cigarette smoke-induced apoptosis and EMT in COPD
PMID: 40698118
Disease Associationsⓘ20
aortic diseaseOpen Targets
0.32Weak
immune system diseaseOpen Targets
0.31Weak
obesityOpen Targets
0.30Weak
prostatitisOpen Targets
0.27Weak
myopiaOpen Targets
0.09Suggestive
refractive errorOpen Targets
0.09Suggestive
HypermetropiaOpen Targets
0.09Suggestive
metabolic diseaseOpen Targets
0.09Suggestive
response to antihypertensive drugOpen Targets
0.08Suggestive
benign chondrogenic neoplasmOpen Targets
0.08Suggestive
retinal detachmentOpen Targets
0.07Suggestive
retinal perforationOpen Targets
0.07Suggestive
ovarian dysfunctionOpen Targets
0.07Suggestive
vascular diseaseOpen Targets
0.06Suggestive
Abnormality of refractionOpen Targets
0.06Suggestive
amblyopiaOpen Targets
0.06Suggestive
AstigmatismOpen Targets
0.06Suggestive
eye diseaseOpen Targets
0.06Suggestive
Progressive visual lossOpen Targets
0.06Suggestive
Rare genetic vascular diseaseOpen Targets
0.06Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
PEAK3Shared pathway50%ARHGAP15Shared pathway50%RHOFShared pathway38%RHOBTB1Shared pathway33%ARHGAP40Shared pathway33%ARHGAP9Shared pathway33%
Tissue Expression6 tissues
Lung
100%
Heart
39%
Bone Marrow
25%
Ovary
21%
Brain
12%
Liver
11%
Gene Interaction Network
Click a node to explore
ARHGAP18PEAK3ARHGAP15RHOFRHOBTB1ARHGAP40ARHGAP9
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q8N392
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.93LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.75 [0.61–0.93]
RankingsWhere ARHGAP18 stands among ~20K protein-coding genes
  • #9,300of 20,598
    Most Researched46
  • #8,603of 17,882
    Most Constrained (LOEUF)0.93
Genes detectedARHGAP18
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Chemotherapy-induced cellular senescence promotes stemness of aggressive B-cell non-Hodgkin's lymphoma via CCR7/ARHGAP18/IKBα signaling activation.
PMID: 39773566
J Immunother Cancer · 2025
1.00
2
ARHGAP18: A Flow-Responsive Gene That Regulates Endothelial Cell Alignment and Protects Against Atherosclerosis.
PMID: 30630384
J Am Heart Assoc · 2019
0.90
3
Advanced glycosylation end products (AGEs) controls proliferation, invasion and permeability through orchestrating ARHGAP18/RhoA pathway in human umbilical vein endothelial cells.
PMID: 32016689
Glycoconj J · 2020
0.80
4
Upregulation of ARHGAP18 by miR-613 Inhibits Cigarette Smoke Extract-Induced Apoptosis and Epithelial-Mesenchymal Transition in Bronchial Epithelial Cells.
PMID: 40698118
Int J Chron Obstruct Pulmon Dis · 2025
0.70
5
Activation of human gonadotropin-releasing hormone receptor promotes down regulation of ARHGAP18 and regulates the cell invasion of MDA-MB-231 cells.
PMID: 28709956
Mol Cell Endocrinol · 2018
0.60