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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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DAPK3
death associated protein kinase 3
Chromosome 19 · 19p13.3
NCBI Gene: 1613Ensembl: ENSG00000167657.15HGNC: HGNC:2676UniProt: B3KNJ3
101PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
ApoptosisKinaseTranscription FactorTumor Suppressor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein kinase activityprotein serine/threonine kinase activityprotein bindingATP bindingneurodegenerative diseaseneoplasmattention deficit hyperactivity disordergastric cancer
✦AI Summary

DAPK3 is a serine/threonine kinase functioning as a tumor suppressor with pleiotropic roles in cellular regulation. Primary function: DAPK3 regulates apoptosis, autophagy, cytoskeletal dynamics, and smooth muscle contraction through phosphorylation of multiple substrates including myosin light chains, ribosomal proteins, and kinases 1. Mechanism: DAPK3 coordinates post-translational modifications of STING to activate the cGAMP-STING-IFN-β pathway, driving anti-tumor immunity through CD8+ T cell and dendritic cell infiltration 1. In gastric cancer, DAPK3 phosphorylates ULK1 at Ser556 to activate autophagy-dependent tumor suppression 2. DAPK3 regulates actin cytoskeleton reorganization and myogenic responses in cerebral arteries independently of myosin light chain phosphorylation, likely through focal adhesion dynamics 3. In triple-negative breast cancer, DAPK3/LUZP1 heterodimers promote EMT and invasion by suppressing desmoplakin levels 4. Disease relevance: DAPK3 downregulation correlates with aggressive behavior in endometrial, gastric, and breast cancers, predicting poor prognosis 526. Metabolic regulation: insulin and glucose reciprocally alter DAPK3 DNA methylation in skeletal muscle, affecting palmitate oxidation 7. Clinical significance: DAPK3 inhibitors may provide therapeutic benefit in hypertension by reducing vascular smooth muscle contractility 8, while restoring DAPK3 activity represents a potential cancer immunotherapy strategy.

Sources cited
1
DAPK3 drives tumor-intrinsic immunity through STING-mediated cytosolic DNA sensing and IFN-β production
PMID: 33767426
2
DAPK3 is overexpressed in triple-negative breast cancer and promotes migration/invasion through desmoplakin suppression via LUZP1 interaction
PMID: 39319326
3
Insulin increases and glucose decreases DAPK3 DNA methylation in skeletal muscle, affecting metabolism
PMID: 28011458
4
DAPK3 inhibitors reduce vascular smooth muscle contractility and blood pressure in hypertensive mice
PMID: 30033129
5
DAPK3 regulates myogenic responses in cerebral arteries through actin cytoskeleton mechanisms
PMID: 37084168
6
Low DAPK3 expression correlates with aggressive endometrial cancer and poor patient prognosis
PMID: 27320893
7
DAPK3 suppresses gastric cancer by phosphorylating ULK1 to activate autophagy
PMID: 33037394
8
DAPK3 is required for normal development and acts as tumor suppressor in breast tissue
PMID: 25304685
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.21Weak
neoplasmOpen Targets
0.10Weak
attention deficit hyperactivity disorderOpen Targets
0.09Suggestive
gastric cancerOpen Targets
0.09Suggestive
prostate cancerOpen Targets
0.08Suggestive
triple-negative breast cancerOpen Targets
0.07Suggestive
movement disorderOpen Targets
0.07Suggestive
attention deficit-hyperactivity disorder 8Open Targets
0.07Suggestive
hereditary attention deficit-hyperactivity disorderOpen Targets
0.07Suggestive
intellectual disability, autosomal recessive 59Open Targets
0.07Suggestive
schizophrenia 15Open Targets
0.07Suggestive
brain aneurysmOpen Targets
0.06Suggestive
cryopyrin-associated periodic syndromeOpen Targets
0.06Suggestive
Phelan-McDermid syndromeOpen Targets
0.05Suggestive
autismOpen Targets
0.05Suggestive
Tourette syndromeOpen Targets
0.05Suggestive
X-linked non-syndromic intellectual disabilityOpen Targets
0.04Suggestive
intellectual disability, autosomal dominant 50Open Targets
0.04Suggestive
Potocki-Lupski syndromeOpen Targets
0.04Suggestive
breast cancerOpen Targets
0.04Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
CALML4Protein interaction100%CALML5Protein interaction100%CALML3Protein interaction100%CALML6Protein interaction100%MAPK3Protein interaction99%LUZP1Protein interaction99%
Tissue Expression6 tissues
Lung
100%
Heart
97%
Ovary
74%
Brain
50%
Liver
46%
Bone Marrow
16%
Gene Interaction Network
Click a node to explore
DAPK3CALML4CALML5CALML3CALML6MAPK3LUZP1
PROTEIN STRUCTURE
Preparing viewer…
PDB3BHY · 1.24 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.18LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.77 [0.51–1.18]
RankingsWhere DAPK3 stands among ~20K protein-coding genes
  • #4,714of 20,598
    Most Researched101 · top quartile
  • #12,398of 17,882
    Most Constrained (LOEUF)1.18
Genes detectedDAPK3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
The tumor suppressor kinase DAPK3 drives tumor-intrinsic immunity through the STING-IFN-β pathway.
PMID: 33767426
Nat Immunol · 2021
1.00
2
Death-associated protein kinase 3 modulates migration and invasion of triple-negative breast cancer cells.
PMID: 39319326
PNAS Nexus · 2024
0.90
3
Insulin and Glucose Alter Death-Associated Protein Kinase 3 (DAPK3) DNA Methylation in Human Skeletal Muscle.
PMID: 28011458
Diabetes · 2017
0.80
4
Targeting Pim Kinases and DAPK3 to Control Hypertension.
PMID: 30033129
Cell Chem Biol · 2018
0.70
5
Death-associated protein kinase 3 regulates the myogenic reactivity of cerebral arteries.
PMID: 37084168
Exp Physiol · 2023
0.60