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GeneE
10 sources retrieved Β· Most recent: April 2026 Β· Index updated 14 days ago
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DPH5
diphthamide biosynthesis 5
Chromosome 1 Β· 1p21.2
NCBI Gene: 51611Ensembl: ENSG00000117543.23HGNC: HGNC:24270UniProt: B3KWP1
27PubMed Papers
21Diseases
0Drugs
3Pathogenic Variants
CLINICAL
OMIM Disease Gene
DATA QUALITY
βœ“ Experimental GO Evidenceβœ“ Swiss-Prot Reviewed
diphthine methyl ester synthase activityprotein histidyl modification to diphthamidecytosoldiphthine synthase activityneurodevelopmental disorder with short stature, prominent forehead, and feeding difficultiesneurodegenerative diseaseovarian dysfunctionNeurodevelopmental disorder
✦AI Summary

DPH5 encodes a cytosolic S-adenosyl-L-methionine-dependent methyltransferase that catalyzes four successive methylation reactions on modified histidine residues in translation elongation factor 2 (eEF2), forming diphthine methyl ester as an intermediate in diphthamide biosynthesis 1. Diphthamide is a post-translational modification essential for messenger RNA translation and ribosomal protein synthesis 1. DPH5 functions as part of a seven-protein system (DPH1-7) required for complete diphthamide synthesis, with DPH5 catalyzing the second biosynthetic step 2. Loss-of-function DPH5 variants cause DPH5-related diphthamide-deficiency syndrome, manifesting as embryonic lethality or profound neurodevelopmental disorders with multisystem abnormalities including craniofacial dysmorphology, developmental delay, intellectual disability, and growth impairment 13. Homozygous DPH5 mutations are embryonically lethal in mice, while hypomorphic variants produce milder phenotypes with variable severity 3. Recent evidence suggests DPH5 dysregulation may be implicated in intervertebral disc degeneration, with decreased DPH5 expression observed in degenerative nucleus pulposus tissue 4. Functionally compromised DPH5 variants can affect cellular sensitivity to ADP-ribosylating toxins and immunotoxin-based therapies that target diphthamide-containing eEF2 5.

Sources cited
1
DPH5 is a novel cause of embryonic lethality and profound neurodevelopmental delays; DPH5 catalyzes methylations of eEF2 histidine; diphthamide is essential for mRNA translation
PMID: 35482014
2
DPH5 catalyzes the second step of diphthamide biosynthesis, generating methylated diphthine as an intermediate; diphthamide synthesis requires seven proteins (DPH1-7)
PMID: 24739148
3
DPH5-related diphthamide deficiency syndrome causes developmental delay, intellectual disability, and multisystemic abnormalities; hypomorphic variants produce milder phenotypes
PMID: 40725455
4
DPH5 expression is decreased in degenerative nucleus pulposus tissue in intervertebral disc degeneration
PMID: 39953636
5
DPH5 variants affect diphthamide synthesis and cellular sensitivity to ADP-ribosylating toxins and immunotoxin-based therapies
PMID: 28245596
Disease Associationsβ“˜21
neurodevelopmental disorder with short stature, prominent forehead, and feeding difficultiesOpen Targets
0.68Moderate
neurodegenerative diseaseOpen Targets
0.37Weak
ovarian dysfunctionOpen Targets
0.29Weak
Neurodevelopmental disorderOpen Targets
0.19Weak
multiple sclerosisOpen Targets
0.05Suggestive
hyperaldosteronismOpen Targets
0.03Suggestive
response to stimulusOpen Targets
0.02Suggestive
type 2 diabetes mellitusOpen Targets
0.02Suggestive
Neurodevelopmental delayOpen Targets
0.02Suggestive
neoplasmOpen Targets
0.01Suggestive
Intellectual disabilityOpen Targets
0.00Suggestive
myelodysplastic syndromeOpen Targets
0.00Suggestive
cancerOpen Targets
0.00Suggestive
chronic lymphocytic leukemiaOpen Targets
0.00Suggestive
hepatocellular carcinomaOpen Targets
0.00Suggestive
Uveal MelanomaOpen Targets
0.00Suggestive
inflammatory bowel diseaseOpen Targets
0.00Suggestive
rasopathyOpen Targets
0.00Suggestive
pancreatic carcinomaOpen Targets
0.00Suggestive
SepsisOpen Targets
0.00Suggestive
Neurodevelopmental disorder with short stature, prominent forehead, and feeding difficultiesUniProt
Pathogenic Variants3
NM_015958.3(DPH5):c.779A>G (p.His260Arg)Pathogenic
Neurodevelopmental disorder with short stature, prominent forehead, and feeding difficulties
β˜…β˜…β˜†β˜†2023β†’ Residue 260
NM_015958.3(DPH5):c.619C>T (p.Arg207Ter)Pathogenic
Neurodevelopmental disorder with short stature, prominent forehead, and feeding difficulties
β˜†β˜†β˜†β˜†2022β†’ Residue 207
NM_015958.3(DPH5):c.329A>G (p.Asn110Ser)Pathogenic
Neurodevelopmental disorder with short stature, prominent forehead, and feeding difficulties
β˜†β˜†β˜†β˜†2022β†’ Residue 110
View on ClinVar β†—
Related Genes
DPH1Protein interaction100%EEF2Protein interaction99%DPH6Protein interaction88%DPH2Protein interaction84%DPH3Protein interaction81%DPH7Protein interaction79%
Tissue Expression6 tissues
Ovary
100%
Heart
98%
Brain
76%
Liver
58%
Lung
43%
Bone Marrow
39%
Gene Interaction Network
Click a node to explore
DPH5DPH1EEF2DPH6DPH2DPH3DPH7
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted Β· UniProt Q9H2P9
View on AlphaFold β†—
Constraintβ“˜
LOEUFβ“˜
1.29LoF Tolerant
pLIβ“˜
0.00Tolerant
Observed/Expected LoF0.88 [0.61–1.29]
RankingsWhere DPH5 stands among ~20K protein-coding genes
  • #12,549of 20,598
    Most Researched27
  • #4,133of 5,498
    Most Pathogenic Variants3
  • #13,639of 17,882
    Most Constrained (LOEUF)1.29
Genes detectedDPH5
Sources retrieved10 papers
Response timeβ€”
πŸ“„ Sources
10β–Ό
1
A diarylheptanoid compound from Alpinia officinarum Hance ameliorates high glucose-induced insulin resistance by regulating PI3K/AKT-Nrf2-GSK3Ξ² signaling pathways in HepG2 cells.
PMID: 35605918
J Ethnopharmacol Β· 2022
1.00
2
A novel DPH5-related diphthamide-deficiency syndrome causing embryonic lethality or profound neurodevelopmental disorder.
PMID: 35482014
Genet Med Β· 2022
0.90
3
Integrated bulk and single-cell RNA sequencing to identify potential biomarkers in intervertebral disc degeneration.
PMID: 39953636
Eur J Med Res Β· 2025
0.80
4
Expanding the Phenotypic Spectrum Associated with DPH5-Related Diphthamide Deficiency.
PMID: 40725455
Genes (Basel) Β· 2025
0.70
5
Influence of DPH1 and DPH5 Protein Variants on the Synthesis of Diphthamide, the Target of ADPRibosylating Toxins.
PMID: 28245596
Toxins (Basel) Β· 2017
0.60