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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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FBXO45
F-box protein 45
Chromosome 3 · 3q29
NCBI Gene: 200933Ensembl: ENSG00000174013.8HGNC: HGNC:29148UniProt: P0C2W1
57PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingprotein ubiquitinationnucleoplasmprotein K48-linked ubiquitinationhepatocellular carcinomabreast cancernon-small cell lung carcinomapachyonychia congenita
✦AI Summary

FBXO45 is a substrate-recognition component of SCF E3 ubiquitin ligase complexes that regulates protein degradation through the ubiquitin-proteasome system 1. The protein functions as an oncogene in multiple cancer types, promoting tumorigenesis through diverse mechanisms. In pancreatic cancer, FBXO45 facilitates progression by targeting tumor suppressor USP49 for ubiquitination and degradation 2. In lung cancers, FBXO45 is overexpressed and associated with poor prognosis, promoting metastasis and the Warburg effect while reducing ferroptosis through stabilization of ZEB1 by inhibiting its ubiquitination 34. In hepatocellular carcinoma with TP53 mutations, FBXO45 drives lung metastasis by promoting TFG ubiquitination and activating the ATF2-NF-κB pathway 5. Beyond cancer, FBXO45 plays roles in HIV-1 regulation by promoting Tat ubiquitination and SQSTM1/p62-mediated autophagic degradation, thereby restricting viral replication 6. In diabetic endothelial dysfunction, FBXO45 mediates GPX4 ubiquitination leading to oxidative stress 7. FBXO45 also regulates germinal center formation and B-cell lymphomagenesis through control of GEF-H1 8. These diverse functions establish FBXO45 as a critical regulator of cellular homeostasis and a potential therapeutic target across multiple diseases.

Sources cited
1
FBXO45 is a substrate-recognition subunit of E3 ligases with roles in human diseases including malignancies
PMID: 32655893
2
FBXO45 facilitates pancreatic cancer progression by targeting USP49 for ubiquitination and degradation
PMID: 35279684
3
FBXO45 promotes Warburg effect and reduces ferroptosis in NSCLC by decreasing ZEB1 ubiquitination
PMID: 39016138
4
FBXO45 is overexpressed in squamous-cell lung carcinoma and associated with poor prognosis
PMID: 29728763
5
FBXO45 drives hepatocellular carcinoma lung metastasis through TFG ubiquitination and ATF2-NF-κB pathway activation
PMID: 41030651
6
FBXO45 restricts HIV-1 replication by promoting Tat ubiquitination and autophagic degradation
PMID: 39936917
7
FBXO45 mediates GPX4 ubiquitination contributing to diabetic endothelial dysfunction
PMID: 40275362
8
FBXO45 controls germinal center formation and B-cell lymphomagenesis through GEF-H1 regulation
PMID: 39820335
Disease Associationsⓘ20
hepatocellular carcinomaOpen Targets
0.09Suggestive
breast cancerOpen Targets
0.08Suggestive
non-small cell lung carcinomaOpen Targets
0.07Suggestive
pachyonychia congenitaOpen Targets
0.07Suggestive
neoplasmOpen Targets
0.06Suggestive
skin cancerOpen Targets
0.05Suggestive
triple-negative breast cancerOpen Targets
0.05Suggestive
lymphomaOpen Targets
0.05Suggestive
skin neoplasmOpen Targets
0.04Suggestive
glomerulonephritisOpen Targets
0.04Suggestive
diffuse large B-cell lymphomaOpen Targets
0.04Suggestive
asthmaOpen Targets
0.04Suggestive
esophageal squamous cell carcinomaOpen Targets
0.03Suggestive
intrahepatic bile duct cancerOpen Targets
0.03Suggestive
liver cancerOpen Targets
0.03Suggestive
cancerOpen Targets
0.03Suggestive
schizophreniaOpen Targets
0.03Suggestive
gliomaOpen Targets
0.03Suggestive
gastric cancerOpen Targets
0.03Suggestive
colorectal carcinomaOpen Targets
0.03Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
SIAH1Protein interaction100%SKP1Protein interaction100%CUL1Protein interaction100%FBXW7Protein interaction100%UNC13AProtein interaction86%SPRYD3Protein interaction79%
Tissue Expression6 tissues
Bone Marrow
100%
Brain
99%
Heart
24%
Liver
21%
Ovary
17%
Lung
16%
Gene Interaction Network
Click a node to explore
FBXO45SIAH1SKP1CUL1FBXW7UNC13ASPRYD3
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt P0C2W1
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.40Moderately Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.15 [0.07–0.40]
RankingsWhere FBXO45 stands among ~20K protein-coding genes
  • #7,959of 20,598
    Most Researched57
  • #1,954of 17,882
    Most Constrained (LOEUF)0.40 · top quartile
Genes detectedFBXO45
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
FBXO45 is a potential therapeutic target for cancer therapy.
PMID: 32655893
Cell Death Discov · 2020
1.00
2
SETD7 drives diabetic endothelial dysfunction through FBXO45-mediated GPX4 ubiquitylation.
PMID: 40275362
Cardiovasc Diabetol · 2025
0.90
3
Elevated FBXO45 promotes TFG ubiquitination and drives lung metastasis of hepatocellular carcinoma.
PMID: 41030651
JHEP Rep · 2025
0.80
4
FBXO45 restricts HIV-1 replication by inducing SQSTM1/p62-mediated autophagic degradation of Tat.
PMID: 39936917
J Virol · 2025
0.70
5
Fbxo45 facilitates pancreatic carcinoma progression by targeting USP49 for ubiquitination and degradation.
PMID: 35279684
Cell Death Dis · 2022
0.60