HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
50 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
HSPA5
heat shock protein family A (Hsp70) member 5
Chromosome 9 · 9q33.3
NCBI Gene: 3309Ensembl: ENSG00000044574.10HGNC: HGNC:5238UniProt: P11021
1,168PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Hub Gene
RESEARCH IMPACT
Highly StudiedTrending
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
membraneendoplasmic reticulum lumencytoplasmregulation of IRE1-mediated unfolded protein responsedengue diseaseneurodegenerative diseaseneoplasmhepatocellular carcinoma
✦AI Summary

HSPA5 (also known as BiP/GRP78) is a heat shock protein family A member 5 that functions as a master regulator of endoplasmic reticulum (ER) homeostasis and stress responses. As an Hsp70 family chaperone localized in the ER lumen, HSPA5 assists protein folding via its nucleotide-binding and substrate-binding domains, facilitates ER protein translocation, regulates calcium homeostasis, and mediates ER-associated protein degradation 1. Upon ER stress, HSPA5 initiates the unfolded protein response (UPR) to manage misfolded protein accumulation and can crosstalk with apoptosis machinery 12. Beyond its canonical ER function, cell surface-translocated HSPA5 serves as a receptor for pathogenic fungi, particularly CotH proteins from Mucorales species, facilitating epithelial cell invasion during mucormycosis infection 3. In cancer contexts, HSPA5 negatively regulates ferroptosis by stabilizing glutathione peroxidase 4 (GPX4), promoting chemotherapy resistance in pancreatic adenocarcinoma 4. Additionally, HSPA5 palmitoylation and deubiquitination regulate its ER localization and activity, influencing cancer cell survival versus apoptosis decisions 56. HSPA5 is associated with multiple diseases including cancers, cardiovascular disease, neurodegenerative conditions, and immunological disorders 1, making it an emerging therapeutic target across diverse pathologies.

Sources cited
1
HSPA5 encodes BiP, an Hsp70 chaperone with nucleotide-binding and substrate-binding domains that facilitates protein folding, translocation, calcium homeostasis, and ER-associated protein degradation; initiates UPR and associates with multiple diseases
PMID: 28286085
2
GRP78/HSPA5 is the master regulator of the unfolded protein response in the ER; under stress, membrane-overexpressed HSPA5 becomes a tool for pathogen entry
PMID: 30978349
3
HSPA5 acts as a receptor for R. delemar CotH3 in nasal epithelial cells, playing a role in mucormycosis epithelial cell invasion and rhinoorbital/cerebral disease progression
PMID: 32487760
4
HSPA5 negatively regulates ferroptosis in pancreatic ductal adenocarcinoma by binding and protecting glutathione peroxidase 4 from degradation, promoting chemotherapy resistance
PMID: 28130223
5
ZDHHC9-mediated S-palmitoylation of HSPA5/BiP at Cys420 inhibits the unfolded protein response and promotes bladder cancer progression
PMID: 39002690
6
GCS1 recruits USP10 to deubiquitinate GRP78/HSPA5, reducing ER stress-mediated apoptosis and promoting colorectal cancer cell proliferation and metastasis
PMID: 39267084
Disease Associationsⓘ20
dengue diseaseOpen Targets
0.51Moderate
neurodegenerative diseaseOpen Targets
0.47Moderate
neoplasmOpen Targets
0.12Weak
hepatocellular carcinomaOpen Targets
0.12Weak
cancerOpen Targets
0.12Weak
gastric cancerOpen Targets
0.11Weak
gliomaOpen Targets
0.11Weak
breast cancerOpen Targets
0.11Weak
colorectal carcinomaOpen Targets
0.11Weak
rheumatoid arthritisOpen Targets
0.11Weak
anxiety disorderOpen Targets
0.11Weak
head and neck squamous cell carcinomaOpen Targets
0.11Weak
COVID-19Open Targets
0.11Weak
Parkinson diseaseOpen Targets
0.11Weak
esophageal squamous cell carcinomaOpen Targets
0.10Weak
acute myeloid leukemiaOpen Targets
0.10Weak
oral squamous cell carcinomaOpen Targets
0.10Weak
cervical cancerOpen Targets
0.10Suggestive
renal cell carcinomaOpen Targets
0.10Suggestive
lung cancerOpen Targets
0.10Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
CALUProtein interaction100%CLGNProtein interaction100%SEL1LProtein interaction100%SYVN1Protein interaction100%TAPBPProtein interaction100%ERP29Protein interaction100%
Tissue Expression6 tissues
Bone Marrow
100%
Liver
53%
Heart
39%
Lung
38%
Ovary
23%
Brain
21%
Gene Interaction Network
Click a node to explore
HSPA5CALUCLGNSEL1LSYVN1TAPBPERP29
PROTEIN STRUCTURE
Preparing viewer…
PDB5F0X · 1.60 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.50Moderately Constrained
pLIⓘ
0.98Intolerant
Observed/Expected LoF0.32 [0.21–0.50]
RankingsWhere HSPA5 stands among ~20K protein-coding genes
  • #126of 20,598
    Most Researched1,168 · top 1%
  • #3,043of 17,882
    Most Constrained (LOEUF)0.50 · top quartile
Genes detectedHSPA5
Sources retrieved50 papers
Response time—
📄 Sources
50▼
1
GRP78: A cell's response to stress.
PMID: 30978349
Life Sci · 2019
1.00
2
HSPA5 Regulates Ferroptotic Cell Death in Cancer Cells.
PMID: 28130223
Cancer Res · 2017
0.90
3
Efficacy of DMARDs and methylprednisolone treatment on the gene expression levels of HSPA5, MMD, and non-coding RNAs MALAT1, H19, miR-199a-5p, and miR-1-3p, in patients with rheumatoid arthritis.
PMID: 35623291
Int Immunopharmacol · 2022
0.88
4
ER stress as a sentinel mechanism for ER Ca
PMID: 39471738
Cell Calcium · 2024
0.80
5
GRP78 in lung cancer.
PMID: 33743739
J Transl Med · 2021
0.80