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50 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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ITGAV
integrin subunit alpha V
Chromosome 2 · 2q32.1
NCBI Gene: 3685Ensembl: ENSG00000138448.14HGNC: HGNC:6150UniProt: L7RXH0
698PubMed Papers
20Diseases
9Drugs
5Pathogenic Variants
FUNCTIONAL ROLE
Hub GeneReceptor
RESEARCH IMPACT
Highly StudiedTrending
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
extracellular exosomecalcium ion transmembrane transportprotease bindingpositive regulation of intracellular signal transductionneurodegenerative diseaseangina pectorismyocardial infarctionintermediate coronary syndrome
✦AI Summary

ITGAV encodes integrin alpha V, a cell adhesion molecule that functions as part of heterodimeric integrin complexes (αVβ3, αVβ5) mediating cell-extracellular matrix interactions and signaling 1. Mechanistically, ITGAV-containing integrins activate TGF-β1 signaling through latent TGF-β1 binding and activation 2, regulate immune cell communication via ligand-receptor partnerships 3, and promote epithelial-mesenchymal transition through POSTN-ITGAV/ITGB5 axis activation of PI3K/AKT/β-catenin pathways 4. Loss-of-function ITGAV variants cause a previously unreported human disease characterized by brain abnormalities, immune dysregulation, inflammatory bowel disease, and developmental defects through disrupted TGF-β and αVβ3-regulated immune signaling 1. ITGAV shows clinical significance as a Parkinson's disease biomarker, with decreased plasma levels consistently associated with disease risk (hazard ratio: 0.11-0.57) in large prospective cohorts 5. Additionally, ITGAV plays pathogenic roles in cancer progression and fibrotic diseases; elevated SPP1-ITGAV signaling promotes pancreatic and pituitary tumor invasion 46, while endothelial ITGAV dysregulation drives thoracic aortic dissection through focal adhesion disruption 7. These findings position ITGAV as a therapeutic target across multiple diseases.

Sources cited
1
ITGAV encodes integrin alpha V, a cell adhesion molecule that functions as part of heterodimeric integrin complexes (αVβ3, αVβ5) mediating cell-extracellular matrix interactions and signaling .
PMID: 39526957
2
Mechanistically, ITGAV-containing integrins activate TGF-β1 signaling through latent TGF-β1 binding and activation , regulate immune cell communication via ligand-receptor partnerships , and promote epithelial-mesenchymal transition through POSTN-ITGAV/ITGB5 axis activation of PI3K/AKT/β-catenin pathways .
PMID: 38239077
3
Mechanistically, ITGAV-containing integrins activate TGF-β1 signaling through latent TGF-β1 binding and activation , regulate immune cell communication via ligand-receptor partnerships , and promote epithelial-mesenchymal transition through POSTN-ITGAV/ITGB5 axis activation of PI3K/AKT/β-catenin pathways .
PMID: 37269061
4
Mechanistically, ITGAV-containing integrins activate TGF-β1 signaling through latent TGF-β1 binding and activation , regulate immune cell communication via ligand-receptor partnerships , and promote epithelial-mesenchymal transition through POSTN-ITGAV/ITGB5 axis activation of PI3K/AKT/β-catenin pathways .
PMID: 40520021
5
ITGAV shows clinical significance as a Parkinson's disease biomarker, with decreased plasma levels consistently associated with disease risk (hazard ratio: 0.11-0.57) in large prospective cohorts .
PMID: 39979637
6
Additionally, ITGAV plays pathogenic roles in cancer progression and fibrotic diseases; elevated SPP1-ITGAV signaling promotes pancreatic and pituitary tumor invasion , , while endothelial ITGAV dysregulation drives thoracic aortic dissection through focal adhesion disruption .
PMID: 40171827
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.42Moderate
angina pectorisOpen Targets
0.39Weak
myocardial infarctionOpen Targets
0.38Weak
intermediate coronary syndromeOpen Targets
0.37Weak
Recurrent thrombophlebitisOpen Targets
0.37Weak
inflammatory bowel diseaseOpen Targets
0.35Weak
strokeOpen Targets
0.32Weak
glioblastoma multiformeOpen Targets
0.30Weak
rheumatoid arthritisOpen Targets
0.30Weak
handednessOpen Targets
0.29Weak
acute myocardial infarctionOpen Targets
0.29Weak
gastric adenocarcinomaOpen Targets
0.28Weak
ST Elevation Myocardial InfarctionOpen Targets
0.26Weak
urinary bladder carcinomaOpen Targets
0.25Weak
pancreatic carcinomaOpen Targets
0.23Weak
gastric carcinomaOpen Targets
0.23Weak
melanomaOpen Targets
0.21Weak
esophageal squamous cell carcinomaOpen Targets
0.21Weak
non-small cell lung carcinomaOpen Targets
0.21Weak
colorectal carcinomaOpen Targets
0.21Weak
Pathogenic Variants5
NM_002210.5(ITGAV):c.903+1G>CLikely pathogenic
Susceptibility to severe COVID-19
★☆☆☆2024
NM_002210.5(ITGAV):c.432G>C (p.Trp144Cys)Pathogenic
ITGAV deficiency|Immune dysregulation, neurodevelopmental defects, and colitis
★☆☆☆2023→ Residue 144
NM_002210.5(ITGAV):c.1136A>T (p.Asp379Val)Pathogenic
ITGAV deficiency|Immune dysregulation, neurodevelopmental defects, and colitis
★☆☆☆2023→ Residue 379
NM_002210.5(ITGAV):c.1564+3_1564+6delPathogenic
ITGAV deficiency|Immune dysregulation, neurodevelopmental defects, and colitis
☆☆☆☆2025
NM_002210.5(ITGAV):c.2247-1G>APathogenic
ITGAV deficiency|Immune dysregulation, neurodevelopmental defects, and colitis
☆☆☆☆2025
View on ClinVar ↗
Drug Targets9
ABCIXIMABApproved
Integrin alpha-IIb/beta-3 inhibitor
intermediate coronary syndrome
ABITUZUMABPhase II
Integrin alpha-V/beta-5 inhibitor
colorectal cancer
ATN-161Phase II
Integrin alpha-5/beta-1 antagonist
renal cell carcinoma
CILENGITIDEPhase III
Integrin alpha-V/beta-3 antagonist
rheumatoid arthritis
ETARACIZUMABPhase II
Integrin alpha-V/beta-3 antagonist
IMGN-388Phase I
Vitronectin receptor alpha binding agent
INTETUMUMABPhase II
Integrin alpha-V/beta-3 antagonist
prostate cancer
RG-7594Phase I
Integrin alpha-V/beta-1 binding agent
STX-100Phase II
Integrin alpha-V/beta-6 inhibitor
idiopathic pulmonary fibrosis
Related Genes
CHADProtein interaction100%COL1A1Protein interaction100%COL6A5Protein interaction100%FN1Protein interaction99%TGFB3Protein interaction99%DMP1Protein interaction98%
Tissue Expression6 tissues
Heart
100%
Brain
37%
Ovary
28%
Lung
19%
Liver
9%
Bone Marrow
9%
Gene Interaction Network
Click a node to explore
ITGAVCHADCOL1A1COL6A5FN1TGFB3DMP1
PROTEIN STRUCTURE
Preparing viewer…
PDB9CZD · 2.23 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.81LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.63 [0.50–0.81]
RankingsWhere ITGAV stands among ~20K protein-coding genes
  • #308of 20,598
    Most Researched698 · top 5%
  • #728of 1,025
    FDA-Approved Drug Targets1
  • #3,456of 5,498
    Most Pathogenic Variants5
  • #6,749of 17,882
    Most Constrained (LOEUF)0.81
Genes detectedITGAV
Sources retrieved50 papers
Response time—
📄 Sources
50▼
1
Large-scale proteomic analyses of incident Parkinson's disease reveal new pathophysiological insights and potential biomarkers.
PMID: 39979637
Nat Aging · 2025
1.00
2
Human ITGAV variants are associated with immune dysregulation, brain abnormalities, and colitis.
PMID: 39526957
J Exp Med · 2024
0.90
3
Mechanisms of immune escape and extramedullary tropism in leukemia cutis.
PMID: 41026928
Blood · 2026
0.82
4
Integrative Single-Cell and Spatial Transcriptomics Analysis Reveals ECM-remodeling Cancer-associated Fibroblast-Derived POSTN as a Key Mediator in Pancreatic Ductal Adenocarcinoma Progression.
PMID: 40520021
Int J Biol Sci · 2025
0.80
5
Identifying novel drug targets for calcific aortic valve disease through Mendelian randomization.
PMID: 39922081
Atherosclerosis · 2025
0.80