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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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LPAR3
lysophosphatidic acid receptor 3
Chromosome 1 · 1p22.3
NCBI Gene: 23566Ensembl: ENSG00000171517.7HGNC: HGNC:14298UniProt: Q9UBY5
68PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingplasma membraneadenylate cyclase-activating G protein-coupled receptor signaling pathwaycytoplasmspermatoceletesticular diseaseleg injurybiliary tract disease
✦AI Summary

LPAR3 (lysophosphatidic acid receptor 3) is a G protein-coupled receptor that binds lysophosphatidic acid (LPA) and mediates diverse cellular signaling pathways through Gi/Go and Gq protein coupling 1. The receptor activates calcium signaling via the Gq/PLC pathway and regulates chloride transport through calcium-activated chloride channels in ocular surface epithelial cells 1. LPAR3 plays significant roles in cancer progression, promoting epithelial-mesenchymal transition and angiogenesis in nasopharyngeal carcinoma in response to matrix stiffness 2, and enhancing proliferation in malignant peripheral nerve sheath tumors while LPAR1 mediates migration 3. In liver disease, TEAD4-mediated upregulation of LPAR3 promotes hepatic stellate cell activation and fibrosis through p38 MAPK and PI3K/AKT signaling pathways 4. Therapeutically, LPAR3 shows protective effects in knee osteoarthritis, where lipoxin A4 activates the ESR2/LPAR3/Nrf2 axis to inhibit ferroptosis in fibroblast-like synoviocytes 5. The receptor is aberrantly expressed in various cancers including osteosarcoma, where it is regulated by ceRNA networks 6, and oral squamous cell carcinoma via circular RNA mechanisms 7. LPAR3 also contributes to macrophage polarization and anti-tumor immune responses in colorectal cancer 8.

Sources cited
1
LPAR3 is a G protein-coupled receptor that activates calcium signaling via Gq/PLC pathway and regulates chloride transport
PMID: 40112945
2
LPAR3 promotes nasopharyngeal carcinoma metastasis through epithelial-mesenchymal transition and angiogenesis in response to matrix stiffness
PMID: 40049264
3
LPAR3 enhances proliferation in malignant peripheral nerve sheath tumors while LPAR1 mediates migration
PMID: 36416236
4
TEAD4-mediated LPAR3 upregulation promotes hepatic stellate cell activation through p38 MAPK and PI3K/AKT signaling
PMID: 40591004
5
LPAR3 shows protective effects in knee osteoarthritis through the ESR2/LPAR3/Nrf2 axis inhibiting ferroptosis
PMID: 38754271
6
LPAR3 is regulated by ceRNA networks in osteosarcoma
PMID: 37727685
7
LPAR3 is involved in oral squamous cell carcinoma progression via circular RNA mechanisms
PMID: 34922206
8
LPAR3 contributes to macrophage polarization and anti-tumor immune responses in colorectal cancer
PMID: 32296017
Disease Associationsⓘ20
spermatoceleOpen Targets
0.33Weak
testicular diseaseOpen Targets
0.33Weak
leg injuryOpen Targets
0.31Weak
biliary tract diseaseOpen Targets
0.28Weak
pathological myopiaOpen Targets
0.20Weak
endometriosisOpen Targets
0.19Weak
chronic kidney diseaseOpen Targets
0.19Weak
female infertilityOpen Targets
0.18Weak
cancerOpen Targets
0.12Weak
neoplasmOpen Targets
0.11Weak
breast cancerOpen Targets
0.10Suggestive
lung adenocarcinomaOpen Targets
0.09Suggestive
hepatocellular carcinomaOpen Targets
0.09Suggestive
Alzheimer diseaseOpen Targets
0.09Suggestive
acute myeloid leukemiaOpen Targets
0.09Suggestive
triple-negative breast cancerOpen Targets
0.08Suggestive
psychiatric disorderOpen Targets
0.08Suggestive
SepsisOpen Targets
0.08Suggestive
Bartsocas-Papas syndrome 1Open Targets
0.07Suggestive
major depressive disorderOpen Targets
0.07Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
GNASProtein interaction98%AGTProtein interaction98%CHRM1Protein interaction98%GNAQProtein interaction98%PLA1AProtein interaction92%AVPProtein interaction91%
Tissue Expression6 tissues
Heart
100%
Brain
16%
Ovary
15%
Lung
9%
Bone Marrow
4%
Liver
1%
Gene Interaction Network
Click a node to explore
LPAR3GNASAGTCHRM1GNAQPLA1AAVP
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q9UBY5
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.62LoF Tolerant
pLIⓘ
0.78Intermediate
Observed/Expected LoF0.33 [0.19–0.62]
RankingsWhere LPAR3 stands among ~20K protein-coding genes
  • #6,912of 20,598
    Most Researched68
  • #4,372of 17,882
    Most Constrained (LOEUF)0.62 · top quartile
Genes detectedLPAR3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Lipoxin A
PMID: 38754271
Redox Biol · 2024
1.00
2
LPAR3 and COL8A1, as matrix stiffness-related biomarkers, promote nasopharyngeal carcinoma metastasis by triggering EMT and angiogenesis.
PMID: 40049264
Cell Signal · 2025
0.90
3
TEAD4-mediated upregulation of LPAR3 augments hepatic stellate cell activation in portal hypertension.
PMID: 40591004
Cell Biol Toxicol · 2025
0.80
4
Lysophosphatidic acid receptor 3 (LPAR3) regulates ocular surface chloride transport via calcium signaling.
PMID: 40112945
Exp Eye Res · 2025
0.70
5
The Agpat4/LPA axis in colorectal cancer cells regulates antitumor responses via p38/p65 signaling in macrophages.
PMID: 32296017
Signal Transduct Target Ther · 2020
0.60