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25 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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MAP2K6
mitogen-activated protein kinase kinase 6
Chromosome 17 · 17q24.3
NCBI Gene: 5608Ensembl: ENSG00000108984.17HGNC: HGNC:6846UniProt: A8K3Y2
159PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
KinaseTranscription Factor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
MAP kinase kinase activityprotein kinase bindingcytosolnucleoplasmneurodegenerative diseaseosteoarthritis, hiposteoarthritis, kneeAbnormality of the skeletal system
✦AI Summary

MAP2K6 (mitogen-activated protein kinase kinase 6) is a dual-specificity protein kinase that serves as an essential component of the p38 MAPK signaling cascade, catalyzing phosphorylation of p38 MAPK family members (MAPK11-14) in response to cellular stresses and cytokines. MAP2K6 plays a major role in TNF-induced p38 MAPK activation and mediates stress responses through downstream transcription factors ATF2 and ELK1, as well as STAT4 activation by IL-12. 1 Mechanistically, MAP2K6 integrates multiple signaling inputs: mTORC1 increases MAP2K6 protein synthesis to drive intestinal stem cell aging via p38 MAPK-p53 pathway activation 1, while stress-activated kinases MKK3 and MKK6 activate the Mirk checkpoint kinase during cellular stress responses 2. The kinase is dysregulated in multiple malignancies, where it promotes cancer cell proliferation and radioresistance through LIFR/p70S6K signaling in nasopharyngeal carcinoma 3 and enhances paclitaxel sensitivity via autophagy induction in ovarian cancer 4. Clinically, MAP2K6 represents a therapeutic target in polycystic ovary syndrome and gastric cancer, where downregulation of regulatory microRNAs (miR-375, miR-324-3p, miR-1298-5p) leads to MAP2K6 overexpression and enhanced granulosa cell/cancer cell proliferation 567. In hepatocellular carcinoma, APEX1-mediated upregulation of MAP2K6 promotes malignant properties 8, suggesting MAP2K6 as a prognostic biomarker and therapeutic target across multiple cancer types.

Sources cited
1
Mechanistically, MAP2K6 integrates multiple signaling inputs: mTORC1 increases MAP2K6 protein synthesis to drive intestinal stem cell aging via p38 MAPK-p53 pathway activation , while stress-activated kinases MKK3 and MKK6 activate the Mirk checkpoint kinase during cellular stress responses .
PMID: 31896747
2
Mechanistically, MAP2K6 integrates multiple signaling inputs: mTORC1 increases MAP2K6 protein synthesis to drive intestinal stem cell aging via p38 MAPK-p53 pathway activation , while stress-activated kinases MKK3 and MKK6 activate the Mirk checkpoint kinase during cellular stress responses .
PMID: 17583556
3
The kinase is dysregulated in multiple malignancies, where it promotes cancer cell proliferation and radioresistance through LIFR/p70S6K signaling in nasopharyngeal carcinoma and enhances paclitaxel sensitivity via autophagy induction in ovarian cancer .
PMID: 30245131
4
The kinase is dysregulated in multiple malignancies, where it promotes cancer cell proliferation and radioresistance through LIFR/p70S6K signaling in nasopharyngeal carcinoma and enhances paclitaxel sensitivity via autophagy induction in ovarian cancer .
PMID: 28604448
5
In hepatocellular carcinoma, APEX1-mediated upregulation of MAP2K6 promotes malignant properties , suggesting MAP2K6 as a prognostic biomarker and therapeutic target across multiple cancer types.
PMID: 36205565
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.50Moderate
osteoarthritis, hipOpen Targets
0.47Moderate
osteoarthritis, kneeOpen Targets
0.46Moderate
Abnormality of the skeletal systemOpen Targets
0.44Moderate
osteoarthritisOpen Targets
0.43Moderate
total hip arthroplastyOpen Targets
0.40Weak
medical procedureOpen Targets
0.37Weak
anthrax infectionOpen Targets
0.37Weak
neuroinflammatory disorderOpen Targets
0.37Weak
eye colorOpen Targets
0.32Weak
total knee arthroplastyOpen Targets
0.30Weak
glaucomaOpen Targets
0.29Weak
Non-Neoplastic Bile Duct DisorderOpen Targets
0.29Weak
total joint arthroplastyOpen Targets
0.27Weak
retinal degenerationOpen Targets
0.24Weak
ulcerative colitisOpen Targets
0.19Weak
liver diseaseOpen Targets
0.17Weak
knee fractureOpen Targets
0.11Weak
heart failureOpen Targets
0.11Weak
congestive heart failureOpen Targets
0.11Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
TAB3Protein interaction100%TAB2Protein interaction100%TRAF6Protein interaction100%MAP3K3Protein interaction99%MAP3K4Protein interaction99%RIPK1Protein interaction98%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
72%
Heart
43%
Lung
28%
Liver
27%
Ovary
18%
Gene Interaction Network
Click a node to explore
MAP2K6TAB3TAB2TRAF6MAP3K3MAP3K4RIPK1
PROTEIN STRUCTURE
Preparing viewer…
PDB2Y8O · 1.95 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.64LoF Tolerant
pLIⓘ
0.58Intermediate
Observed/Expected LoF0.38 [0.23–0.64]
RankingsWhere MAP2K6 stands among ~20K protein-coding genes
  • #2,831of 20,598
    Most Researched159 · top quartile
  • #4,534of 17,882
    Most Constrained (LOEUF)0.64
Genes detectedMAP2K6
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
Gut stem cell aging is driven by mTORC1 via a p38 MAPK-p53 pathway.
PMID: 31896747
Nat Commun · 2020
1.00
2
Mirk/Dyrk1B in cancer.
PMID: 17583556
J Cell Biochem · 2007
0.90
3
CircASPH promotes KGN cells proliferation through miR-375/MAP2K6 axis in Polycystic Ovary Syndrome.
PMID: 33372369
J Cell Mol Med · 2022
0.80
4
PMID: 36205565
Aging (Albany NY) · 2022
0.70
5
Nuclear translocation of CDK5RAP3 regulated by NXF3 promotes the progression of gastric cancer.
PMID: 40032765
Cell Mol Life Sci · 2025
0.64