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GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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MAPK10
mitogen-activated protein kinase 10
Chromosome 4 · 4q21.3
NCBI Gene: 5602Ensembl: ENSG00000109339.24HGNC: HGNC:6872UniProt: A0A286YEQ0
126PubMed Papers
20Diseases
5Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
nucleoplasmprotein phosphorylationprotein bindingJUN kinase activitygouthearing lossparasitic infectioncolor vision disorder
✦AI Summary

MAPK10 (also known as JNK3) is a serine/threonine protein kinase that functions as a critical component of the stress-activated protein kinase/c-Jun N-terminal kinase signaling pathway 1. Upon activation by upstream dual specificity kinases MAP2K4/MKK4 and MAP2K7/MKK7, MAPK10 phosphorylates transcription factors including components of AP-1 such as JUN and ATF2, thereby regulating AP-1 transcriptional activity. The kinase plays essential roles in neuronal processes including proliferation, differentiation, migration, and programmed cell death, and phosphorylates neuronal substrates like STMN2 and the amyloid-beta precursor protein APP during neuronal differentiation. In metabolic regulation, MAPK10 exhibits opposing functions to JNK1 in hypothalamic AgRP neurons, where its deletion impairs insulin and leptin signaling and promotes feeding behavior 1. MAPK10 demonstrates significant disease relevance across multiple cancers. In neuroblastoma, its upregulation contributes to disease development 2. In non-small cell lung cancer (NSCLC), MAPK10 acts as a tumor suppressor when activated, as HACD3 promotes malignant progression by directly interacting with and suppressing the MKK7/MAPK10 signaling axis 3. Additionally, MAPK10-mediated mitochondrial autophagy represents a therapeutic target, as demonstrated by traditional Chinese medicine treatments that attenuate chr4 atrophic gastritis progression through MAPK10 modulation 4. The kinase also participates in inflammatory responses and cytokine storms in various pathological conditions 5.

Sources cited
1
MAPK10 is a stress-activated kinase in the JNK pathway with opposing roles to JNK1 in hypothalamic neurons
PMID: 33200240
2
MAPK10 upregulation contributes to neuroblastoma development
PMID: 31432180
3
HACD3 promotes NSCLC progression by suppressing MKK7/MAPK10 signaling through direct interaction
PMID: 40817125
4
MAPK10-mediated mitochondrial autophagy is involved in chronic atrophic gastritis progression
PMID: 40103313
5
MAPK10 expression is increased in cytokine storm-related inflammatory conditions
PMID: 39462545
Disease Associationsⓘ20
goutOpen Targets
0.52Moderate
hearing lossOpen Targets
0.33Weak
parasitic infectionOpen Targets
0.32Weak
color vision disorderOpen Targets
0.32Weak
mental or behavioural disorderOpen Targets
0.31Weak
conduction system disorderOpen Targets
0.29Weak
osteoarthritisOpen Targets
0.28Weak
nervous system diseaseOpen Targets
0.26Weak
Lennox-Gastaut syndromeOpen Targets
0.25Weak
Epileptic encephalopathyOpen Targets
0.22Weak
HypercholesterolemiaOpen Targets
0.19Weak
Back painOpen Targets
0.17Weak
Alzheimer diseaseOpen Targets
0.15Weak
prostate cancerOpen Targets
0.13Weak
hypothyroidismOpen Targets
0.12Weak
Familial prostate cancerOpen Targets
0.11Weak
neoplasmOpen Targets
0.10Weak
hepatocellular carcinomaOpen Targets
0.10Suggestive
Parkinson diseaseOpen Targets
0.10Suggestive
gastric cancerOpen Targets
0.08Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets5
BENTAMAPIMODPhase II
c-Jun N-terminal kinase, JNK inhibitor
endometriosis
BRIMAPITIDEPhase I
c-Jun N-terminal kinase 3 inhibitor
inflammation
BRIMAPITIDE, C-TERMINAL ACIDPhase III
c-Jun N-terminal kinase 3 inhibitor
nervous system disease
CC-401Phase II
c-Jun N-terminal kinase 1 inhibitor
TANZISERTIBPhase II
c-Jun N-terminal kinase 3 inhibitor
discoid lupus erythematosus
Related Genes
MAPK14Protein interaction100%MAPK3Protein interaction94%MAPK12Protein interaction92%MAPK1Protein interaction91%DUSP16Protein interaction89%IP6K2Protein interaction77%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
33%
Ovary
32%
Heart
21%
Lung
6%
Liver
4%
Gene Interaction Network
Click a node to explore
MAPK10MAPK14MAPK3MAPK12MAPK1DUSP16IP6K2
PROTEIN STRUCTURE
Preparing viewer…
PDB3OY1 · 1.70 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.54Moderately Constrained
pLIⓘ
0.91Intolerant
Observed/Expected LoF0.35 [0.23–0.54]
RankingsWhere MAPK10 stands among ~20K protein-coding genes
  • #3,733of 20,598
    Most Researched126 · top quartile
  • #3,412of 17,882
    Most Constrained (LOEUF)0.54 · top quartile
Genes detectedMAPK10
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Berberine modulates ovarian cancer autophagy and glycolysis through the LINC01123/P65/MAPK10 signaling axis.
PMID: 39395322
Phytomedicine · 2024
1.00
2
Unveiling ac4C modification pattern: a prospective target for improving the response to immunotherapeutic strategies in melanoma.
PMID: 40050821
J Transl Med · 2025
0.90
3
Brain JNK and metabolic disease.
PMID: 33200240
Diabetologia · 2021
0.80
4
Transcriptome analysis of the cytokine storm-related genes among the subtypes of idiopathic multicentric Castleman disease.
PMID: 39462545
J Clin Exp Hematop · 2024
0.70
5
Colchicine alleviates atherosclerosis combined with diabetes mellitus by targeting PIM2 and regulating the NF-κB signaling pathway.
PMID: 40865347
Phytomedicine · 2025
0.60