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GeneE
50 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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MAPK8
mitogen-activated protein kinase 8
Chromosome 10 · 10q11.22
NCBI Gene: 5599Ensembl: ENSG00000107643.18HGNC: HGNC:6881UniProt: A1L4K2
1,055PubMed Papers
20Diseases
3Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Hub GeneKinase
RESEARCH IMPACT
Highly StudiedTrending
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
histone deacetylase regulator activityresponse to UVnegative regulation of apoptotic processcellular response to lipopolysaccharidecancerneurodegenerative diseasepoisoningmuscle cramp
✦AI Summary

MAPK8 (mitogen-activated protein kinase 8), also known as JNK1, is a serine/threonine kinase that functions as a key signaling hub in cellular stress responses and inflammatory pathways. 1 MAPK8 displays multiple isoforms with distinct substrate binding patterns, where the beta-1 isoform preferentially binds c-Jun, while alpha and other isoforms show lower affinity for both c-Jun and ATF2 transcription factors, though all isoforms achieve similar phosphorylation efficiency. 2 In neuropathic pain, MAPK8 phosphorylation (p-MAPK8/JNK) mediates neuroinflammatory responses by promoting TRAF6 binding to ubiquitinated proteins and activating NF-κB signaling, suggesting autophagy-mediated regulation of MAPK8 activity modulates pain maintenance. 3 MAPK8 functions within the MAPK8/FOXO3 signaling pathway to regulate autophagy and mitophagy in bone cells, contributing to homeostasis in osteoblasts and osteoclasts. 4 In polycystic ovary syndrome, MAPK8/JNK participates in autophagy-related pathophysiology affecting ovarian follicular development. 1 Network analysis identifies MAPK8 as a central hub in rheumatoid arthritis pathogenesis, where naringin-mediated inhibition of MAPK8 phosphorylation suppresses inflammatory cytokine production and promotes fibroblast-like synoviocyte apoptosis. These findings establish MAPK8 as a critical regulator of inflammation, autophagy, and cellular stress responses across multiple disease contexts.

Sources cited
1
MAPK8 is a central hub protein in rheumatoid arthritis pathogenesis with high network centrality; MAPK8 phosphorylation inhibition reduces inflammation
PMID: 34054546
2
MAPK8 phosphorylation (p-MAPK8/JNK) mediates neuroinflammatory responses in neuropathic pain by promoting TRAF6 binding and NFKB activation
PMID: 33834930
3
MAPK8/FOXO3 signaling pathway regulates autophagy and mitophagy in bone cells (osteoblasts and osteoclasts)
PMID: 32792864
4
MAPK8/JNK is involved in autophagy-related pathophysiology in polycystic ovary syndrome
PMID: 34161185
⚠Limited data available — This gene has 4 indexed publications. Summary and analysis may be incomplete.
Disease Associationsⓘ20
cancerOpen Targets
0.57Moderate
neurodegenerative diseaseOpen Targets
0.38Weak
muscle crampOpen Targets
0.31Weak
poisoningOpen Targets
0.31Weak
response to xenobiotic stimulusOpen Targets
0.30Weak
neuroinflammatory disorderOpen Targets
0.26Weak
response to antihypertensive drugOpen Targets
0.23Weak
diabetes mellitusOpen Targets
0.20Weak
type 2 diabetes mellitusOpen Targets
0.19Weak
neoplasmOpen Targets
0.12Weak
breast cancerOpen Targets
0.11Weak
hepatocellular carcinomaOpen Targets
0.11Weak
cystOpen Targets
0.11Weak
obesityOpen Targets
0.11Weak
Insulin resistanceOpen Targets
0.10Weak
gastric cancerOpen Targets
0.10Weak
Pallister-Hall syndromeOpen Targets
0.10Suggestive
acute respiratory distress syndromeOpen Targets
0.10Suggestive
myopiaOpen Targets
0.10Suggestive
melanomaOpen Targets
0.10Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets3
BENTAMAPIMODPhase II
c-Jun N-terminal kinase, JNK inhibitor
endometriosis
CC-401Phase II
c-Jun N-terminal kinase 1 inhibitor
TANZISERTIBPhase II
c-Jun N-terminal kinase 3 inhibitor
discoid lupus erythematosus
Related Genes
APBB1Protein interaction100%KLC1Protein interaction100%RELAProtein interaction100%MAP2K3Protein interaction100%MAPK8IP1Protein interaction100%KLC2Protein interaction100%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
76%
Ovary
68%
Liver
57%
Heart
47%
Lung
41%
Gene Interaction Network
Click a node to explore
MAPK8APBB1KLC1RELAMAP2K3MAPK8IP1KLC2
PROTEIN STRUCTURE
Preparing viewer…
PDB2XRW · 1.33 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.53Moderately Constrained
pLIⓘ
0.95Intolerant
Observed/Expected LoF0.30 [0.18–0.53]
RankingsWhere MAPK8 stands among ~20K protein-coding genes
  • #146of 20,598
    Most Researched1,055 · top 1%
  • #3,335of 17,882
    Most Constrained (LOEUF)0.53 · top quartile
Genes detectedMAPK8
Sources retrieved50 papers
Response time—
📄 Sources
50▼
1
Autophagy in ovary and polycystic ovary syndrome: role, dispute and future perspective.
PMID: 34161185
Autophagy · 2021
1.00
2
The Role of Autophagy and Mitophagy in Bone Metabolic Disorders.
PMID: 32792864
Int J Biol Sci · 2020
0.90
3
MAPK8 and HDAC6: potential biomarkers related to autophagy in diabetic retinopathy based on bioinformatics analysis.
PMID: 40469433
Front Endocrinol (Lausanne) · 2025
0.82
4
AKT1 and MAPK8: New Targets for Gestational Diabetes Mellitus?
PMID: 39177257
Fetal Pediatr Pathol · 2024
0.80
5
Autophagy in the physiological endometrium and cancer.
PMID: 32401642
Autophagy · 2021
0.80