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GeneE
2 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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OPRPN
opiorphin prepropeptide
Chromosome 4 · 4q13.3
NCBI Gene: 58503Ensembl: ENSG00000171199.11HGNC: HGNC:17279UniProt: Q99935
27PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
endopeptidase inhibitor activitypeptidase inhibitor activityregulation of sensory perception of painextracellular regionneoplasmhepatocellular carcinomaglioblastoma multiformebreast carcinoma
✦AI Summary

OPRPN encodes opiorphin prepropeptide, an endogenous inhibitor of neprilysin and aminopeptidase N involved in neuropeptide degradation. UniProt annotations document that opiorphin inhibits breakdown of substance P, enkephalins, and bradykinin with IC50 values of 29-65 μM, and demonstrates potent analgesic effects in rats. GO terms indicate peptidase inhibitor activity and roles in pain perception regulation. Based on limited published evidence, OPRPN expression is induced by ionizing radiation in head and neck squamous cell carcinoma cells 1, where elevated OPRPN may associate with improved clinical outcomes, suggesting potential protective functions in radiotherapy response 1. OPRPN is expressed in salivary glands, though specific functional roles in salivary biology remain understudied.

Sources cited
1
OPRPN expression is induced by fractionated irradiation in head and neck squamous cell carcinoma and may exert protective function in radiotherapy outcomes
PMID: 35856431
2
OPRPN is expressed in salivary glands and may be altered in disease states such as diabetes mellitus
PMID: 19659899
⚠Limited data available — This gene has 2 indexed publications. Summary and analysis may be incomplete.
Disease Associationsⓘ20
neoplasmOpen Targets
0.09Suggestive
hepatocellular carcinomaOpen Targets
0.08Suggestive
glioblastoma multiformeOpen Targets
0.08Suggestive
breast carcinomaOpen Targets
0.05Suggestive
gliomaOpen Targets
0.04Suggestive
lung cancerOpen Targets
0.04Suggestive
colitisOpen Targets
0.03Suggestive
cancerOpen Targets
0.03Suggestive
diabetic nephropathyOpen Targets
0.03Suggestive
stage 5 chronic kidney diseaseOpen Targets
0.03Suggestive
acanthosis nigricansOpen Targets
0.03Suggestive
burning mouth syndromeOpen Targets
0.02Suggestive
AnxietyOpen Targets
0.02Suggestive
psoriasisOpen Targets
0.02Suggestive
PriapismOpen Targets
0.02Suggestive
depressive disorderOpen Targets
0.02Suggestive
mucous membrane pemphigoidOpen Targets
0.02Suggestive
geroderma osteodysplasticaOpen Targets
0.02Suggestive
albuminuriaOpen Targets
0.02Suggestive
colorectal carcinomaOpen Targets
0.02Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
SMR3BShared pathway100%SMR3AShared pathway100%PIRTShared pathway100%ZFHX2Shared pathway100%ANPEPProtein interaction89%PLGLB1Protein interaction86%
Tissue Expression6 tissues
Liver
100%
Brain
0%
Ovary
0%
Heart
0%
Lung
0%
Bone Marrow
0%
Gene Interaction Network
Click a node to explore
OPRPNSMR3BSMR3APIRTZFHX2ANPEPPLGLB1
PROTEIN STRUCTURE
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AlphaFoldAI-predicted · UniProt Q99935
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.65LoF Tolerant
pLIⓘ
0.44Tolerant
Observed/Expected LoF0.00 [0.00–1.65]
RankingsWhere OPRPN stands among ~20K protein-coding genes
  • #12,629of 20,598
    Most Researched27
  • #15,907of 17,882
    Most Constrained (LOEUF)1.65
Genes detectedOPRPN
Sources retrieved2 papers
Response time—
📄 Sources
2
1
Conjoint analysis of OPRPN and SMR3A protein expression as potential predictive biomarkers for head and neck squamous cell carcinoma after radiotherapy.
PMID: 35856431
Oncol Rep · 2022
1.00
2
Protein expression in salivary glands of rats with streptozotocin diabetes.
PMID: 19659899
Int J Exp Pathol · 2009
0.50