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GeneE
26 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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PIM1
Pim-1 proto-oncogene, serine/threonine kinase
Chromosome 6 · 6p21.2
NCBI Gene: 5292Ensembl: ENSG00000137193.15HGNC: HGNC:8986UniProt: P11309
301PubMed Papers
20Diseases
3Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
KinaseOncogene
RESEARCH IMPACT
Trending
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
positive regulation of cardioblast proliferationnucleusnucleoplasmnucleolusdiffuse large B-cell lymphomaneurodegenerative diseaseprostate carcinomaCentral Nervous System Lymphoma
✦AI Summary

PIM1 is a serine/threonine kinase proto-oncogene that functions as a key regulator of cell survival and proliferation, conferring selective advantages in tumorigenesis 1. The kinase exerts oncogenic activity through multiple interconnected mechanisms: phosphorylation and stabilization of MYC to enhance its transcriptional activity, inhibition of pro-apoptotic proteins (BAD, MAP3K5, FOXO3) to suppress apoptosis, and promotion of cell cycle progression via phosphorylation of CDC25A/C and CDKN1A/B 23. Beyond canonical oncogenic pathways, PIM1 acts as a positive regulator of mTORC1 signaling through DEPDC5 phosphorylation and negatively regulates innate immunity by inactivating GBP1, preventing unwanted immune damage 45. Recent evidence reveals PIM1's broader pathological significance: it promotes endothelial-to-mesenchymal transition via NDRG1 phosphorylation, contributing to atherosclerosis progression 6; drives myofibroblast ferroptosis resistance in skin fibrosis diseases 7; and regulates T helper cell differentiation through the AKT/FOXO1 pathway in autoimmune uveitis 8. PIM1 overexpression is implicated in both hematologic and solid malignancies, positioning it as an emerging therapeutic target 910. PIM1 inhibition demonstrates promise in suppressing cancer cell proliferation and modulating pathologic immune responses across multiple disease contexts.

Sources cited
1
PIM1 is a proto-oncogene providing selective advantage in tumorigenesis
PMID: 15528381
2
PIM1 regulates MYC stability, phosphorylates pro-apoptotic proteins, and modulates cell cycle regulators CDKN1A/B
PMID: 18593906
3
PIM1 phosphorylates MAP3K5 to inhibit apoptosis by reducing JNK/p38MAPK signaling and caspase-3 activation
PMID: 19749799
4
PIM1 acts as positive regulator of mTORC1 through DEPDC5 phosphorylation and inhibition
PMID: 31548394
5
PIM1 negatively regulates innate immunity by phosphorylating and sequestering GBP1
PMID: 37797010
6
PIM1 promotes endothelial-to-mesenchymal transition and atherosclerosis progression via NDRG1/PTBP1 pathway
PMID: 39744686
7
PIM1 is upregulated in skin fibrosis diseases and inhibition promotes ferroptosis in myofibroblasts
PMID: 40168881
8
PIM1 regulates Th17/Treg balance via AKT/FOXO1 pathway in autoimmune uveitis
PMID: 36195600
9
PIM1 is overexpressed in solid and hematologic malignancies and is a therapeutic target in cancer
PMID: 39487435
10
PIM1 plays prominent roles in immunoinflammatory diseases through phosphorylation of inflammatory substrates
PMID: 39372407
Disease Associationsⓘ20
diffuse large B-cell lymphomaOpen Targets
0.54Moderate
neurodegenerative diseaseOpen Targets
0.53Moderate
prostate carcinomaOpen Targets
0.51Moderate
Central Nervous System LymphomaOpen Targets
0.38Weak
diffuse large B-cell lymphoma of the central nervous systemOpen Targets
0.37Weak
lymphoid neoplasmOpen Targets
0.37Weak
Hodgkins lymphomaOpen Targets
0.37Weak
neoplasm of mature B-cellsOpen Targets
0.37Weak
multiple myelomaOpen Targets
0.35Weak
pulmonary arterial hypertensionOpen Targets
0.35Weak
Alzheimer diseaseOpen Targets
0.33Weak
lysosomal storage diseaseOpen Targets
0.32Weak
multiple sclerosisOpen Targets
0.32Weak
Parkinson diseaseOpen Targets
0.32Weak
acute myeloid leukemiaOpen Targets
0.31Weak
hepatocellular carcinomaOpen Targets
0.30Weak
esophageal squamous cell carcinomaOpen Targets
0.30Weak
chronic lymphocytic leukemiaOpen Targets
0.30Weak
urinary bladder carcinomaOpen Targets
0.30Weak
astrocytomaOpen Targets
0.30Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets3
AZD-1208Phase I
Serine/threonine-protein kinase PIM inhibitor
LGH-447Phase I/II
Serine/threonine-protein kinase PIM inhibitor
multiple myeloma
SGI-1776Phase I
Serine/threonine-protein kinase PIM inhibitor
non-Hodgkins lymphoma
Related Genes
STAT5BProtein interaction100%EDC3Protein interaction100%STAT5AProtein interaction100%DCP1AProtein interaction99%MYCProtein interaction99%SERPINA1Protein interaction91%
Tissue Expression6 tissues
Bone Marrow
100%
Lung
46%
Ovary
36%
Brain
30%
Liver
28%
Heart
8%
Gene Interaction Network
Click a node to explore
PIM1STAT5BEDC3STAT5ADCP1AMYCSERPINA1
PROTEIN STRUCTURE
Preparing viewer…
PDB3A99 · 1.60 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.44Moderately Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.25 [0.15–0.44]
RankingsWhere PIM1 stands among ~20K protein-coding genes
  • #1,160of 20,598
    Most Researched301 · top 10%
  • #2,391of 17,882
    Most Constrained (LOEUF)0.44 · top quartile
Genes detectedPIM1
Sources retrieved26 papers
Response time—
📄 Sources
26▼
1
PIM1 instigates endothelial-to-mesenchymal transition to aggravate atherosclerosis.
PMID: 39744686
Theranostics · 2025
1.00
2
Targeting PIM1 by Bruceine D attenuates skin fibrosis via myofibroblast ferroptosis.
PMID: 40168881
Redox Biol · 2025
0.90
3
Multicellular immune dynamics implicate PIM1 as a potential therapeutic target for uveitis.
PMID: 36195600
Nat Commun · 2022
0.80
4
The role of Pim-1 kinases in inflammatory signaling pathways.
PMID: 39079978
Inflamm Res · 2024
0.76
5
PIM1 drives lipid droplet accumulation to promote proliferation and survival in prostate cancer.
PMID: 38097734
Oncogene · 2024
0.72