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GeneE
25 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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PTGS1
prostaglandin-endoperoxide synthase 1
Chromosome 9 · 9q33.2
NCBI Gene: 5742Ensembl: ENSG00000095303.17HGNC: HGNC:9604UniProt: A0A087X296
284PubMed Papers
20Diseases
65Drugs
0Pathogenic Variants
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
prostaglandin-endoperoxide synthase activityprotein bindingcytoplasmextracellular exosomehemorrhagerheumatoid arthritisulcerative colitisosteoarthritis
✦AI Summary

PTGS1 (cyclooxygenase-1) is a dual cyclooxygenase/peroxidase enzyme that catalyzes the first committed step in prostanoid biosynthesis from arachidonic acid, converting it to prostaglandin H2 (PGH2), the precursor for all 2-series prostaglandins and thromboxanes [UniProt]. The enzyme abstracts hydrogen at carbon 13 of arachidonic acid and sequentially inserts two oxygen molecules to form the characteristic endoperoxide bridge, with peroxidase activity then reducing the intermediate to PGH2 [UniProt]. PTGS1 is constitutively expressed in the stomach and platelets, where it generates cytoprotective prostaglandins (particularly PGE2) and prothrombotic thromboxane A2, respectively [UniProt]. Clinically, PTGS1 is the primary target of nonsteroidal anti-inflammatory drugs (NSAIDs), whose inhibition contributes to gastrointestinal damage through multiple mechanisms including barrier dysfunction and increased intestinal permeability 1. PTGS1 polymorphisms influence individual responses to NSAID therapy and may modulate cancer risk, with specific variants showing altered metabolic activity and indomethacin sensitivity 23. Gene expression is dynamically regulated by nutritional factors (omega-3 supplementation) and signaling pathways implicated in cancer progression 45. PTGS1 expression occurs early in human embryonic development, suggesting roles in embryogenesis and implantation 6.

Sources cited
1
PTGS1 inhibition by NSAIDs contributes to gastrointestinal damage through COX-mediated and independent processes
PMID: 29221664
2
PTGS1 polymorphisms influence cancer risk association with NSAID use
PMID: 23967159
3
PTGS1 gene expression in PBMCs is regulated by omega-3 fatty acid supplementation and arachidonic acid levels
PMID: 26672987
4
PTGS1 is transcriptionally regulated by ZBTB46 and associated with neuroendocrine prostate cancer progression
PMID: 30312731
5
Multiple nonsynonymous PTGS1 polymorphisms significantly alter basal COX-1 metabolic activity and indomethacin sensitivity
PMID: 17301694
6
PTGS1 is expressed during early human preimplantation embryonic development
PMID: 12050227
Disease Associationsⓘ20
hemorrhageOpen Targets
0.63Moderate
rheumatoid arthritisOpen Targets
0.61Moderate
ulcerative colitisOpen Targets
0.61Moderate
osteoarthritisOpen Targets
0.61Moderate
migraine disorderOpen Targets
0.61Moderate
goutOpen Targets
0.61Moderate
PainOpen Targets
0.61Moderate
DysmenorrheaOpen Targets
0.61Moderate
HeadacheOpen Targets
0.61Moderate
ankylosing spondylitisOpen Targets
0.61Moderate
FeverOpen Targets
0.61Moderate
juvenile idiopathic arthritisOpen Targets
0.61Moderate
Nasal congestionOpen Targets
0.60Moderate
common coldOpen Targets
0.60Moderate
CoughOpen Targets
0.60Moderate
pharyngitisOpen Targets
0.60Moderate
rheumatic diseaseOpen Targets
0.60Moderate
toothacheOpen Targets
0.60Moderate
inflammationOpen Targets
0.60Moderate
arthritisOpen Targets
0.60Moderate
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets65
ACEMETACINApproved
Cyclooxygenase inhibitor
rheumatic disease
ACETAMINOPHENApproved
Cyclooxygenase inhibitor
Pain
ALCLOFENACApproved
Cyclooxygenase-1 inhibitor
rheumatoid arthritis
ALOXIPRINApproved
Cyclooxygenase inhibitor
Recurrent thrombophlebitis
ANTIPYRINEApproved
Cyclooxygenase-1 inhibitor
Fever
APAZONEApproved
Cyclooxygenase inhibitor
rheumatic disease
ASPIRINApproved
Cyclooxygenase inhibitor
arthritis
BALSALAZIDEApproved
Peroxisome proliferator-activated receptor gamma agonist
inflammatory bowel disease
BALSALAZIDE DISODIUMApproved
Peroxisome proliferator-activated receptor gamma agonist
ulcerative colitis
BENZYDAMINEApproved
Cyclooxygenase inhibitor
vaginal inflammation
BENZYDAMINE HYDROCHLORIDEPhase III
Cyclooxygenase inhibitor
medical procedure
BISMUTH SUBSALICYLATEApproved
Cyclooxygenase inhibitor
Nausea
BROMFENACApproved
Cyclooxygenase inhibitor
BROMFENAC SODIUMApproved
Cyclooxygenase inhibitor
inflammation
CLOMETACINUNKNOWN
Cyclooxygenase inhibitor
DEXIBUPROFENApproved
Cyclooxygenase inhibitor
ankylosing spondylitis
DEXKETOPROFENApproved
Cyclooxygenase inhibitor
rheumatic disease
DICLOFENACApproved
Cyclooxygenase inhibitor
rheumatoid arthritis
DICLOFENAC EPOLAMINEApproved
Cyclooxygenase inhibitor
sprain
DICLOFENAC ETALHYALURONATE SODIUMApproved
Cyclooxygenase inhibitor
DICLOFENAC POTASSIUMApproved
Cyclooxygenase inhibitor
DICLOFENAC SODIUMApproved
Cyclooxygenase inhibitor
osteoarthritis
DIFLUNISALApproved
Cyclooxygenase inhibitor
DIPYRONEApproved
Cyclooxygenase inhibitor
Fever
ESFLURBIPROFENApproved
Cyclooxygenase inhibitor
Pain
FENCLOFENACUNKNOWN
Cyclooxygenase inhibitor
FENOPROFENApproved
Cyclooxygenase inhibitor
rheumatoid arthritis
FENOPROFEN CALCIUMApproved
Cyclooxygenase inhibitor
rheumatoid arthritis
FLURBIPROFENApproved
Cyclooxygenase inhibitor
Miosis
GLAFENINEApproved
Cyclooxygenase inhibitor
Fever
IBUFENACUNKNOWN
Cyclooxygenase inhibitor
IBUPROFENApproved
Cyclooxygenase inhibitor
Dysmenorrhea
IBUPROFEN LYSINEApproved
Cyclooxygenase inhibitor
Patent ductus arteriosus
IBUPROFEN SODIUMPhase I
Cyclooxygenase inhibitor
INDOMETHACINApproved
Cyclooxygenase inhibitor
osteoarthritis
INDOPROFENApproved
Cyclooxygenase inhibitor
rheumatic disease
ISOXICAMUNKNOWN
Cyclooxygenase inhibitor
KETOPROFENApproved
Cyclooxygenase inhibitor
KETOROLACApproved
Cyclooxygenase inhibitor
KETOROLAC TROMETHAMINEApproved
Cyclooxygenase inhibitor
Pain
LORNOXICAMApproved
Cyclooxygenase inhibitor
migraine disorder
LOXOPROFENApproved
Cyclooxygenase inhibitor
inflammation
MECLOFENAMATE SODIUMApproved
Arachidonate 5-lipoxygenase inhibitor
juvenile idiopathic arthritis
MECLOFENAMIC ACIDApproved
Arachidonate 5-lipoxygenase inhibitor
ankylosing spondylitis
MEFENAMIC ACIDApproved
Cyclooxygenase inhibitor
Dysmenorrhea
MESALAMINEApproved
Arachidonate 5-lipoxygenase inhibitor
ulcerative colitis
METAMIZOLEPhase I
Cyclooxygenase inhibitor
NAPROXCINODApproved
Cyclooxygenase inhibitor
rheumatic disease
NAPROXENApproved
Cyclooxygenase inhibitor
arthritis
NAPROXEN ETEMESILPhase II/III
Cyclooxygenase inhibitor
ankylosing spondylitis
NAPROXEN SODIUMApproved
Cyclooxygenase inhibitor
osteoarthritis
NEPAFENACApproved
Cyclooxygenase inhibitor
inflammation
OLSALAZINEApproved
Peroxisome proliferator-activated receptor gamma agonist
ulcerative colitis
OLSALAZINE SODIUMApproved
Peroxisome proliferator-activated receptor gamma agonist
ulcerative colitis
OXAPROZINApproved
Cyclooxygenase inhibitor
OXYPHENBUTAZONEApproved
Cyclooxygenase inhibitor
arthritis
OXYPHENBUTAZONE ANHYDROUSUNKNOWN
Cyclooxygenase inhibitor
PHENYLBUTAZONEApproved
Cyclooxygenase inhibitor
Chronic pain
PIROXICAMApproved
Cyclooxygenase inhibitor
rheumatoid arthritis
PIRPROFENApproved
Cyclooxygenase inhibitor
Dysmenorrhea
SULFASALAZINEApproved
Arachidonate 5-lipoxygenase inhibitor
ulcerative colitis
SULINDACApproved
Cyclooxygenase inhibitor
spondylitis
SUPROFENApproved
Cyclooxygenase inhibitor
Miosis
TOLMETINApproved
Cyclooxygenase inhibitor
rheumatoid arthritis
TOLMETIN SODIUMApproved
Cyclooxygenase inhibitor
rheumatoid arthritis
Related Genes
CYP4F2Protein interaction98%PTGER3Protein interaction97%PTGIRProtein interaction97%PTGES3Protein interaction96%PLA2G1BProtein interaction96%PLA2G2AProtein interaction96%
Tissue Expression6 tissues
Lung
100%
Bone Marrow
52%
Heart
37%
Brain
29%
Liver
13%
Ovary
12%
Gene Interaction Network
Click a node to explore
PTGS1CYP4F2PTGER3PTGIRPTGES3PLA2G1BPLA2G2A
PROTEIN STRUCTURE
Preparing viewer…
PDB6Y3C · 3.36 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.82LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.64 [0.50–0.82]
RankingsWhere PTGS1 stands among ~20K protein-coding genes
  • #1,274of 20,598
    Most Researched284 · top 10%
  • #37of 1,025
    FDA-Approved Drug Targets56 · top 5%
  • #6,948of 17,882
    Most Constrained (LOEUF)0.82
Genes detectedPTGS1
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
Mechanisms of Damage to the Gastrointestinal Tract From Nonsteroidal Anti-Inflammatory Drugs.
PMID: 29221664
Gastroenterology · 2018
1.00
2
The associations of candidate gene polymorphisms with aspirin resistance in patients with ischemic disease: a meta-analysis.
PMID: 39617913
Hum Genomics · 2024
0.92
3
A meta-analysis of PTGS1 and PTGS2 polymorphisms and NSAID intake on the risk of developing cancer.
PMID: 23967159
PLoS One · 2013
0.90
4
PMID: 32584621
Platelets · 2021
0.80
5
Changes in PTGS1 and ALOX12 Gene Expression in Peripheral Blood Mononuclear Cells Are Associated with Changes in Arachidonic Acid, Oxylipins, and Oxylipin/Fatty Acid Ratios in Response to Omega-3 Fatty Acid Supplementation.
PMID: 26672987
PLoS One · 2015
0.70