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50 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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RACK1
receptor for activated C kinase 1
Chromosome 5 · 5q35.3
NCBI Gene: 10399Ensembl: ENSG00000204628.13HGNC: HGNC:4399UniProt: E9KL35
628PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Highly ConstrainedHub Gene
RESEARCH IMPACT
Highly StudiedTrending
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
ribosome bindingprotein kinase C bindingpositive regulation of apoptotic processpositive regulation of GTPase activityAlzheimer diseasebreast cancerhepatocellular carcinomamelanoma
✦AI Summary

RACK1 is a multifunctional scaffolding protein that regulates diverse cellular processes through protein-protein interactions and post-translational modifications. Mechanistically, RACK1 serves as a critical adaptor protein that binds transcription factors (such as Pax5) 1 and signaling kinases (including ZAK at collided ribosomes) 2 to modulate their stability and activation. RACK1 also participates in translational control by interacting with eIF4E and PKCβII to regulate oncogene translation 3, 4. RACK1 expression is tightly regulated by ubiquitination and SUMOylation: SMURF2 targets RACK1 for proteasomal degradation through K48-linked ubiquitination 5, while SENP3 deSUMOylation and OTUB1 non-canonical ubiquitination stabilize RACK1 3, 4. In the immune microenvironment, elevated RACK1 promotes M2 macrophage polarization via NF-κB signaling in oral cancer 6. Clinically, RACK1 dysregulation associates with multiple malignancies including ovarian, oral squamous cell, and hepatocellular carcinomas, where elevated expression correlates with poor prognosis 5, 6, 3. Additionally, RACK1 is essential for normal B-cell development 1 and prenatal cortical development, where FMRP-mediated regulation maintains normal mitochondrial function and neuronal excitability 7.

Sources cited
1
SMURF2 is an E3 ligase that ubiquitinates RACK1 at K6, K33, and K48, regulating its stability in ovarian cancer
PMID: 37828084
2
RACK1 interacts with ZAK kinase at collided ribosomes to enable ZAK activation through SAM domain dimerization
PMID: 41261136
3
High RACK1 expression promotes M2 macrophage polarization through NF-κB pathway and is associated with poor prognosis in oral squamous cell carcinoma
PMID: 31997535
4
RACK1 stabilizes the transcription factor Pax5 through direct binding and prevents its ubiquitination, essential for B-cell development
PMID: 39256480
5
FMRP regulates RACK1 levels through CNOT1 interaction in a species-specific manner, critical for prenatal cortical development and mitochondrial function
PMID: 37820724
6
SENP3 deSUMOylates RACK1 to increase its stability and interaction with PKCβII, promoting eIF4E-mediated translation of oncogenes in hepatocellular carcinoma
PMID: 39755756
7
OTUB1 stabilizes RACK1 through non-canonical suppression of K48-linked ubiquitination, activating oncogenic transcription in hepatocellular carcinoma
PMID: 38315284
Disease Associationsⓘ20
Alzheimer diseaseOpen Targets
0.21Weak
breast cancerOpen Targets
0.11Weak
hepatocellular carcinomaOpen Targets
0.11Weak
melanomaOpen Targets
0.11Weak
gastric cancerOpen Targets
0.10Weak
neoplasmOpen Targets
0.10Weak
cancerOpen Targets
0.10Suggestive
oral squamous cell carcinomaOpen Targets
0.09Suggestive
colorectal carcinomaOpen Targets
0.09Suggestive
gliomaOpen Targets
0.09Suggestive
cervical cancerOpen Targets
0.09Suggestive
esophageal squamous cell carcinomaOpen Targets
0.09Suggestive
nasopharyngeal carcinomaOpen Targets
0.08Suggestive
non-small cell lung carcinomaOpen Targets
0.08Suggestive
cholangiocarcinomaOpen Targets
0.08Suggestive
gastrointestinal stromal tumorOpen Targets
0.07Suggestive
acute lymphoblastic leukemiaOpen Targets
0.07Suggestive
Hepatic fibrosisOpen Targets
0.07Suggestive
meningiomaOpen Targets
0.07Suggestive
Mobius syndromeOpen Targets
0.07Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
EEF1A1Protein interaction100%EEF1B2Protein interaction100%EEF1DProtein interaction100%EEF1GProtein interaction100%EEF2Protein interaction100%EIF5AProtein interaction100%
Tissue Expression6 tissues
Ovary
100%
Lung
52%
Bone Marrow
49%
Liver
35%
Heart
35%
Brain
26%
Gene Interaction Network
Click a node to explore
RACK1EEF1A1EEF1B2EEF1DEEF1GEEF2EIF5A
PROTEIN STRUCTURE
Preparing viewer…
PDB8GLP · 1.67 Å · EM
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.24Highly Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.09 [0.04–0.24]
RankingsWhere RACK1 stands among ~20K protein-coding genes
  • #364of 20,598
    Most Researched628 · top 5%
  • #699of 17,882
    Most Constrained (LOEUF)0.24 · top 5%
Genes detectedRACK1
Sources retrieved50 papers
Response time—
📄 Sources
50▼
1
Loss of SMURF2 expression enhances RACK1 stability and promotes ovarian cancer progression.
PMID: 37828084
Cell Death Differ · 2023
1.00
2
ZAK activation at the collided ribosome.
PMID: 41261136
Nature · 2026
0.90
3
Roles of RACK1 in centrosome regulation and carcinogenesis.
PMID: 34843916
Cell Signal · 2022
0.88
4
Inhibition of RACK1-Mediated NLRP3 Oligomerization (Active Conformation) Ameliorates Acute Respiratory Distress Syndrome.
PMID: 40349158
Adv Sci (Weinh) · 2025
0.86
5
Ribosome customization and functional diversification among P-stalk proteins regulate late poxvirus protein synthesis.
PMID: 39786991
Cell Rep · 2025
0.84