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25 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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UBE2M
ubiquitin conjugating enzyme E2 M
Chromosome 19 · 19q13.43
NCBI Gene: 9040Ensembl: ENSG00000130725.9HGNC: HGNC:12491UniProt: A0A024R4T4
195PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Highly ConstrainedHub Gene
RESEARCH IMPACT
Trending
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein neddylationprotein bindingNEDD8 transferase activityprotein modification processuterine fibroidhepatocellular carcinomabreast cancerneoplasm
✦AI Summary

UBE2M is a NEDD8-conjugating enzyme (E2) that catalyzes the covalent attachment of NEDD8 to target proteins in the neddylation pathway 1. The enzyme specifically interacts with E3 ligase RBX1 to form the UBE2M-RBX1 complex, which neddylates cullin proteins including CUL1, CUL2, CUL3, and CUL4, thereby activating Cullin-RING E3 ligases (CRLs) 2. UBE2M activity requires both an N-terminal docking peptide and a conserved E2 catalytic core domain for NEDD8 transfer 1. The enzyme plays critical roles in immune regulation, particularly in maintaining regulatory T cell homeostasis and controlling double-negative T cell apoptosis through Bim degradation pathways 23. In cancer contexts, UBE2M promotes tumor progression through multiple mechanisms, including activation of β-catenin/cyclin D1 signaling in hepatocellular carcinoma and formation of positive feedback loops with estrogen receptor α in breast cancer 45. UBE2M function can be enhanced by post-translational modifications such as PRMT1-mediated arginine methylation, which affects metabolic pathways in kidney injury 6. The enzyme represents a promising therapeutic target, with inhibitors like MLN4924 showing efficacy in treating renal cell carcinoma and other malignancies 7.

Sources cited
1
UBE2M is a NEDD8-conjugating enzyme requiring N-terminal docking peptide and catalytic core domain
PMID: 33827629
2
UBE2M-RBX1 complex neddylates cullins and is essential for regulatory T cell maintenance
PMID: 35641500
3
UBE2M regulates double-negative T cell apoptosis through Bim degradation pathways
PMID: 38221551
4
UBE2M promotes hepatocellular carcinoma through β-catenin/cyclin D1 signaling
PMID: 32012120
5
UBE2M forms positive feedback loop with estrogen receptor α in breast cancer
PMID: 39138151
6
PRMT1-mediated methylation enhances UBE2M function in kidney injury
PMID: 40744915
7
MLN4924 inhibitor targets UBE2M-dependent neddylation in renal cell carcinoma
PMID: 29667067
Disease Associationsⓘ20
uterine fibroidOpen Targets
0.16Weak
hepatocellular carcinomaOpen Targets
0.10Suggestive
breast cancerOpen Targets
0.09Suggestive
neoplasmOpen Targets
0.09Suggestive
colorectal carcinomaOpen Targets
0.08Suggestive
melanomaOpen Targets
0.08Suggestive
lung cancerOpen Targets
0.08Suggestive
systemic lupus erythematosusOpen Targets
0.06Suggestive
SepsisOpen Targets
0.05Suggestive
hypoparathyroidism, familial isolated, 2Open Targets
0.04Suggestive
acute myeloid leukemiaOpen Targets
0.04Suggestive
cancerOpen Targets
0.04Suggestive
isolated hyperchlorhidrosisOpen Targets
0.04Suggestive
Hearing loss - familial salivary gland insensitivity to aldosteroneOpen Targets
0.03Suggestive
hearing loss-familial salivary gland insensitivity to aldosterone syndromeOpen Targets
0.03Suggestive
familial isolated hyperparathyroidismOpen Targets
0.03Suggestive
hyperparathyroidismOpen Targets
0.03Suggestive
Escherichia coli InfectionsOpen Targets
0.03Suggestive
intrahepatic cholangiocarcinomaOpen Targets
0.02Suggestive
triple-negative breast cancerOpen Targets
0.02Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
GPS1Protein interaction100%CUL5Protein interaction100%CUL4AProtein interaction100%CUL3Protein interaction100%COPS3Protein interaction100%RBX1Protein interaction100%
Tissue Expression6 tissues
Brain
100%
Heart
67%
Lung
51%
Liver
42%
Ovary
42%
Bone Marrow
35%
Gene Interaction Network
Click a node to explore
UBE2MGPS1CUL5CUL4ACUL3COPS3RBX1
PROTEIN STRUCTURE
Preparing viewer…
PDB3TDU · 1.50 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.27Highly Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.09 [0.03–0.27]
RankingsWhere UBE2M stands among ~20K protein-coding genes
  • #2,190of 20,598
    Most Researched195 · top quartile
  • #926of 17,882
    Most Constrained (LOEUF)0.27 · top 10%
Genes detectedUBE2M
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
Neddylation is a novel therapeutic target for lupus by regulating double negative T cell homeostasis.
PMID: 38221551
Signal Transduct Target Ther · 2024
1.00
2
The Ube2m-Rbx1 neddylation-Cullin-RING-Ligase proteins are essential for the maintenance of Regulatory T cell fitness.
PMID: 35641500
Nat Commun · 2022
0.90
3
Potent 5-Cyano-6-phenyl-pyrimidin-Based Derivatives Targeting DCN1-UBE2M Interaction.
PMID: 31157974
J Med Chem · 2019
0.84
4
UBE2M forms a positive feedback loop with estrogen receptor to drive breast cancer progression and drug resistance.
PMID: 39138151
Cell Death Dis · 2024
0.80
5
UBE2M-mediated p27(Kip1) degradation in gemcitabine cytotoxicity.
PMID: 21477582
Biochem Pharmacol · 2011
0.72