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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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AKR7A3
aldo-keto reductase family 7 member A3
Chromosome 1 · 1p36.13
NCBI Gene: 22977Ensembl: ENSG00000162482.6HGNC: HGNC:390UniProt: A0A384MDN8
26PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingalcohol dehydrogenase (NADP+) activityidentical protein bindingaflatoxin catabolic processhepatocellular carcinomaneoplasmBarrett's esophaguscholelithiasis
✦AI Summary

AKR7A3 (aldo-keto reductase family 7 member A3) is a human enzyme that catalyzes NADPH-dependent reduction of carbonyl-containing compounds, including aldehydes and ketones 1. Its primary function involves detoxification of toxic metabolites, particularly aflatoxin B1 (AFB1) dialdehyde, which it reduces to less harmful alcohol derivatives via monoaldehyde intermediates 2. The enzyme demonstrates high catalytic efficiency with AFB1 dihydrodiol, with kinetic parameters comparable to other AFB1-metabolizing enzymes like cytochrome P450s and glutathione S-transferases 1. AKR7A3 shares 88% identity with human AKR7A2 and is expressed in liver and various extrahepatic tissues including stomach, pancreas, and kidney 1. Disease relevance includes its downregulation in gastric cancer and pancreatic ductal adenocarcinoma (PDAC), where reduced expression correlates with poor prognosis and increased metastasis 34. In PDAC, AKR7A3 inhibits progression by regulating PHGDH-mediated autophagy 4. Clinically, genetic polymorphisms in AKR7A3 (rs1738023/rs1738025) are associated with bleeding complications in elderly patients treated with rivaroxaban 5. The gene contains Nrf2 binding sites in its promoter, making it highly inducible by antioxidants 6. AKR7A3 represents a potential therapeutic target and prognostic marker for cancer treatment.

Sources cited
1
AKR7A3 catalyzes NADPH-dependent reduction of carbonyl compounds and has high catalytic efficiency with AFB1 dihydrodiol
PMID: 10383892
2
AKR7A3 reduces AFB1 dialdehyde to alcohol derivatives and provides protection against AFB1-induced cytotoxicity
PMID: 18416522
3
AKR7A3 expression is lower in gastric cancer tissues and correlates with better prognosis when highly expressed
PMID: 36827074
4
AKR7A3 is downregulated in pancreatic cancer and inhibits progression by regulating PHGDH-mediated autophagy
PMID: 36951402
5
AKR7A3 polymorphisms (rs1738023/rs1738025) are associated with bleeding in elderly patients on rivaroxaban
PMID: 34859601
6
AKR7A3 contains Nrf2 binding sites and is highly inducible by antioxidants
PMID: 31529389
Disease Associationsⓘ20
hepatocellular carcinomaOpen Targets
0.09Suggestive
neoplasmOpen Targets
0.08Suggestive
Barrett's esophagusOpen Targets
0.06Suggestive
cholelithiasisOpen Targets
0.06Suggestive
phototoxic dermatitisOpen Targets
0.04Suggestive
esophageal adenocarcinomaOpen Targets
0.03Suggestive
non-small cell lung carcinomaOpen Targets
0.03Suggestive
nontoxic goiterOpen Targets
0.02Suggestive
clear cell renal carcinomaOpen Targets
0.02Suggestive
gastric carcinomaOpen Targets
0.02Suggestive
gastric non-cardia carcinomaOpen Targets
0.01Suggestive
multiple myelomaOpen Targets
0.01Suggestive
gastric cardia carcinomaOpen Targets
0.01Suggestive
kidney oncocytomaOpen Targets
0.01Suggestive
pancreatic ductal adenocarcinomaOpen Targets
0.01Suggestive
cancerOpen Targets
0.01Suggestive
pancreatic carcinomaOpen Targets
0.01Suggestive
liver cancerOpen Targets
0.01Suggestive
transitional cell carcinoma of kidneyOpen Targets
0.01Suggestive
pachyonychia congenitaOpen Targets
0.01Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
ALDH16A1Shared pathway100%AKR1B1Protein interaction99%AKR1A1Protein interaction99%MSCProtein interaction75%AKR7A2Protein interaction61%ALDH3A1Shared pathway50%
Tissue Expression6 tissues
Liver
100%
Ovary
2%
Bone Marrow
2%
Brain
1%
Lung
0%
Heart
0%
Gene Interaction Network
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AKR7A3ALDH16A1AKR1B1AKR1A1MSCAKR7A2ALDH3A1
PROTEIN STRUCTURE
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PDB2CLP · 3.00 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.41LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF1.07 [0.82–1.41]
RankingsWhere AKR7A3 stands among ~20K protein-coding genes
  • #12,729of 20,598
    Most Researched26
  • #14,573of 17,882
    Most Constrained (LOEUF)1.41
Genes detectedAKR7A3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Protection against aflatoxin B1-induced cytotoxicity by expression of the cloned aflatoxin B1-aldehyde reductases rat AKR7A1 and human AKR7A3.
PMID: 18416522
Chem Res Toxicol · 2008
1.00
2
cDNA cloning, expression and activity of a second human aflatoxin B1-metabolizing member of the aldo-keto reductase superfamily, AKR7A3.
PMID: 10383892
Carcinogenesis · 1999
0.90
3
Non-synonymous alterations in AKR7A3 and ABCA6 correlate with bleeding in aged patients treated with rivaroxaban.
PMID: 34859601
Clin Transl Sci · 2022
0.80
4
Expression of AKRs superfamily and prognostic in human gastric cancer.
PMID: 36827074
Medicine (Baltimore) · 2023
0.70
5
AKR7A3 modulates the metastasis of pancreatic ductal adenocarcinoma through regulating PHGDH-suppressed autophagy.
PMID: 36951402
Cancer Sci · 2023
0.60