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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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ARHGDIB
Rho GDP dissociation inhibitor beta
Chromosome 12 · 12p12.3
NCBI Gene: 397Ensembl: ENSG00000111348.10HGNC: HGNC:679UniProt: P52566
108PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
GTPase activityRho GDP-dissociation inhibitor activityprotein bindingsmall GTPase bindinggastric cancerneoplasmbreast cancerdiabetes mellitus
✦AI Summary

ARHGDIB (Rho GDP dissociation inhibitor beta) is a cytosolic protein that regulates Rho family GTPase signaling by inhibiting GDP dissociation and GTP binding 12, thereby controlling actin cytoskeleton reorganization 3. Beyond its canonical GTPase regulatory function, ARHGDIB exhibits diverse roles across multiple pathological contexts. In bladder cancer, the FOXA1-KDM6A-ARHGDIB axis suppresses metastasis by inhibiting Rac1 activation 4, while ARHGDIB delactylation by HDAC2 promotes metastasis and cisplatin resistance through impaired Rac1 binding 5. In glioma, elevated ARHGDIB expression correlates with poor prognosis and recruits immunosuppressive M2 macrophages, reshaping the tumor microenvironment 6. In melanoma, the circSipa1l1-IGF2BP1-ARHGDIB axis regulates cell differentiation via ERK signaling 7. Clinically, anti-ARHGDIB autoantibodies associate with kidney allograft rejection; combined presence with donor-specific HLA antibodies increases graft failure risk 19.5-fold 89. ARHGDIB also emerged as a diagnostic biomarker for sepsis-induced acute lung injury 10. These findings establish ARHGDIB as a multifunctional regulator with significant implications for cancer progression, transplant immunity, and acute inflammatory conditions.

Sources cited
1
ARHGDIB inhibits GDP dissociation from Rho proteins and subsequent GTP binding
PMID: 7512369
2
ARHGDIB regulates GDP/GTP exchange reaction of Rho proteins
PMID: 8356058
3
ARHGDIB regulates actin cytoskeleton reorganization mediated by Rho family members
PMID: 8262133
4
KDM6A promotes ARHGDIB transcription to inhibit Rac1 and suppress bladder cancer metastasis
PMID: 34006303
5
HDAC2-mediated delactylation of ARHGDIB attenuates Rac1 binding and promotes bladder cancer metastasis and chemoresistance
PMID: 41637189
6
ARHGDIB is overexpressed in glioma, recruits immunosuppressive M2 macrophages, and serves as a prognostic biomarker
PMID: 40372473
7
CircSipa1l1-IGF2BP1-ARHGDIB axis regulates melanoma cell differentiation via ERK signaling
PMID: 41163180
8
Anti-ARHGDIB antibodies combined with DSA increase kidney allograft graft failure risk 19.5-fold
PMID: 31651716
9
Anti-ARHGDIB autoantibodies are elevated in chronic-active antibody-mediated rejection of kidney allografts
PMID: 33358038
10
ARHGDIB is among five consensus biomarkers for diagnosing sepsis-induced acute lung injury
PMID: 37700323
Disease Associationsⓘ20
gastric cancerOpen Targets
0.11Weak
neoplasmOpen Targets
0.09Suggestive
breast cancerOpen Targets
0.08Suggestive
diabetes mellitusOpen Targets
0.08Suggestive
gliomaOpen Targets
0.07Suggestive
acute lymphoblastic leukemiaOpen Targets
0.07Suggestive
Abruptio PlacentaeOpen Targets
0.06Suggestive
cancerOpen Targets
0.05Suggestive
hepatocellular carcinomaOpen Targets
0.04Suggestive
colorectal carcinomaOpen Targets
0.04Suggestive
lung cancerOpen Targets
0.04Suggestive
melanomaOpen Targets
0.04Suggestive
combined immunodeficiency with skin granulomasOpen Targets
0.04Suggestive
immune deficiency, familial variableOpen Targets
0.04Suggestive
placenta praeviaOpen Targets
0.04Suggestive
Raynaud diseaseOpen Targets
0.04Suggestive
Alymphoid cystic thymic dysgenesisOpen Targets
0.04Suggestive
neutropenia, severe congenital, 2, autosomal dominantOpen Targets
0.04Suggestive
spermatogenic failure 48Open Targets
0.04Suggestive
Townes-Brocks syndromeOpen Targets
0.04Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
RHOAProtein interaction96%NGFRProtein interaction96%CDC42Protein interaction92%PRKACAProtein interaction91%PRKACGProtein interaction91%PRKACBProtein interaction91%
Tissue Expression6 tissues
Bone Marrow
100%
Lung
43%
Heart
13%
Liver
7%
Brain
5%
Ovary
3%
Gene Interaction Network
Click a node to explore
ARHGDIBRHOANGFRCDC42PRKACAPRKACGPRKACB
PROTEIN STRUCTURE
Preparing viewer…
PDB5H1D · 1.49 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.88LoF Tolerant
pLIⓘ
0.05Tolerant
Observed/Expected LoF0.50 [0.30–0.88]
RankingsWhere ARHGDIB stands among ~20K protein-coding genes
  • #4,393of 20,598
    Most Researched108 · top quartile
  • #7,834of 17,882
    Most Constrained (LOEUF)0.88
Genes detectedARHGDIB
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
KDM6A-ARHGDIB axis blocks metastasis of bladder cancer by inhibiting Rac1.
PMID: 34006303
Mol Cancer · 2021
1.00
2
A diagnostic model for sepsis-induced acute lung injury using a consensus machine learning approach and its therapeutic implications.
PMID: 37700323
J Transl Med · 2023
0.90
3
Antibodies Against ARHGDIB and ARHGDIB Gene Expression Associate With Kidney Allograft Outcome.
PMID: 31651716
Transplantation · 2020
0.80
4
ARHGDIB as a prognostic biomarker and modulator of the immunosuppressive microenvironment in glioma.
PMID: 40372473
Cancer Immunol Immunother · 2025
0.70
5
Delactylation of the tumor suppressor ARHGDIB drives metastasis and chemoresistance in bladder cancer.
PMID: 41637189
Cell Rep · 2026
0.60