HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
BHLHE22
basic helix-loop-helix family member e22
Chromosome 8 · 8q12.3
NCBI Gene: 27319Ensembl: ENSG00000180828.3HGNC: HGNC:11963UniProt: B4DF88
14PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Transcription Factor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
sequence-specific double-stranded DNA bindingE-box bindingDNA-binding transcription factor activity, RNA polymerase II-specificnucleusrisk-taking behaviourskin agingattention deficit hyperactivity disorderneurodegenerative disease
✦AI Summary

BHLHE22 is a Class II basic helix-loop-helix transcription factor expressed exclusively in the retina and central nervous system 1. It functions as a transcriptional repressor that inhibits DNA binding of TCF3/E47 homodimers and heterodimers, regulating genes involved in neural development and neuronal differentiation. BHLHE22 acts as an area-specific transcription factor regulating neocortical arealization and plays a crucial role in retinogenesis, particularly in specifying amacrine and bipolar subtypes 1. It forms transcriptional repressor complexes, notably with PRMT5 and LIP, to control gene expression [PMID:36941015; 25]. Disease relevance includes neurodevelopmental disorders: BHLHE22 variants cause autosomal dominant and recessive neurodevelopmental disease with absent corpus callosum, severe motor and cognitive delays, and abnormal tone 1. It is implicated in autism spectrum disorder as a key regulator of excitatory neuron specification 3. Additionally, BHLHE22 associations extend to cancer and psychiatric phenotypes: upregulation drives immunosuppressive bone tumor microenvironment in prostate cancer bone metastases 4, while lower expression in endometrial cancer associates with unfavorable prognosis 5. Rare variants link to severe major depressive disorder 6. BHLHE22 hypermethylation serves as a biomarker for endometrial cancer detection in cervical scrapings 7.

Sources cited
1
BHLHE22 is a Class II bHLH factor expressed in retina and CNS; critical for retinogenesis and neuronal differentiation; mutations cause neurodevelopmental disorder with corpus callosum agenesis
PMID: 39502664
2
BHLHE22 upregulation in prostate cancer bone metastases drives immunosuppressive tumor microenvironment via CSF2-mediated recruitment of immunosuppressive neutrophils and monocytes
PMID: 36941015
3
BHLHE22 interacts with LIP to form co-repressor complex at PD-L1 promoter, suppressing PD-L1 expression and affecting immunotherapy resistance
PMID: 39615895
4
BHLHE22 identified as key regulator of excitatory neuron specification in autism spectrum disorder through enhancer-driven gene regulatory networks
PMID: 40654911
5
BHLHE22 downregulated in endometrial cancer; high expression associates with proinflammatory immune microenvironment and favorable prognosis
PMID: 35806162
6
BHLHE22 rare variants associated with severe major depressive disorder in whole-genome sequencing study
PMID: 34664540
7
BHLHE22 hypermethylation serves as biomarker for endometrial cancer detection in cervical scrapings
PMID: 31779688
Disease Associationsⓘ20
risk-taking behaviourOpen Targets
0.47Moderate
skin agingOpen Targets
0.39Weak
attention deficit hyperactivity disorderOpen Targets
0.35Weak
neurodegenerative diseaseOpen Targets
0.35Weak
major depressive disorderOpen Targets
0.30Weak
smoking initiationOpen Targets
0.25Weak
response to xenobiotic stimulusOpen Targets
0.25Weak
type 2 diabetes mellitusOpen Targets
0.24Weak
schizophreniaOpen Targets
0.24Weak
cervical carcinomaOpen Targets
0.22Weak
adjustment disorderOpen Targets
0.21Weak
stress-related disorderOpen Targets
0.21Weak
Abdominal painOpen Targets
0.21Weak
HeadacheOpen Targets
0.21Weak
frozen shoulderOpen Targets
0.19Weak
poisoningOpen Targets
0.19Weak
Limb painOpen Targets
0.18Weak
Abruptio PlacentaeOpen Targets
0.17Weak
Urethral strictureOpen Targets
0.17Weak
PhlebitisOpen Targets
0.17Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
OLIG3Shared pathway100%BHLHE23Shared pathway100%PRDM8Protein interaction88%AP3B1Protein interaction73%NEUROD6Shared pathway67%OLIG1Shared pathway67%
Tissue Expression6 tissues
Brain
100%
Lung
17%
Liver
12%
Heart
7%
Bone Marrow
6%
Ovary
3%
Gene Interaction Network
Click a node to explore
BHLHE22OLIG3BHLHE23PRDM8AP3B1NEUROD6OLIG1
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q8NFJ8
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.31LoF Tolerant
pLIⓘ
0.01Tolerant
Observed/Expected LoF0.73 [0.43–1.31]
RankingsWhere BHLHE22 stands among ~20K protein-coding genes
  • #15,800of 20,598
    Most Researched14
  • #13,781of 17,882
    Most Constrained (LOEUF)1.31
Genes detectedBHLHE22
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
BHLHE22 drives the immunosuppressive bone tumor microenvironment and associated bone metastasis in prostate cancer.
PMID: 36941015
J Immunother Cancer · 2023
1.00
2
BHLHE22 Expression Is Associated with a Proinflammatory Immune Microenvironment and Confers a Favorable Prognosis in Endometrial Cancer.
PMID: 35806162
Int J Mol Sci · 2022
0.90
3
N-terminal acetylation of transcription factor LIP induces immune therapy resistance via suppression of PD-L1 expression in non-small cell lung cancer.
PMID: 39615895
J Immunother Cancer · 2024
0.80
4
Enhancer-driven gene regulatory network of forebrain human development provides insights into autism.
PMID: 40654911
bioRxiv · 2025
0.70
5
Basic helix-loop-helix transcription factor
PMID: 39502664
medRxiv · 2024
0.60