HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
CREBZF
CREB/ATF bZIP transcription factor
Chromosome 11 · 11q14.1
NCBI Gene: 58487Ensembl: ENSG00000137504.16HGNC: HGNC:24905UniProt: E9PIM0
50PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Transcription Factor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
negative regulation of DNA-templated transcriptionpositive regulation of transcription by RNA polymerase IInucleusprotein bindingneurodegenerative diseasebreast cancerInsulin resistancegastric cancer
✦AI Summary

CREBZF is a CREB/ATF bZIP transcription factor that plays crucial roles in metabolic regulation, stress responses, and disease pathogenesis. The protein functions as a metabolic regulator in adipose tissue, where it promotes inflammatory responses in macrophages that contribute to insulin resistance and type 2 diabetes by competitively inhibiting IκBα binding to p65, enhancing NF-κB activity 1. In thermogenesis regulation, CREBZF undergoes glucose-induced acetylation at Lys208 by CBP/p300 and HDAC3, which stabilizes the protein and allows it to associate with PGC-1α to repress thermogenic gene expression 2. CREBZF also serves as a critical checkpoint in liver disease progression, promoting hepatocyte injury and NASH development by stimulating osteopontin production through miR-6964-3p inhibition 3. The transcription factor responds to amino acid deprivation through an AARE-like element in its promoter 4 and functions as a positive regulator of p53 tumor suppressor activity, stabilizing p53 through post-translational modifications 5. CREBZF expression is dysregulated in various cancers, where it can suppress breast cancer progression through feedback loops involving circPAPD4 6 and is targeted by miRNAs in gastric cancer 7.

Sources cited
1
CREBZF promotes inflammatory responses in adipose tissue macrophages contributing to insulin resistance by enhancing NF-κB activity
PMID: 38286660
2
CREBZF undergoes glucose-induced acetylation and associates with PGC-1α to repress thermogenic gene expression
PMID: 38588421
3
CREBZF promotes liver fibrosis and NASH progression by stimulating osteopontin production
PMID: 36680394
4
CREBZF responds to amino acid deprivation through an AARE-like element in its promoter
PMID: 20026304
5
CREBZF functions as a positive regulator of p53 tumor suppressor activity
PMID: 22983008
6
CREBZF suppresses breast cancer progression through feedback loops involving circPAPD4
PMID: 37264406
7
CREBZF is targeted by miRNAs and affects migration in gastric cancer cells
PMID: 32218690
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.40Weak
breast cancerOpen Targets
0.08Suggestive
Insulin resistanceOpen Targets
0.07Suggestive
gastric cancerOpen Targets
0.06Suggestive
neoplasmOpen Targets
0.05Suggestive
dyshidrosisOpen Targets
0.04Suggestive
device complicationOpen Targets
0.04Suggestive
obesityOpen Targets
0.03Suggestive
type 2 diabetes mellitusOpen Targets
0.03Suggestive
non-alcoholic steatohepatitisOpen Targets
0.03Suggestive
osteomyelitisOpen Targets
0.03Suggestive
mathematical abilityOpen Targets
0.02Suggestive
Abnormal nasolacrimal system morphologyOpen Targets
0.02Suggestive
metabolic diseaseOpen Targets
0.02Suggestive
rheumatoid arthritisOpen Targets
0.02Suggestive
cancerOpen Targets
0.02Suggestive
HyperglycemiaOpen Targets
0.02Suggestive
overnutritionOpen Targets
0.01Suggestive
osteosarcomaOpen Targets
0.01Suggestive
Hepatic steatosisOpen Targets
0.01Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
HCFC1Protein interaction97%CREB3Protein interaction97%HCFC2Protein interaction97%ATF4Protein interaction93%NOL9Protein interaction85%CREB3L4Protein interaction83%
Tissue Expression6 tissues
Ovary
100%
Lung
58%
Liver
53%
Bone Marrow
47%
Heart
35%
Brain
32%
Gene Interaction Network
Click a node to explore
CREBZFHCFC1CREB3HCFC2ATF4NOL9CREB3L4
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q9NS37
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.74LoF Tolerant
pLIⓘ
0.32Tolerant
Observed/Expected LoF0.41 [0.24–0.74]
RankingsWhere CREBZF stands among ~20K protein-coding genes
  • #8,791of 20,598
    Most Researched50
  • #5,791of 17,882
    Most Constrained (LOEUF)0.74
Genes detectedCREBZF
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Macrophage CREBZF Orchestrates Inflammatory Response to Potentiate Insulin Resistance and Type 2 Diabetes.
PMID: 38286660
Adv Sci (Weinh) · 2024
1.00
2
Glucose regulation of adipose tissue browning by CBP/p300- and HDAC3-mediated reversible acetylation of CREBZF.
PMID: 38588421
Proc Natl Acad Sci U S A · 2024
0.90
3
Intrahepatic osteopontin signaling by CREBZF defines a checkpoint for steatosis-to-NASH progression.
PMID: 36680394
Hepatology · 2023
0.80
4
CREBZF mRNA nanoparticles suppress breast cancer progression through a positive feedback loop boosted by circPAPD4.
PMID: 37264406
J Exp Clin Cancer Res · 2023
0.70
5
Amino acid deprivation induces CREBZF/Zhangfei expression via an AARE-like element in the promoter.
PMID: 20026304
Biochem Biophys Res Commun · 2010
0.60