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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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CSNK1G3
casein kinase 1 gamma 3
Chromosome 5 · 5q23.2
NCBI Gene: 1456Ensembl: ENSG00000151292.19HGNC: HGNC:2456UniProt: A0A8V8TKT3
60PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingprotein serine/threonine kinase activityplasma membranepositive regulation of canonical Wnt signaling pathwayessential hypertensioncardiovascular diseasehypertensionAlzheimer disease
✦AI Summary

CSNK1G3 (casein kinase 1 gamma 3) is a serine/threonine-protein kinase that phosphorylates acidic protein substrates and participates in multiple cellular pathways including Wnt signaling and synaptic transmission 1. The protein localizes to the nucleus, plasma membrane, and cytoplasm, where it regulates canonical Wnt signaling, endocytosis, and signal transduction processes. Mechanistically, CSNK1G3 functions as a nodal kinase in cancer signaling networks. RNAi screening identified CSNK1G3 as an Akt-cooperating kinase; CSNK1G3 inhibition combined with Akt inhibition enhanced cancer cell killing and reduced phosphorylation of Akt Ser-473 and ribosomal protein S6 2. In triple-negative breast cancer, the curcumin derivative N17 exerts anti-cancer effects by targeting CSNK1G3 to suppress p-AKT(S473) phosphorylation, triggering apoptosis and inhibiting epithelial-mesenchymal transition 3. Clinically, CSNK1G3 alterations occur as fusion partners in cancer; a CSNK1G3-ALK fusion was identified in lung squamous cell carcinoma and responded to ALK tyrosine kinase inhibitors with durable disease control exceeding 30 months 4. Additionally, CSNK1G3 expression is dysregulated in vitiligo, with significantly reduced mRNA levels in depigmented lesional skin compared to non-lesional skin in an autoimmune mouse model 5. CSNK1G3 also shows signatures of positive natural selection in Taiwanese Han populations with associations to metabolic traits 6.

Sources cited
1
Protocol describes CSNK1G3 as a casein kinase subfamily member with cellular expression capabilities
PMID: 37119140
2
CSNK1G3 is a therapeutic target in triple-negative breast cancer; inhibition of CSNK1G3 suppresses p-AKT(S473), triggers apoptosis and inhibits EMT
PMID: 39127154
3
CSNK1G3-ALK fusion identified in lung squamous cell carcinoma with response to ALK tyrosine kinase inhibitors
PMID: 40783309
4
CSNK1G3 expression significantly reduced in depigmented lesional skin in autoimmune vitiligo model
PMID: 33084421
5
CSNK1G3 identified as positive selection signature in Taiwanese Han population with associations to metabolic traits
PMID: 33170928
6
CSNK1G3 identified as Akt-cooperating kinase; combined CSNK1G3 and Akt inhibition enhances cancer cell killing
PMID: 16247451
7
siRNA targeting CSNK1G3 negatively regulates translation readthrough
PMID: 29177465
Disease Associationsⓘ20
essential hypertensionOpen Targets
0.29Weak
cardiovascular diseaseOpen Targets
0.29Weak
hypertensionOpen Targets
0.24Weak
Alzheimer diseaseOpen Targets
0.24Weak
burnOpen Targets
0.22Weak
cataractOpen Targets
0.20Weak
trauma complicationOpen Targets
0.20Weak
glomerulonephritisOpen Targets
0.17Weak
ProptosisOpen Targets
0.17Weak
dementiaOpen Targets
0.15Weak
Abnormality of the skeletal systemOpen Targets
0.13Weak
postmenopausal atrophic vaginitisOpen Targets
0.13Weak
malunion fractureOpen Targets
0.13Weak
placenta praeviaOpen Targets
0.13Weak
preeclampsiaOpen Targets
0.12Weak
systemic lupus erythematosusOpen Targets
0.12Weak
response to xenobiotic stimulusOpen Targets
0.04Suggestive
hemoglobin D diseaseOpen Targets
0.04Suggestive
type 2 diabetes mellitusOpen Targets
0.04Suggestive
Hemoglobin E - beta-thalassemiaOpen Targets
0.03Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
PRKACBProtein interaction97%PRKACGProtein interaction97%PRKACAProtein interaction97%GRK2Protein interaction91%GRK3Protein interaction91%SMOProtein interaction91%
Tissue Expression6 tissues
Liver
100%
Brain
99%
Heart
98%
Bone Marrow
92%
Ovary
85%
Lung
74%
Gene Interaction Network
Click a node to explore
CSNK1G3PRKACBPRKACGPRKACAGRK2GRK3SMO
PROTEIN STRUCTURE
Preparing viewer…
PDB2IZR · 1.30 Å · X-ray
View on RCSB ↗
RankingsWhere CSNK1G3 stands among ~20K protein-coding genes
  • #7,647of 20,598
    Most Researched60
Genes detectedCSNK1G3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Protocol for casein kinase 1γ3 CSNK1G3 gene knockout and recombinant gene expression in cultured HeLa cells.
PMID: 37119140
STAR Protoc · 2023
1.00
2
Cloning and chromosome mapping of the human casein kinase I gamma3 gene (CSNK1G3).
PMID: 9925945
Cytogenet Cell Genet · 1998
0.90
3
Novel curcumin derivatives N17 exert anti-cancer effects through the CSNK1G3/AKT axis in triple-negative breast cancer.
PMID: 39127154
Biochem Pharmacol · 2024
0.80
4
Clinical Outcomes of Patients With Advanced ALK-Rearranged Lung Squamous Cell Carcinoma Treated With ALK Tyrosine Kinase Inhibitors.
PMID: 40783309
Clin Lung Cancer · 2025
0.70
5
Autoimmune response against tyrosinase induces depigmentation in C57BL/6 black mice.
PMID: 33084421
Autoimmunity · 2020
0.60