HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
DACT2
dishevelled binding antagonist of beta catenin 2
Chromosome 6 · 6q27
NCBI Gene: 168002Ensembl: ENSG00000164488.12HGNC: HGNC:21231UniProt: Q5SW24
37PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein kinase C bindingbeta-catenin bindingtranscription factor bindingprotein kinase A bindingfood allergydiabetes mellitusparasitic infectionleukemia
✦AI Summary

DACT2 (dishevelled binding antagonist of beta-catenin 2) is a negative regulator of Wnt/β-catenin signaling that functions as a tumor suppressor across multiple cancer types. DACT2 antagonizes the canonical Wnt pathway and negatively regulates Nodal signaling, likely through promotion of receptor degradation 1. The gene is frequently silenced in human cancers via promoter hypermethylation, including gastric cancer (55.7% of cases), breast cancer (49.7%), colorectal cancer, and oral squamous cell carcinoma 1234. In gastric cancer, DACT2 methylation correlates with reduced expression, increased tumor invasion, and intravascular emboli, though paradoxically with improved chemotherapy response 1. In colorectal cancer, DACT2 downregulation associates with advanced tumor stage and poor prognosis 56. Restoration of DACT2 expression suppresses cancer cell proliferation, migration, and xenograft growth by inhibiting both canonical and noncanonical Wnt signaling 13. Recent evidence indicates DACT2 regulates Wnt signaling in mesenchymal progenitor cells to control osteogenic differentiation 7. The gene represents a promising epigenetic biomarker and therapeutic target; kaempferol-mediated DACT2 demethylation reduces colorectal cancer tumor burden 6.

Sources cited
1
DACT2 is frequently methylated in gastric cancer, suppresses cell proliferation and invasion through Wnt pathway inhibition, and influences chemotherapy response
PMID: 25520862
2
DACT2 is downregulated in colorectal cancer tissues and functions as a tumor suppressor associated with tumor stage
PMID: 37610179
3
DACT2 promoter hypermethylation occurs in 32.9% of breast cancers and correlates with advanced tumor stages
PMID: 29745077
4
DACT2 methylation in breast cancer activates Wnt signaling and is associated with tumor size; DACT2 restoration suppresses Wnt/β-catenin signaling and cancer growth
PMID: 28607412
5
DACT2 promoter hypermethylation increases with age over 56 years in oral squamous cell carcinoma patients
PMID: 25524937
6
DACT2 is silenced via hypermethylation in colorectal cancer with poor prognosis correlation; kaempferol demethylates DACT2 and inhibits Wnt pathway to reduce tumor burden
PMID: 29199082
7
DACT2 regulates canonical Wnt signaling in mesenchymal progenitor cells to control osteogenic differentiation
PMID: 39025061
8
DACT2 is a paralog of DACT1 containing conserved DAPH domains and represents an evolutionarily distinct member of the Wnt signaling regulator family
PMID: 15870912
Disease Associationsⓘ20
food allergyOpen Targets
0.29Weak
diabetes mellitusOpen Targets
0.28Weak
parasitic infectionOpen Targets
0.18Weak
leukemiaOpen Targets
0.18Weak
breast cancerOpen Targets
0.10Weak
chronic pulmonary heart diseaseOpen Targets
0.10Weak
psoriatic arthritisOpen Targets
0.08Suggestive
esophageal cancerOpen Targets
0.08Suggestive
nasopharyngeal carcinomaOpen Targets
0.08Suggestive
papillary thyroid carcinomaOpen Targets
0.08Suggestive
gliomaOpen Targets
0.08Suggestive
neoplasmOpen Targets
0.07Suggestive
hepatocellular carcinomaOpen Targets
0.07Suggestive
atrial fibrillationOpen Targets
0.07Suggestive
thyroid cancerOpen Targets
0.06Suggestive
cervical carcinomaOpen Targets
0.05Suggestive
retinitis pigmentosa 1Open Targets
0.05Suggestive
hypothyroidismOpen Targets
0.04Suggestive
esophageal squamous cell carcinomaOpen Targets
0.04Suggestive
CachexiaOpen Targets
0.04Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
DACT3Protein interaction93%CTNNB1Protein interaction71%VSIG1Shared pathway25%RILPL2Shared pathway25%ARHGDIGShared pathway25%RILPL1Shared pathway20%
Tissue Expression6 tissues
Liver
100%
Heart
46%
Brain
34%
Lung
5%
Bone Marrow
3%
Ovary
2%
Gene Interaction Network
Click a node to explore
DACT2DACT3CTNNB1VSIG1RILPL2ARHGDIGRILPL1
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q5SW24
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.47LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.93 [0.60–1.47]
RankingsWhere DACT2 stands among ~20K protein-coding genes
  • #10,610of 20,598
    Most Researched37
  • #14,980of 17,882
    Most Constrained (LOEUF)1.47
Genes detectedDACT2
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
DACT2 is frequently methylated in human gastric cancer and methylation of DACT2 activated Wnt signaling.
PMID: 25520862
Am J Cancer Res · 2014
1.00
2
Different expression of
PMID: 37610179
Nucleosides Nucleotides Nucleic Acids · 2024
0.90
3
Association between promoter hypermethylation of the DACT2 gene and tumor stages in breast cancer.
PMID: 29745077
J BUON · 2018
0.80
4
Expression and epigenetic regulation of DACT1 and DACT2 in oral squamous cell carcinoma.
PMID: 25524937
Cancer Biomark · 2015
0.70
5
Identification and characterization of rat Dact1 and Dact2 genes in silico.
PMID: 15870912
Int J Mol Med · 2005
0.60