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26 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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FGF1
fibroblast growth factor 1
Chromosome 5 · 5q31.3
NCBI Gene: 2246Ensembl: ENSG00000113578.19HGNC: HGNC:3665UniProt: A8K147
262PubMed Papers
20Diseases
6Drugs
0Pathogenic Variants
RESEARCH IMPACT
Trending
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
positive regulation of cell population proliferationfibroblast growth factor receptor signaling pathwayfibroblast growth factor receptor bindingintegrin bindingcancerbone development diseasefemale reproductive endometrioid cancerAbnormality of the skeletal system
✦AI Summary

FGF1 (fibroblast growth factor 1) is a pleiotropic signaling molecule that regulates cell survival, proliferation, angiogenesis, and differentiation 1. FGF1 functions as a ligand for FGFR1 and integrins, with heparin-dependent binding to FGFR1 triggering receptor dimerization and autophosphorylation of tyrosine residues that activate downstream cascades including MAPK and AKT signaling 1. FGF1 is highly expressed in adult brain and kidney tissues and during development 1. Clinically, FGF1 demonstrates therapeutic potential across multiple disease contexts. In type 2 diabetes, exogenous FGF1 delivery suppresses hepatic glucose production by inhibiting adipose lipolysis through FGF receptor 1-dependent activation of phosphodiesterase 4D, achieving insulin sensitization without weight gain or hepatic steatosis 23. In inflammatory bowel disease, colonic epithelial FGF1 promotes intestinal stem cell differentiation toward goblet cells via FGFR2-TCF4-ATOH1 signaling, with FGF1 levels inversely correlated with disease severity 4. FGF1 protects against diabetic cardiomyopathy through AMPK/Nur77-dependent mitochondrial function improvement and oxidative stress reduction 5. Additionally, non-mitogenic FGF1 variants mitigate drug-induced liver injury by regulating bile acid homeostasis via FGFR4-ERK signaling 6. Gene therapy approaches utilizing FGF1 show promise for promoting angiogenesis in peripheral arterial disease 7.

Sources cited
1
FGF1 regulation of cell survival, proliferation, and differentiation; tissue expression patterns; diabetic phenotype in FGF1 mutants on high-fat diet
PMID: 39074995
2
FGF1 suppresses hepatic glucose production by inhibiting adipose lipolysis through PDE4D activation in type 2 diabetes
PMID: 34986332
3
Exogenous FGF1 achieves insulin sensitization and glucose lowering without weight gain or liver steatosis via FGFR1 signaling
PMID: 25043058
4
Colonic epithelial FGF1 directs intestinal stem cell commitment toward goblet cells via FGFR2-TCF4-ATOH1 axis to suppress IBD
PMID: 40188210
5
FGF1 protects against diabetic cardiomyopathy through AMPK/Nur77-dependent mitochondrial function and ROS reduction
PMID: 33762571
6
Hepatocyte FGF1 regulates bile acid homeostasis via FGFR4-ERK signaling to protect against drug-induced liver injury
PMID: 39731358
7
FGF1 gene therapy promotes angiogenesis for treatment of peripheral arterial disease
PMID: 20860417
8
Piezo1-mediated FGF1 release from adipocytes induces preadipocyte differentiation through FGFR1 during obesity development
PMID: 32385276
Disease Associationsⓘ20
cancerOpen Targets
0.61Moderate
bone development diseaseOpen Targets
0.60Moderate
female reproductive endometrioid cancerOpen Targets
0.50Moderate
Abnormality of the skeletal systemOpen Targets
0.47Moderate
ovarian carcinomaOpen Targets
0.47Moderate
neurodegenerative diseaseOpen Targets
0.37Weak
acrocephalosyndactylyOpen Targets
0.37Weak
craniosynostosisOpen Targets
0.37Weak
LeishmaniasisOpen Targets
0.37Weak
trypanosomiasisOpen Targets
0.37Weak
prostate cancerOpen Targets
0.34Weak
acquired thrombocytopeniaOpen Targets
0.29Weak
hepatocellular carcinomaOpen Targets
0.29Weak
ovarian dysfunctionOpen Targets
0.28Weak
hypertrophic cardiomyopathyOpen Targets
0.26Weak
sclerosing cholangitisOpen Targets
0.21Weak
medical procedureOpen Targets
0.19Weak
osteoarthritis, kneeOpen Targets
0.19Weak
type 2 diabetes mellitusOpen Targets
0.13Weak
diabetes mellitusOpen Targets
0.13Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets6
ALDAFERMINPhase II/III
FGFR4-KLB activator
sclerosing cholangitis
FAZPILODEMABPhase II
FGF1/KLB agonist
non-alcoholic fatty liver disease
MUPARFOSTATPhase III
Acidic fibroblast growth factor inhibitor
hepatocellular carcinoma
PEGBELFERMINPhase II
FGF1/KLB agonist
type 2 diabetes mellitus
SURAMINPhase II
Acidic fibroblast growth factor inhibitor
non-small cell lung carcinoma
SURAMIN HEXASODIUMApproved
Acidic fibroblast growth factor inhibitor
trypanosomiasis
Related Genes
FGFR1Protein interaction100%FGFR2Protein interaction100%NGFProtein interaction100%S100A13Protein interaction100%FGFR4Protein interaction100%EGFProtein interaction99%
Tissue Expression6 tissues
Heart
100%
Brain
81%
Lung
1%
Liver
1%
Ovary
0%
Bone Marrow
0%
Gene Interaction Network
Click a node to explore
FGF1FGFR1FGFR2NGFS100A13FGFR4EGF
PROTEIN STRUCTURE
Preparing viewer…
PDB1RG8 · 1.10 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.04LoF Tolerant
pLIⓘ
0.13Tolerant
Observed/Expected LoF0.50 [0.26–1.04]
RankingsWhere FGF1 stands among ~20K protein-coding genes
  • #1,441of 20,598
    Most Researched262 · top 10%
  • #817of 1,025
    FDA-Approved Drug Targets1
  • #10,370of 17,882
    Most Constrained (LOEUF)1.04
Genes detectedFGF1
Sources retrieved26 papers
Response time—
📄 Sources
26â–¼
1
FGF1.
PMID: 39074995
Differentiation · 2024
1.00
2
FGF1 and insulin control lipolysis by convergent pathways.
PMID: 34986332
Cell Metab · 2022
0.90
3
Colonic epithelial-derived FGF1 drives intestinal stem cell commitment toward goblet cells to suppress inflammatory bowel disease.
PMID: 40188210
Nat Commun · 2025
0.80
4
FGF1
PMID: 33762571
Signal Transduct Target Ther · 2021
0.70
5
Fibroblast Growth Factors for Nonalcoholic Fatty Liver Disease: Opportunities and Challenges.
PMID: 36902015
Int J Mol Sci · 2023
0.64