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GeneE
25 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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IGF2BP3
insulin like growth factor 2 mRNA binding protein 3
Chromosome 7 · 7p15.3
NCBI Gene: 10643Ensembl: ENSG00000136231.15HGNC: HGNC:28868UniProt: O00425
501PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Highly ConstrainedTransporter
RESEARCH IMPACT
Highly StudiedTrending
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
cytoplasmic stress granuleP-bodymRNA 3'-UTR bindingprotein bindingneurodegenerative diseasetype 2 diabetes mellitusdiabetes mellitusceliac disease
✦AI Summary

IGF2BP3 is an m6A-reader RNA-binding protein that stabilizes target mRNAs by recruiting them into cytoplasmic ribonucleoprotein complexes, protecting transcripts from degradation and modulating their translation 1. IGF2BP3 preferentially recognizes N6-methyladenosine-modified mRNAs and increases their stability 1, while also binding internal m7G modifications to promote transcript degradation in specific contexts 2. Clinically, IGF2BP3 drives multiple cancer-associated phenotypes through metabolic and epigenetic reprogramming. In hepatocellular carcinoma, lactylation of IGF2BP3 enhances its binding to PCK2 and NRF2 mRNAs, promoting lenvatinib resistance via antioxidant pathway activation 3. In non-small cell lung cancer, IGF2BP3 stabilizes COX6B2 mRNA in an m6A-dependent manner, increasing oxidative phosphorylation and conferring EGFR-TKI resistance 4. IGF2BP3 also promotes immune escape in breast cancer by stabilizing PD-L1 mRNA through METTL3-mediated m6A modification 5. Additionally, IGF2BP3 enhances lipid metabolism in cervical cancer by upregulating stearoyl-CoA desaturase through m6A-dependent mechanisms 6, promotes AML progression via IGF2BP3-SENP1-HDAC2-AKT signaling 7, and drives lung cancer metastasis by stabilizing MCM5 mRNA to activate Notch signaling 8. These findings establish IGF2BP3 as a critical oncogenic regulator linking epitranscriptomic modifications to metabolic reprogramming and therapeutic resistance.

Sources cited
1
IGF2BP3 preferentially binds N6-methyladenosine-containing mRNAs and increases their stability
PMID: 29476152
2
Lactylated IGF2BP3 stabilizes PCK2 and NRF2 mRNAs to promote lenvatinib resistance in HCC
PMID: 39450426
3
IGF2BP3 stabilizes COX6B2 mRNA in m6A-dependent manner to increase OXPHOS and EGFR-TKI resistance
PMID: 37061993
4
METTL3/m6A/IGF2BP3 axis stabilizes PD-L1 mRNA to promote immune escape in breast cancer
PMID: 35197058
5
IGF2BP3 enhances lipid metabolism in cervical cancer by upregulating SCD through m6A-dependent mechanisms
PMID: 38355626
6
IGF2BP3 binds SENP1 3-UTR in m6A-dependent manner to activate AKT signaling in AML
PMID: 38822351
7
IGF2BP3 can preferentially bind internal mRNA m7G and promote degradation of m7G target transcripts
PMID: 39198433
8
IGF2BP3 stabilizes MCM5 mRNA in m6A-dependent manner to activate Notch signaling and promote lung cancer metastasis
PMID: 37171793
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.54Moderate
type 2 diabetes mellitusOpen Targets
0.42Moderate
diabetes mellitusOpen Targets
0.33Weak
celiac diseaseOpen Targets
0.31Weak
alcohol drinkingOpen Targets
0.18Weak
Abruptio PlacentaeOpen Targets
0.13Weak
hepatocellular carcinomaOpen Targets
0.12Weak
neoplasmOpen Targets
0.12Weak
urinary bladder carcinomaOpen Targets
0.11Weak
lung adenocarcinomaOpen Targets
0.11Weak
gliomaOpen Targets
0.11Weak
Primary microcephalyOpen Targets
0.11Weak
gastric cancerOpen Targets
0.11Weak
acute myeloid leukemiaOpen Targets
0.11Weak
cancerOpen Targets
0.11Weak
triple-negative breast cancerOpen Targets
0.10Weak
breast cancerOpen Targets
0.10Weak
nasopharyngeal carcinomaOpen Targets
0.10Weak
colorectal carcinomaOpen Targets
0.10Weak
melanomaOpen Targets
0.10Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
IGF2Protein interaction99%YTHDC1Protein interaction95%METTL3Protein interaction95%YBX1Protein interaction94%ZC3H13Protein interaction93%METTL14Protein interaction93%
Tissue Expression6 tissues
Lung
100%
Bone Marrow
76%
Brain
51%
Ovary
41%
Liver
38%
Heart
0%
Gene Interaction Network
Click a node to explore
IGF2BP3IGF2YTHDC1METTL3YBX1ZC3H13METTL14
PROTEIN STRUCTURE
Preparing viewer…
PDB6FQ1 · 1.31 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.20Highly Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.09 [0.05–0.20]
RankingsWhere IGF2BP3 stands among ~20K protein-coding genes
  • #532of 20,598
    Most Researched501 · top 5%
  • #423of 17,882
    Most Constrained (LOEUF)0.20 · top 5%
Genes detectedIGF2BP3
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
Lactylation-Driven IGF2BP3-Mediated Serine Metabolism Reprogramming and RNA m6A-Modification Promotes Lenvatinib Resistance in HCC.
PMID: 39450426
Adv Sci (Weinh) · 2024
1.00
2
METTL3/IGF2BP3 axis inhibits tumor immune surveillance by upregulating N
PMID: 35197058
Mol Cancer · 2022
0.90
3
Metabolic Reprogramming Driven by IGF2BP3 Promotes Acquired Resistance to EGFR Inhibitors in Non-Small Cell Lung Cancer.
PMID: 37061993
Cancer Res · 2023
0.80
4
N
PMID: 32444598
Nat Commun · 2020
0.70
5
N6-Methyladenosine modification activates the serine synthesis pathway to mediate therapeutic resistance in liver cancer.
PMID: 39489921
Mol Ther · 2024
0.68