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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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PDE4B
phosphodiesterase 4B
Chromosome 1 · 1p31.3
NCBI Gene: 5142Ensembl: ENSG00000184588.18HGNC: HGNC:8781UniProt: Q07343
114PubMed Papers
20Diseases
28Drugs
0Pathogenic Variants
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
cAMP bindingprotein binding3',5'-cyclic-AMP phosphodiesterase activitypositive regulation of type II interferon productionasthmachronic obstructive pulmonary diseasepsoriasisatopic eczema
✦AI Summary

PDE4B encodes phosphodiesterase 4B, an enzyme that hydrolyzes the second messenger cAMP, playing a crucial role in regulating various physiological processes 1. The primary function involves degrading cAMP to terminate cAMP-mediated signaling pathways, thereby controlling inflammatory and fibrotic responses 2. PDE4B shows preferential expression in lungs and is distinct from other PDE4 isoforms in its cellular effects - unlike PDE4D, PDE4B overexpression exhibits protective effects against oxidative stress and hypertrophy in cardiomyocytes without affecting CREB-SIRT1 pathways 3. The enzyme is significantly involved in inflammatory diseases, with PDE4B-expressing macrophages infiltrating colonic mucosae in pediatric inflammatory bowel disease 4. Therapeutically, PDE4B represents a promising target for treating pulmonary fibrosis and other fibro-inflammatory conditions. Selective PDE4B inhibitors like nerandomilast (BI 1015550) demonstrate antifibrotic effects by inhibiting myofibroblast transformation, reducing extracellular matrix protein expression, and improving lung function parameters in preclinical models 15. These inhibitors show improved tolerability compared to pan-PDE4 inhibitors while maintaining anti-inflammatory and antifibrotic efficacy 6. Genome-wide association studies have also implicated PDE4B in neuropsychiatric conditions, including suicide attempt risk 7.

Sources cited
1
PDE4B hydrolyzes cAMP and shows preferential enzymatic inhibition, with therapeutic potential in pulmonary fibrosis
PMID: 35517783
2
PDE4B inhibition by nerandomilast improves lung function and reverses fibrosis-related gene expression changes
PMID: 39183442
3
PDE4B overexpression has protective effects against oxidative stress and hypertrophy, distinct from PDE4D effects
PMID: 40015131
4
PDE4B-expressing macrophages infiltrate colonic mucosae in pediatric inflammatory bowel disease
PMID: 31730855
5
Nerandomilast inhibits myofibroblast contractility and differentiation through multiple signaling pathways
PMID: 40239038
6
PDE4B inhibitors show improved tolerability while maintaining anti-inflammatory and antifibrotic effects
PMID: 36813290
7
PDE4B is implicated in suicide attempt risk through genome-wide association studies
PMID: 37777856
Disease Associationsⓘ20
asthmaOpen Targets
0.61Moderate
chronic obstructive pulmonary diseaseOpen Targets
0.60Moderate
psoriasisOpen Targets
0.60Moderate
atopic eczemaOpen Targets
0.59Moderate
psoriatic arthritisOpen Targets
0.58Moderate
Airway obstructionOpen Targets
0.58Moderate
coronary artery diseaseOpen Targets
0.57Moderate
psoriasis vulgarisOpen Targets
0.56Moderate
strokeOpen Targets
0.54Moderate
chronic bronchitisOpen Targets
0.53Moderate
Behcet's syndromeOpen Targets
0.52Moderate
stress-related disorderOpen Targets
0.49Moderate
substance-related disorderOpen Targets
0.48Moderate
Eczematoid dermatitisOpen Targets
0.47Moderate
major depressive disorderOpen Targets
0.47Moderate
schizophreniaOpen Targets
0.47Moderate
anxiety disorderOpen Targets
0.47Moderate
dysuriaOpen Targets
0.46Moderate
Oral ulcerOpen Targets
0.46Moderate
smoking initiationOpen Targets
0.46Moderate
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets28
AMINOPHYLLINEApproved
Adenosine receptor antagonist
asthma
AMLEXANOXApproved
Phosphodiesterase 4 inhibitor
APREMILASTApproved
Phosphodiesterase 4 inhibitor
psoriasis
CILOMILASTPhase III
Phosphodiesterase 4 inhibitor
bronchitis
CRISABOROLEApproved
Phosphodiesterase 4 inhibitor
atopic eczema
DIFAMILASTPhase III
Phosphodiesterase 4 inhibitor
atopic eczema
DIPYRIDAMOLEApproved
3',5'-cyclic phosphodiesterase inhibitor
coronary artery disease
DOVRAMILASTPhase II
Phosphodiesterase 4 inhibitor
cutaneous lupus erythematosus
DROTAVERINEApproved
Phosphodiesterase 4 inhibitor
gastrointestinal disease
DYPHYLLINEApproved
Phosphodiesterase 4 inhibitor
ENSIFENTRINEApproved
Phosphodiesterase 3 inhibitor
FLAVOXATEApproved
Phosphodiesterase 4 inhibitor
dysuria
FLAVOXATE HYDROCHLORIDEApproved
Phosphodiesterase 4 inhibitor
urethritis
GSK-256066Phase II
Phosphodiesterase 4 inhibitor
asthma
HT-0712Phase II
Phosphodiesterase 4 inhibitor
Cognitive impairment
IBUDILASTApproved
Phosphodiesterase 10A inhibitor
Castleman disease
LOTAMILASTPhase II
Phosphodiesterase 4 inhibitor
atopic eczema
MK-0873Phase II
Phosphodiesterase 4 inhibitor
psoriasis vulgaris
OGLEMILASTPhase II
Phosphodiesterase 4 inhibitor
asthma
OXTRIPHYLLINEApproved
Adenosine receptor antagonist
Cough
PENTOXIFYLLINEApproved
Adenosine A2 receptor antagonist
cardiovascular disease
REVAMILASTPhase II
Phosphodiesterase 4 inhibitor
asthma
ROFLUMILASTApproved
Phosphodiesterase 4 inhibitor
chronic bronchitis
ROLIPRAMPhase II
Phosphodiesterase 4 inhibitor
multiple sclerosis
TETOMILASTPhase III
Phosphodiesterase 4 inhibitor
ulcerative colitis
THEOPHYLLINEApproved
Phosphodiesterase 4 inhibitor
asthma
TOFIMILASTPhase II
Phosphodiesterase 4 inhibitor
chronic obstructive pulmonary disease
TRANIMILASTPhase III
Phosphodiesterase 4 inhibitor
chronic obstructive pulmonary disease
Related Genes
DISC1Protein interaction100%NDE1Protein interaction98%PRKACAProtein interaction96%PRKACGProtein interaction96%PRKACBProtein interaction96%AMPD2Protein interaction95%
Tissue Expression6 tissues
Bone Marrow
100%
Brain
43%
Lung
15%
Heart
9%
Liver
4%
Ovary
2%
Gene Interaction Network
Click a node to explore
PDE4BDISC1NDE1PRKACAPRKACGPRKACBAMPD2
PROTEIN STRUCTURE
Preparing viewer…
PDB4KP6 · 1.50 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.37Moderately Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.24 [0.16–0.37]
RankingsWhere PDE4B stands among ~20K protein-coding genes
  • #4,159of 20,598
    Most Researched114 · top quartile
  • #108of 1,025
    FDA-Approved Drug Targets15 · top quartile
  • #1,759of 17,882
    Most Constrained (LOEUF)0.37 · top 10%
Genes detectedPDE4B
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
PDE4B inhibition by nerandomilast: Effects on lung fibrosis and transcriptome in fibrotic rats and on biomarkers in human lung epithelial cells.
PMID: 39183442
Br J Pharmacol · 2024
1.00
2
BI 1015550 is a PDE4B Inhibitor and a Clinical Drug Candidate for the Oral Treatment of Idiopathic Pulmonary Fibrosis.
PMID: 35517783
Front Pharmacol · 2022
0.90
3
PDE4D inhibition ameliorates cardiac hypertrophy and heart failure by activating mitophagy.
PMID: 40015131
Redox Biol · 2025
0.80
4
Phosphodiesterase 4B inhibition: a potential novel strategy for treating pulmonary fibrosis.
PMID: 36813290
Eur Respir Rev · 2023
0.70
5
Insights into the Cellular and Molecular Mechanisms behind the Antifibrotic Effects of Nerandomilast.
PMID: 40239038
Am J Respir Cell Mol Biol · 2025
0.60