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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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PDE4C
phosphodiesterase 4C
Chromosome 19 · 19p13.11
NCBI Gene: 5143Ensembl: ENSG00000105650.23HGNC: HGNC:8782UniProt: O43849
28PubMed Papers
20Diseases
28Drugs
0Pathogenic Variants
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
GO:00056153',5'-cyclic-AMP phosphodiesterase activitynegative regulation of cAMP/PKA signal transductionciliumasthmachronic obstructive pulmonary diseasepsoriasisatopic eczema
✦AI Summary

PDE4C (phosphodiesterase 4C) is a cyclic AMP-specific phosphodiesterase that hydrolyzes the second messenger cAMP, playing a crucial role in regulating intracellular signaling pathways 1. The gene is located on chromosome 19.1 and spans at least 38 kb with multiple alternatively spliced variants that show tissue-specific expression patterns, particularly in lung and testis 21. PDE4C functions as a negative regulator of cAMP/PKA signaling, with its activity directly impacting cellular processes including apoptosis, migration, and calcium homeostasis 34. In cancer contexts, PDE4C appears to function as a tumor suppressor, being downregulated through promoter hypermethylation in high-grade gliomas, where reduced expression correlates with poor prognosis and decreased overall survival 3. The enzyme's role extends to reproductive biology, where aberrant upregulation impairs endometrial decidualization by suppressing cAMP levels and FOXO1 expression, contributing to infertility in adenomyosis patients 4. Additionally, PDE4C serves as a therapeutic target in spinal cord injury, where its suppression by miR-615-3p activates the cAMP/PKA pathway, providing neuroprotective effects through improved calcium signaling and reduced endoplasmic reticulum stress 5.

Sources cited
1
PDE4C is a cyclic AMP-specific phosphodiesterase with multiple splice variants showing tissue-specific expression
PMID: 9349724
2
PDE4C gene is located on chromosome 19p13.1 and spans at least 38 kb with alternative promoters
PMID: 10574328
3
PDE4C functions as a tumor suppressor in gliomas, being downregulated through promoter hypermethylation
PMID: 24842301
4
PDE4C upregulation impairs endometrial decidualization by suppressing cAMP levels and FOXO1 expression
PMID: 39326465
5
PDE4C suppression activates cAMP/PKA pathway providing neuroprotective effects in spinal cord injury
PMID: 41526970
Disease Associationsⓘ20
asthmaOpen Targets
0.60Moderate
chronic obstructive pulmonary diseaseOpen Targets
0.60Moderate
psoriasisOpen Targets
0.59Moderate
atopic eczemaOpen Targets
0.59Moderate
psoriatic arthritisOpen Targets
0.58Moderate
Airway obstructionOpen Targets
0.58Moderate
psoriasis vulgarisOpen Targets
0.56Moderate
coronary artery diseaseOpen Targets
0.54Moderate
strokeOpen Targets
0.54Moderate
chronic bronchitisOpen Targets
0.53Moderate
Behcet's syndromeOpen Targets
0.52Moderate
Eczematoid dermatitisOpen Targets
0.47Moderate
dysuriaOpen Targets
0.46Moderate
Oral ulcerOpen Targets
0.46Moderate
cardiovascular diseaseOpen Targets
0.39Weak
prostatitisOpen Targets
0.39Weak
Castleman diseaseOpen Targets
0.37Weak
hypertensionOpen Targets
0.37Weak
irritable bowel syndromeOpen Targets
0.37Weak
PolyuriaOpen Targets
0.37Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets28
AMINOPHYLLINEApproved
Adenosine receptor antagonist
asthma
AMLEXANOXApproved
Phosphodiesterase 4 inhibitor
APREMILASTApproved
Phosphodiesterase 4 inhibitor
psoriasis
CILOMILASTPhase III
Phosphodiesterase 4 inhibitor
bronchitis
CRISABOROLEApproved
Phosphodiesterase 4 inhibitor
atopic eczema
DIFAMILASTPhase III
Phosphodiesterase 4 inhibitor
atopic eczema
DIPYRIDAMOLEApproved
3',5'-cyclic phosphodiesterase inhibitor
coronary artery disease
DOVRAMILASTPhase II
Phosphodiesterase 4 inhibitor
cutaneous lupus erythematosus
DROTAVERINEApproved
Phosphodiesterase 4 inhibitor
gastrointestinal disease
DYPHYLLINEApproved
Phosphodiesterase 4 inhibitor
ENSIFENTRINEApproved
Phosphodiesterase 3 inhibitor
FLAVOXATEApproved
Phosphodiesterase 4 inhibitor
dysuria
FLAVOXATE HYDROCHLORIDEApproved
Phosphodiesterase 4 inhibitor
urethritis
GSK-256066Phase II
Phosphodiesterase 4 inhibitor
asthma
HT-0712Phase II
Phosphodiesterase 4 inhibitor
Cognitive impairment
IBUDILASTApproved
Phosphodiesterase 10A inhibitor
Castleman disease
LOTAMILASTPhase II
Phosphodiesterase 4 inhibitor
atopic eczema
MK-0873Phase II
Phosphodiesterase 4 inhibitor
psoriasis vulgaris
OGLEMILASTPhase II
Phosphodiesterase 4 inhibitor
asthma
OXTRIPHYLLINEApproved
Adenosine receptor antagonist
Cough
PENTOXIFYLLINEApproved
Adenosine A2 receptor antagonist
cardiovascular disease
REVAMILASTPhase II
Phosphodiesterase 4 inhibitor
asthma
ROFLUMILASTApproved
Phosphodiesterase 4 inhibitor
chronic bronchitis
ROLIPRAMPhase II
Phosphodiesterase 4 inhibitor
multiple sclerosis
TETOMILASTPhase III
Phosphodiesterase 4 inhibitor
ulcerative colitis
THEOPHYLLINEApproved
Phosphodiesterase 4 inhibitor
asthma
TOFIMILASTPhase II
Phosphodiesterase 4 inhibitor
chronic obstructive pulmonary disease
TRANIMILASTPhase III
Phosphodiesterase 4 inhibitor
chronic obstructive pulmonary disease
Related Genes
PDE4AShared pathway100%PDE7AShared pathway100%ADCY5Protein interaction90%PKD2Protein interaction90%ALDH7A1Protein interaction80%PDE7BShared pathway67%
Tissue Expression6 tissues
Lung
100%
Ovary
55%
Liver
44%
Brain
15%
Heart
14%
Bone Marrow
0%
Gene Interaction Network
Click a node to explore
PDE4CPDE4APDE7AADCY5PKD2ALDH7A1PDE7B
PROTEIN STRUCTURE
Preparing viewer…
PDB2QYM · 1.90 Å · X-ray
View on RCSB ↗
RankingsWhere PDE4C stands among ~20K protein-coding genes
  • #12,414of 20,598
    Most Researched28
  • #110of 1,025
    FDA-Approved Drug Targets15 · top quartile
Genes detectedPDE4C
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Integrated analysis using methylation and gene expression microarrays reveals PDE4C as a prognostic biomarker in human glioma.
PMID: 24842301
Oncol Rep · 2014
1.00
2
Genomic organisation of the human cyclic AMP-specific phosphodiesterase PDE4C gene and its chromosomal localisation to 19p13.1, between RAB3A and JUND.
PMID: 10574328
Cell Signal · 1999
0.90
3
PDE4 subtypes in cancer.
PMID: 32203163
Oncogene · 2020
0.80
4
The plasma peptides of Alzheimer's disease.
PMID: 34182925
Clin Proteomics · 2021
0.70
5
Multiple splice variants of phosphodiesterase PDE4C cloned from human lung and testis.
PMID: 9349724
Biochim Biophys Acta · 1997
0.60