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GeneE
25 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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PTGER4
prostaglandin E receptor 4
Chromosome 5 · 5p13.1
NCBI Gene: 5734Ensembl: ENSG00000171522.7HGNC: HGNC:9596UniProt: A0PJF5
203PubMed Papers
20Diseases
4Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
RESEARCH IMPACT
Trending
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
negative regulation of eosinophil extravasationplasma membraneresponse to mechanical stimulusnegative regulation of integrin activationgastric carcinomaCrohn's diseaseautoimmune diseaseneurodegenerative disease
✦AI Summary

PTGER4 (prostaglandin E receptor 4) is a G-protein coupled receptor that mediates prostaglandin E2 (PGE2) signaling through adenylate cyclase activation 1. The receptor plays critical roles in intestinal homeostasis and immune regulation. In intestinal epithelial cells, PTGER4 activation suppresses necroptosis and promotes resolution of colitis, with EP4 expression correlating with improved inflammatory bowel disease outcomes 2. PTGER4-expressing intestinal macrophages drive mucosal healing by secreting CXCL1 via MAPK signaling, supporting epithelial regeneration during intestinal inflammation 3. During tumorigenesis, PTGER4 signaling promotes stem cell expansion through PGE2-induced YAP dephosphorylation and nuclear translocation, facilitating colorectal cancer initiation 1. In tumor microenvironments, PGE2-PTGER4 signaling impairs CD8+ T cell and macrophage immunity by downregulating metabolic pathways including oxidative phosphorylation and glycolysis 4. PTGER4 also mediates tumor cell-macrophage cross-talk in liver cancer 5. Additionally, PTGER4 participates in fetal immune tolerance mechanisms 6, and genetic variation upstream of PTGER4 associates with perianal fistula susceptibility in Crohn's disease 7. These findings establish PTGER4 as a pleiotropic regulator controlling epithelial repair, immune homeostasis, and cancer pathogenesis through PGE2 signaling.

Sources cited
1
PTGER4 mediates PGE2-driven YAP activation and Sca-1+ stem cell expansion in colorectal cancer initiation via adenylate cyclase signaling
PMID: 32322056
2
PTGER4 (EP4) on intestinal epithelial cells represses necroptosis and promotes resolution of colitis, with expression correlating to improved IBD outcomes
PMID: 34239062
3
PTGER4+ intestinal macrophages promote mucosal healing by secreting CXCL1 through MAPK signaling in response to PGE2
PMID: 33558271
4
PGE2-PTGER4 signaling in CD8+ T cells and macrophages impairs oxidative phosphorylation and MYC-dependent metabolic pathways in tumor microenvironment
PMID: 39487111
5
SPP1-PTGER4 interaction between tumor cells and macrophages is a stable ligand-receptor pair in liver cancer malignant ecosystems
PMID: 36476645
6
PTGES3/PTGER4 signaling pathway functions as a fetal immune tolerance mechanism during human immune system development
PMID: 41161316
7
Genetic loci upstream of PTGER4 associate with perianal fistula pathogenesis in Crohn's disease with population-specific differences
PMID: 38663404
8
PTGER4 mediates TFF3-stimulated colorectal cancer progression through PTGS2-derived PGE2 signaling
PMID: 34262017
Disease Associationsⓘ20
gastric carcinomaOpen Targets
0.45Moderate
Crohn's diseaseOpen Targets
0.44Moderate
autoimmune diseaseOpen Targets
0.36Weak
neurodegenerative diseaseOpen Targets
0.35Weak
allergic rhinitisOpen Targets
0.33Weak
pregnancyOpen Targets
0.32Weak
inflammatory bowel diseaseOpen Targets
0.32Weak
type 1 diabetes mellitusOpen Targets
0.32Weak
Eczematoid dermatitisOpen Targets
0.32Weak
neuroinflammatory disorderOpen Targets
0.31Weak
colorectal cancerOpen Targets
0.31Weak
ulcerative colitisOpen Targets
0.31Weak
asthmaOpen Targets
0.30Weak
respiratory system diseaseOpen Targets
0.30Weak
multiple sclerosisOpen Targets
0.29Weak
allergic diseaseOpen Targets
0.29Weak
psoriasisOpen Targets
0.29Weak
ankylosing spondylitisOpen Targets
0.28Weak
arthritisOpen Targets
0.28Weak
Prosthesis-Related InfectionsOpen Targets
0.28Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets4
DINOPROSTONEApproved
Prostaglandin E2 receptor agonist
GRAPIPRANTPhase II
Prostanoid EP4 receptor antagonist
Pain
RIVENPROSTPhase II
Prostanoid EP4 receptor agonist
bone fracture
VORBIPIPRANTPhase II
Prostanoid EP4 receptor antagonist
rheumatoid arthritis
Related Genes
GNG2Protein interaction100%COX3Protein interaction98%GNAI2Protein interaction95%GNB1Protein interaction90%GNAI3Protein interaction89%ARRB1Protein interaction87%
Tissue Expression6 tissues
Bone Marrow
100%
Lung
19%
Heart
8%
Liver
1%
Brain
1%
Ovary
1%
Gene Interaction Network
Click a node to explore
PTGER4GNG2COX3GNAI2GNB1GNAI3ARRB1
PROTEIN STRUCTURE
Preparing viewer…
PDB8GCP · 3.10 Å · EM
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.55Moderately Constrained
pLIⓘ
0.92Intolerant
Observed/Expected LoF0.33 [0.21–0.55]
RankingsWhere PTGER4 stands among ~20K protein-coding genes
  • #2,073of 20,598
    Most Researched203 · top quartile
  • #864of 1,025
    FDA-Approved Drug Targets1
  • #3,482of 17,882
    Most Constrained (LOEUF)0.55 · top quartile
Genes detectedPTGER4
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
Multiregional single-cell dissection of tumor and immune cells reveals stable lock-and-key features in liver cancer.
PMID: 36476645
Nat Commun · 2022
1.00
2
Paracrine orchestration of intestinal tumorigenesis by a mesenchymal niche.
PMID: 32322056
Nature · 2020
0.90
3
Prostaglandin E
PMID: 33558271
Gut · 2021
0.80
4
Systemic immune activity occurs during human immune system maturation.
PMID: 41161316
Cell · 2025
0.70
5
Multimodal single-cell analyses reveal mechanisms of perianal fistula in diverse patients with Crohn's disease.
PMID: 38663404
Med · 2024
0.60