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26 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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SGK1
serum/glucocorticoid regulated kinase 1
Chromosome 6 · 6q23.2
NCBI Gene: 6446Ensembl: ENSG00000118515.12HGNC: HGNC:10810UniProt: B7Z325
309PubMed Papers
20Diseases
0Drugs
1Pathogenic Variants
FUNCTIONAL ROLE
Kinase
RESEARCH IMPACT
Trending
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingnuclear speckintracellular signal transductionprotein serine/threonine/tyrosine kinase activitydiffuse large B-cell lymphomahair coloralcohol drinkingneurodegenerative disease
✦AI Summary

SGK1 (serum/glucocorticoid regulated kinase 1) is a serine/threonine kinase that plays critical roles in cellular stress response, ion transport regulation, and immune modulation 1. The kinase regulates multiple cellular processes including macrophage function, where dexamethasone upregulates SGK1 via glucocorticoid receptors, subsequently activating store-operated calcium entry (SOCE) and PIEZO1 channels, leading to calcium influx and cytoskeletal remodeling 1. In cardiac pathophysiology, SGK1 promotes fibrosis through the PI3Kγ/SGK1 pathway-dependent M2 macrophage polarization 2 and drives pathological cardiac hypertrophy through a novel noncanonical ERAD mechanism called ERAD-Out, where SGK1 itself becomes a degradation target 3. SGK1 demonstrates tumor suppressor activity in hepatocellular carcinoma metastasis by facilitating CD8+ T cell-mediated RIPK1-dependent necroptosis; loss of SGK1 enables immune evasion and metastatic colonization 4. In vascular pathology, SGK1 promotes smooth muscle cell phenotypic transformation in thoracic aortic dissection by phosphorylating SIRT6 at Ser338, leading to SIRT6 degradation and subsequent MMP9 upregulation 5. Additionally, SGK1 exacerbates inflammatory conditions including pulmonary fibrosis through H3K27ac-mediated macrophage reprogramming 6 and rheumatoid arthritis by promoting macrophage pyroptosis via Slc6a12 channels 7. SGK1 dysregulation is implicated in various cancers, making it a potential therapeutic target 8.

Sources cited
1
SGK1 is upregulated by dexamethasone via glucocorticoid receptors and activates SOCE and PIEZO1 channels
PMID: 38354960
2
SGK1 promotes cardiac fibrosis through PI3Kγ/SGK1 pathway-dependent M2 macrophage polarization
PMID: 37580750
3
SGK1 acts as tumor suppressor in HCC metastasis by facilitating CD8+ T cell-mediated necroptosis
PMID: 39892819
4
SGK1 promotes vascular smooth muscle cell phenotypic transformation by phosphorylating SIRT6 and regulating MMP9
PMID: 39633576
5
SGK1 drives pathological cardiac hypertrophy and is degraded through noncanonical ERAD-Out mechanism
PMID: 36317534
6
SGK1 exacerbates pulmonary fibrosis through H3K27ac-mediated macrophage reprogramming
PMID: 38250161
7
SGK1 promotes macrophage pyroptosis in rheumatoid arthritis via Slc6a12 channels
PMID: 38904021
8
SGK1 dysregulation is implicated in various cancers as potential therapeutic target
PMID: 33542904
Disease Associationsⓘ20
diffuse large B-cell lymphomaOpen Targets
0.51Moderate
hair colorOpen Targets
0.43Moderate
alcohol drinkingOpen Targets
0.42Moderate
neurodegenerative diseaseOpen Targets
0.37Weak
multiple myelomaOpen Targets
0.31Weak
hyperlipidemiaOpen Targets
0.29Weak
neuroinflammatory disorderOpen Targets
0.29Weak
ovarian neoplasmOpen Targets
0.28Weak
Abruptio PlacentaeOpen Targets
0.25Weak
bipolar disorderOpen Targets
0.24Weak
hyperpituitarismOpen Targets
0.24Weak
Varicose veinsOpen Targets
0.23Weak
papillary renal cell carcinomaOpen Targets
0.21Weak
response to stimulusOpen Targets
0.21Weak
COVID-19Open Targets
0.21Weak
cervical carcinomaOpen Targets
0.21Weak
vein disorderOpen Targets
0.21Weak
non-small cell lung carcinomaOpen Targets
0.21Weak
gastric adenocarcinomaOpen Targets
0.20Weak
esophageal squamous cell carcinomaOpen Targets
0.20Weak
Pathogenic Variants1
NM_001143676.3(SGK1):c.1379A>G (p.Asn460Ser)Likely pathogenic
Multiple myeloma
☆☆☆☆2019→ Residue 460
View on ClinVar ↗
Related Genes
PRR5Protein interaction100%NEDD4LProtein interaction100%FKBP5Protein interaction99%FOXO1Protein interaction98%C8orf44-SGK3Protein interaction98%RPTORProtein interaction97%
Tissue Expression6 tissues
Bone Marrow
100%
Ovary
80%
Lung
46%
Liver
31%
Brain
16%
Heart
16%
Gene Interaction Network
Click a node to explore
SGK1PRR5NEDD4LFKBP5FOXO1C8orf44-SGK3RPTOR
PROTEIN STRUCTURE
Preparing viewer…
PDB2R5T · 1.90 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.72LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.51 [0.36–0.72]
RankingsWhere SGK1 stands among ~20K protein-coding genes
  • #1,113of 20,598
    Most Researched309 · top 10%
  • #4,661of 5,498
    Most Pathogenic Variants1
  • #5,500of 17,882
    Most Constrained (LOEUF)0.72
Genes detectedSGK1
Sources retrieved26 papers
Response time—
📄 Sources
26▼
1
Dexamethasone upregulates macrophage PIEZO1 via SGK1, suppressing inflammation and increasing ROS and apoptosis.
PMID: 38354960
Biochem Pharmacol · 2024
1.00
2
TNFSF14/LIGHT promotes cardiac fibrosis and atrial fibrillation vulnerability via PI3Kγ/SGK1 pathway-dependent M2 macrophage polarisation.
PMID: 37580750
J Transl Med · 2023
0.90
3
Loss of SGK1 supports metastatic colonization in hepatocellular carcinoma by promoting resistance to T cell-mediated immunity.
PMID: 39892819
J Hepatol · 2025
0.80
4
High-salt-driven gut microbiota dysfunction aggravates prostatitis by promoting AHR/SGK1/FOXO1 axis-mediated Th17 cell differentiation.
PMID: 40383790
Mil Med Res · 2025
0.76
5
SGK1-Mediated Vascular Smooth Muscle Cell Phenotypic Transformation Promotes Thoracic Aortic Dissection Progression.
PMID: 39633576
Arterioscler Thromb Vasc Biol · 2025
0.70