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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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SGK3
serum/glucocorticoid regulated kinase family member 3
Chromosome 8 · 8q13.1
NCBI Gene: 23678Ensembl: ENSG00000104205.17HGNC: HGNC:10812UniProt: Q53EW6
76PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingprotein serine/threonine kinase activityintracellular signal transductionpotassium channel regulator activityneurodegenerative diseasepoisoningbenign prostatic hyperplasiaAlzheimer disease
✦AI Summary

SGK3 is a serine/threonine kinase that regulates ion channels, membrane transporters, and cellular signaling pathways with emerging roles in disease pathogenesis. Primary function: SGK3 phosphorylates and activates multiple ion channels (ENAC, KCNQ1, TRPV5/6) and nutrient transporters (NHE3, SLC34A2), regulating sodium, potassium, calcium, and phosphate homeostasis [UniProt]. Mechanism: SGK3 operates as a downstream effector of PI3K signaling, enabling AKT-independent mTORC1 activation and transcriptional reprogramming through phosphorylation of chr8 remodeling factors like BRG1 and transcription factors including STAT3 12. Disease relevance: SGK3 promotes vascular calcification in chr8 kidney disease by enhancing Pit-1 phosphate transporter expression and activity in vascular smooth muscle cells 3. In cancer, SGK3 drives estrogen receptor-positive breast cancer proliferation through STAT3/ZMIZ2-mediated β-catenin stabilization 4 and enables drug-tolerant persister survival following HER2 tyrosine kinase inhibitor exposure 1. SGK3 also sustains oncogenic signaling in PIK3CA-mutant colorectal tumors and regulates glucocorticoid-induced adipogenesis through chr8 remodeling 52. Clinical significance: SGK3 inhibition or genetic ablation shows promise in preventing obesity, vascular complications, and treatment resistance in hormone-driven cancers, positioning it as a therapeutic target across multiple disease contexts.

Sources cited
1
SGK3 enables AKT-independent mTORC1 activation in luminal-like drug-tolerant persisters after HER2 TKI exposure
PMID: 34911733
2
SGK3 promotes vascular calcification in CKD by enhancing Pit-1 expression and phosphate uptake in vascular smooth muscle cells
PMID: 38169564
3
SGK3 drives ER+ breast cancer proliferation through STAT3/ZMIZ2 pathway leading to β-catenin stabilization
PMID: 39876548
4
SGK3 sustains cPLA2 stability in PIK3CA-mutant colorectal tumors, promoting oncogenic paracrine signaling
PMID: 38614093
5
SGK3 mediates glucocorticoid-induced adipogenesis by phosphorylating BRG1 to promote chromatin remodeling
PMID: 40767604
6
Macrophage SGK3 promotes Ang II-induced cardiac remodeling through NLRP3/IL-1β pathway and mitochondrial oxidative stress
PMID: 39158709
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.34Weak
poisoningOpen Targets
0.28Weak
benign prostatic hyperplasiaOpen Targets
0.27Weak
Alzheimer diseaseOpen Targets
0.26Weak
lysosomal storage diseaseOpen Targets
0.24Weak
multiple sclerosisOpen Targets
0.24Weak
Parkinson diseaseOpen Targets
0.24Weak
neuroinflammatory disorderOpen Targets
0.16Weak
prostate cancerOpen Targets
0.12Weak
Familial prostate cancerOpen Targets
0.11Weak
ringed hair diseaseOpen Targets
0.10Weak
pili bifurcatiOpen Targets
0.10Weak
uncombable hair syndrome 3Open Targets
0.10Suggestive
wooly hair, autosomal recessive 3Open Targets
0.10Suggestive
uncombable hair syndromeOpen Targets
0.10Suggestive
hepatocellular carcinomaOpen Targets
0.09Suggestive
hypotrichosis simplexOpen Targets
0.09Suggestive
breast cancerOpen Targets
0.09Suggestive
hypotrichosis 4Open Targets
0.09Suggestive
chronic kidney diseaseOpen Targets
0.09Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
MYZAPShared pathway100%LRRC69Shared pathway100%DCDC2CShared pathway100%LRRC18Shared pathway100%ASB18Shared pathway100%LRRC30Shared pathway100%
Tissue Expression6 tissues
Bone Marrow
100%
Heart
34%
Liver
31%
Brain
16%
Ovary
15%
Lung
14%
Gene Interaction Network
Click a node to explore
SGK3MYZAPLRRC69DCDC2CLRRC18ASB18LRRC30
PROTEIN STRUCTURE
Preparing viewer…
PDB6EDX · 2.01 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.87LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.67 [0.53–0.87]
RankingsWhere SGK3 stands among ~20K protein-coding genes
  • #6,284of 20,598
    Most Researched76
  • #7,636of 17,882
    Most Constrained (LOEUF)0.87
Genes detectedSGK3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Autophagy in the physiological endometrium and cancer.
PMID: 32401642
Autophagy · 2021
1.00
2
Ontogeny and Vulnerabilities of Drug-Tolerant Persisters in HER2+ Breast Cancer.
PMID: 34911733
Cancer Discov · 2022
0.90
3
Arachidonic acid released by PIK3CA mutant tumor cells triggers malignant transformation of colonic epithelium by inducing chromatin remodeling.
PMID: 38614093
Cell Rep Med · 2024
0.80
4
SGK3 promotes vascular calcification via Pit-1 in chronic kidney disease.
PMID: 38169564
Theranostics · 2024
0.70
5
SGK3 deficiency in macrophages suppresses angiotensin II-induced cardiac remodeling via regulating Ndufa13-mediated mitochondrial oxidative stress.
PMID: 39158709
Cell Mol Life Sci · 2024
0.60