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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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SIK2
salt inducible kinase 2
Chromosome 11 · 11q23.1
NCBI Gene: 23235Ensembl: ENSG00000170145.6HGNC: HGNC:21680UniProt: Q9H0K1
81PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
magnesium ion bindingprotein phosphorylationintracellular signal transductionprotein autophosphorylationasthmaneuroinflammatory disorderneurodegenerative diseaselower respiratory tract disease
✦AI Summary

SIK2 (salt-inducible kinase 2) is a serine/threonine-protein kinase that regulates multiple metabolic and cellular processes. Primary functions include modulating fatty acid oxidation, autophagy, immune response, and glucose metabolism 12. SIK2 phosphorylates IRS1 in insulin-stimulated adipocytes, potentially modulating insulin signal transduction, and inhibits CREB activity by phosphorylating TORCs 3. The kinase also phosphorylates EP300 to inhibit its histone acetyltransferase activity, thereby regulating transcription factors like PPARA and MLXIPL 42. Mechanistically, SIK2 phosphorylates GABARAPL2 at Ser72 to facilitate autophagosome-lysosome fusion, critical for autophagic flux 5. Disease relevance is significant across multiple cancers: SIK2 mutations occur in lung adenocarcinoma 6; the LKB1-SIK2 module restrains uveal melanoma tumorigenesis, with SIK2 loss promoting proliferation 7; in renal cell carcinoma, FTO-mediated autophagy regulates SIK2 mRNA stability to promote progression 8; and in ovarian cancer, SIK2 enhances the Warburg effect and regulates lipid metabolism 9. Clinically, SIK2 inhibition shows promise: SIC-19, a novel SIK2 inhibitor, exhibits synthetic lethality with PARP inhibitors by impairing DNA homologous recombination repair 10, while SIK2 restoration mitigates Alzheimer's disease pathology 5.

Sources cited
1
SIK2 phosphorylates IRS1 in insulin-stimulated adipocytes, potentially modulating insulin signal transduction, and inhibits CREB activity by phosphorylating TORCs .
PMID: 15454081
2
Mechanistically, SIK2 phosphorylates GABARAPL2 at Ser72 to facilitate autophagosome-lysosome fusion, critical for autophagic flux .
PMID: 41126299
3
Disease relevance is significant across multiple cancers: SIK2 mutations occur in lung adenocarcinoma ; the LKB1-SIK2 module restrains uveal melanoma tumorigenesis, with SIK2 loss promoting proliferation ; in renal cell carcinoma, FTO-mediated autophagy regulates SIK2 mRNA stability to promote progression ; and in ovarian cancer, SIK2 enhances the Warburg effect and regulates lipid metabolism .
PMID: 22980975
4
Disease relevance is significant across multiple cancers: SIK2 mutations occur in lung adenocarcinoma ; the LKB1-SIK2 module restrains uveal melanoma tumorigenesis, with SIK2 loss promoting proliferation ; in renal cell carcinoma, FTO-mediated autophagy regulates SIK2 mRNA stability to promote progression ; and in ovarian cancer, SIK2 enhances the Warburg effect and regulates lipid metabolism .
PMID: 37966164
5
Disease relevance is significant across multiple cancers: SIK2 mutations occur in lung adenocarcinoma ; the LKB1-SIK2 module restrains uveal melanoma tumorigenesis, with SIK2 loss promoting proliferation ; in renal cell carcinoma, FTO-mediated autophagy regulates SIK2 mRNA stability to promote progression ; and in ovarian cancer, SIK2 enhances the Warburg effect and regulates lipid metabolism .
PMID: 36263177
6
Disease relevance is significant across multiple cancers: SIK2 mutations occur in lung adenocarcinoma ; the LKB1-SIK2 module restrains uveal melanoma tumorigenesis, with SIK2 loss promoting proliferation ; in renal cell carcinoma, FTO-mediated autophagy regulates SIK2 mRNA stability to promote progression ; and in ovarian cancer, SIK2 enhances the Warburg effect and regulates lipid metabolism .
PMID: 37317594
7
Clinically, SIK2 inhibition shows promise: SIC-19, a novel SIK2 inhibitor, exhibits synthetic lethality with PARP inhibitors by impairing DNA homologous recombination repair , while SIK2 restoration mitigates Alzheimer's disease pathology .
PMID: 38518726
Disease Associationsⓘ20
asthmaOpen Targets
0.50Moderate
neuroinflammatory disorderOpen Targets
0.37Weak
neurodegenerative diseaseOpen Targets
0.30Weak
lower respiratory tract diseaseOpen Targets
0.27Weak
adult onset asthmaOpen Targets
0.26Weak
respiratory system diseaseOpen Targets
0.25Weak
cardiovascular diseaseOpen Targets
0.25Weak
prostate carcinomaOpen Targets
0.23Weak
WheezingOpen Targets
0.23Weak
hypertensionOpen Targets
0.22Weak
autoimmune thyroid diseaseOpen Targets
0.18Weak
pernicious anemiaOpen Targets
0.18Weak
allergic rhinitisOpen Targets
0.17Weak
allergic diseaseOpen Targets
0.17Weak
mathematical abilityOpen Targets
0.16Weak
Eczematoid dermatitisOpen Targets
0.14Weak
corneal degenerationOpen Targets
0.13Weak
atopic eczemaOpen Targets
0.13Weak
deep vein thrombosisOpen Targets
0.11Weak
sclerosing cholangitisOpen Targets
0.11Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
CRTC2Protein interaction95%CRTC1Protein interaction95%PRKACAProtein interaction94%PRKACBProtein interaction91%PRKACGProtein interaction91%CREB1Protein interaction91%
Tissue Expression6 tissues
Liver
100%
Brain
77%
Heart
58%
Ovary
56%
Lung
54%
Bone Marrow
15%
Gene Interaction Network
Click a node to explore
SIK2CRTC2CRTC1PRKACAPRKACBPRKACGCREB1
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q9H0K1
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.41Moderately Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.30 [0.23–0.41]
RankingsWhere SIK2 stands among ~20K protein-coding genes
  • #5,898of 20,598
    Most Researched81
  • #2,153of 17,882
    Most Constrained (LOEUF)0.41 · top quartile
Genes detectedSIK2
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
The target landscape of clinical kinase drugs.
PMID: 29191878
Science · 2017
1.00
2
Mapping the hallmarks of lung adenocarcinoma with massively parallel sequencing.
PMID: 22980975
Cell · 2012
0.90
3
LKB1-SIK2 loss drives uveal melanoma proliferation and hypersensitivity to SLC8A1 and ROS inhibition.
PMID: 37966164
EMBO Mol Med · 2023
0.80
4
FTO-mediated autophagy promotes progression of clear cell renal cell carcinoma via regulating SIK2 mRNA stability.
PMID: 36263177
Int J Biol Sci · 2022
0.70
5
SIK2: A critical glucolipid metabolic reprogramming regulator and potential target in ovarian cancer.
PMID: 37317594
J Obstet Gynaecol Res · 2023
0.60