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10 sources retrieved Β· Most recent: April 2026 Β· Index updated 14 days ago
β“˜GeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
SIM2
SIM bHLH transcription factor 2
Chromosome 21 Β· 21q22.13
NCBI Gene: 6493Ensembl: ENSG00000159263.16HGNC: HGNC:10883UniProt: Q14190
67PubMed Papers
20Diseases
0Drugs
1Pathogenic Variants
FUNCTIONAL ROLE
Transcription Factor
DATA QUALITY
βœ“ Experimental GO Evidenceβœ“ Swiss-Prot Reviewed
nucleoplasmprotein bindingnuclear bodyRNA polymerase II transcription regulatory region sequence-specific DNA bindingAbnormality of the skeletal systemprostate carcinomagoutbone remodeling disease
✦AI Summary

SIM2 (SIM bHLH transcription factor 2) is a neuron-enriched basic helix-loop-helix/PAS domain transcription factor located within the Down syndrome critical region of chromosome 21 1. The gene encodes multiple isoforms including SIM2-s, a short splice variant 2. SIM2 functions as a master regulator of central nervous system development, showing spatial and temporal expression patterns in embryonic and fetal brain regions including the diencephalon, hippocampal formation, cortical cells, and cerebellar layers 3. The protein regulates transcription through DNA binding and dimerization with partner proteins, with its activity controlled by c-myb and other transcription factors 4. Functionally deficient SIM2 variants found in patients with neurological phenotypes exhibit impaired transcriptional activation, reduced DNA binding, and altered nuclear localization 5. Beyond neurological functions, SIM2 plays roles in cancer progression, promoting glioblastoma invasion through regulation of MMP-2 and TIMP-2 2, and serving as a predictive biomarker for chemoradiotherapy response in esophageal cancer 6. The gene is also involved in mammary gland differentiation, where it regulates STING activity during lactogenic development 7. SIM2 overexpression may contribute to Down syndrome pathogenesis, particularly mental retardation phenotypes 3.

Sources cited
1
SIM2 is located within Down syndrome critical region of chromosome 21 and encodes multiple isoforms
PMID: 9199934
2
SIM2-s short splice variant promotes glioblastoma invasion through MMP-2/TIMP-2 regulation
PMID: 20448453
3
SIM2 shows specific expression patterns in embryonic/fetal brain regions and may contribute to Down syndrome mental retardation
PMID: 15946822
4
SIM2 transcription is regulated by c-myb and other transcription factors through specific promoter elements
PMID: 11404025
5
Functionally deficient SIM2 variants in neurological patients show impaired transcriptional activity and protein function
PMID: 35730699
6
SIM2 regulates CD24 and CK4 expression and serves as predictive biomarker for esophageal cancer therapy
PMID: 32124945
7
SIM2 regulates STING activity during mammary gland lactogenic differentiation
PMID: 39399905
Disease Associationsβ“˜20
Abnormality of the skeletal systemOpen Targets
0.53Moderate
prostate carcinomaOpen Targets
0.50Moderate
goutOpen Targets
0.42Moderate
bone remodeling diseaseOpen Targets
0.32Weak
bilirubin metabolism diseaseOpen Targets
0.21Weak
protozoa infectious diseaseOpen Targets
0.18Weak
esophageal squamous cell carcinomaOpen Targets
0.10Suggestive
posterior cortical atrophyOpen Targets
0.06Suggestive
neoplasmOpen Targets
0.05Suggestive
cleft palateOpen Targets
0.05Suggestive
isolated congenital hypoglossia/aglossiaOpen Targets
0.05Suggestive
bronchopneumoniaOpen Targets
0.05Suggestive
prostate cancerOpen Targets
0.04Suggestive
cleft lipOpen Targets
0.04Suggestive
cleft lip/palateOpen Targets
0.04Suggestive
Lung AbscessOpen Targets
0.04Suggestive
breast ductal carcinoma in situOpen Targets
0.04Suggestive
van der Woude syndromeOpen Targets
0.04Suggestive
OligodontiaOpen Targets
0.04Suggestive
tooth agenesisOpen Targets
0.04Suggestive
Pathogenic Variants1
NM_005069.6(SIM2):c.461A>G (p.Tyr154Cys)Likely pathogenic
Neurodevelopmental with craniofacial anomalies disorder
β˜†β˜†β˜†β˜†2021β†’ Residue 154
View on ClinVar β†—
Related Genes
ARNTProtein interaction96%ARNT2Protein interaction90%SIM1Shared pathway67%NAGLUShared pathway50%CNTNAP3BShared pathway50%BARHL2Shared pathway50%
Tissue Expression6 tissues
Brain
100%
Liver
84%
Ovary
51%
Lung
38%
Heart
31%
Bone Marrow
0%
Gene Interaction Network
Click a node to explore
SIM2ARNTARNT2SIM1NAGLUCNTNAP3BBARHL2
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted Β· UniProt Q14190
View on AlphaFold β†—
Constraintβ“˜
LOEUFβ“˜
0.67LoF Tolerant
pLIβ“˜
0.00Tolerant
Observed/Expected LoF0.49 [0.36–0.67]
RankingsWhere SIM2 stands among ~20K protein-coding genes
  • #7,018of 20,598
    Most Researched67
  • #5,014of 5,498
    Most Pathogenic Variants1
  • #4,904of 17,882
    Most Constrained (LOEUF)0.67
Genes detectedSIM2
Sources retrieved10 papers
Response timeβ€”
πŸ“„ Sources
10β–Ό
1
Single minded 2-s (SIM2-s) gene is expressed in human GBM cells and involved in GBM invasion.
PMID: 20448453
Cancer Biol Ther Β· 2010
1.00
2
Loss of STING impairs lactogenic differentiation.
PMID: 39399905
Development Β· 2024
0.90
3
Molecular mechanisms of human single-minded 2 (SIM2) gene expression: identification of a promoter site in the SIM2 genomic sequence.
PMID: 11404025
Gene Β· 2001
0.80
4
Integrative epitranscriptomic and transcriptomic characterization in human colorectal cancer.
PMID: 40987397
J Adv Res Β· 2025
0.70
5
CD24 and CK4 are upregulated by SIM2, and are predictive biomarkers for chemoradiotherapy and surgery in esophageal cancer.
PMID: 32124945
Int J Oncol Β· 2020
0.60