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25 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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STK3
serine/threonine kinase 3
Chromosome 8 · 8q22.2
NCBI Gene: 6788Ensembl: ENSG00000104375.17HGNC: HGNC:11406UniProt: A0A087WZ06
185PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
RESEARCH IMPACT
Trending
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
negative regulation of canonical Wnt signaling pathwaycentrosomenucleusprotein kinase activityAlzheimer diseasehypotensionplacenta praeviabenign prostatic hyperplasia
✦AI Summary

STK3 (serine/threonine kinase 3) is a stress-activated, pro-apoptotic kinase that serves as a core component of the Hippo signaling pathway, a conserved regulator of organ size control and tumor suppression 1. Following caspase-cleavage, STK3 enters the nucleus to induce chr8 condensation and DNA fragmentation. Within the Hippo cascade, STK3 phosphorylates and activates LATS1/2 kinases, which subsequently phosphorylate and inactivate the YAP1 oncoprotein, preventing its nuclear translocation and suppressing genes promoting cell proliferation and survival 1. STK3 is required to repress proliferation of mature hepatocytes and inhibit tumor formation. Beyond canonical Hippo signaling, STK3 regulates centrosome disjunction through NEK2 phosphorylation and modulates mitophagy in adipocytes by regulating BNIP3, thereby controlling mitochondrial function and energy expenditure 2. In pancreatic cancer, STK3 methylation by PRMT5 at R461/R467 suppresses its autophosphorylation and kinase activity, inactivating Hippo signaling 3. Notably, in gastric cancer, STK3 functions as a YAP1 transcriptional target that activates Wnt/β-catenin signaling through GSK-3β phosphorylation, promoting stemness and chemoresistance 4. These context-dependent roles reveal STK3 as both a tumor suppressor and, under certain conditions, an oncogenic effector.

Sources cited
1
STK3/MST2 is a core kinase in the Hippo pathway cascade that regulates cell growth, organ size, and tumor suppression
PMID: 30566373
2
STK3 and STK4 suppress mitochondrial capacity in adipose tissues and regulate mitophagy through BNIP3 phosphorylation
PMID: 33758424
3
PRMT5-mediated methylation of STK3 (MST2) at R461/R467 suppresses its autophosphorylation and kinase activity in pancreatic cancer
PMID: 37905571
4
STK3 is a YAP1 transcriptional target that activates Wnt/β-catenin signaling through GSK-3β phosphorylation during gastric carcinogenesis
PMID: 40604818
⚠Limited data available — This gene has 4 indexed publications. Summary and analysis may be incomplete.
Disease Associationsⓘ20
Alzheimer diseaseOpen Targets
0.28Weak
hypotensionOpen Targets
0.25Weak
placenta praeviaOpen Targets
0.24Weak
benign prostatic hyperplasiaOpen Targets
0.24Weak
esophageal squamous cell carcinomaOpen Targets
0.08Suggestive
acute myeloid leukemiaOpen Targets
0.08Suggestive
ovarian cancerOpen Targets
0.08Suggestive
familial pancreatic carcinomaOpen Targets
0.06Suggestive
sarcomaOpen Targets
0.06Suggestive
melanomaOpen Targets
0.06Suggestive
Young adult-onset ParkinsonismOpen Targets
0.06Suggestive
episodic ataxia type 1Open Targets
0.05Suggestive
Spinocerebellar ataxia type 40Open Targets
0.05Suggestive
neoplasmOpen Targets
0.05Suggestive
spinocerebellar ataxia type 15/16Open Targets
0.05Suggestive
urocanic aciduriaOpen Targets
0.05Suggestive
atypical juvenile parkinsonismOpen Targets
0.05Suggestive
Malignant Pancreatic NeoplasmOpen Targets
0.05Suggestive
spinocerebellar ataxia type 20Open Targets
0.05Suggestive
gastric cancerOpen Targets
0.05Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
PPP2R1AProtein interaction100%PPP2R2DProtein interaction99%PPP2CAProtein interaction99%RASSF4Protein interaction98%RASSF6Protein interaction98%RASSF1Protein interaction97%
Tissue Expression6 tissues
Ovary
100%
Lung
72%
Liver
66%
Heart
63%
Brain
43%
Bone Marrow
19%
Gene Interaction Network
Click a node to explore
STK3PPP2R1APPP2R2DPPP2CARASSF4RASSF6RASSF1
PROTEIN STRUCTURE
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PDB4L0N · 1.40 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.06LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.80 [0.61–1.06]
RankingsWhere STK3 stands among ~20K protein-coding genes
  • #2,337of 20,598
    Most Researched185 · top quartile
  • #10,730of 17,882
    Most Constrained (LOEUF)1.06
Genes detectedSTK3
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
The Hippo Pathway: Biology and Pathophysiology.
PMID: 30566373
Annu Rev Biochem · 2019
1.00
2
Glycogen accumulation and phase separation drives liver tumor initiation.
PMID: 34678143
Cell · 2021
0.90
3
TLR4 signalling via Piezo1 engages and enhances the macrophage mediated host response during bacterial infection.
PMID: 34112781
Nat Commun · 2021
0.80
4
STK3/STK4 signalling in adipocytes regulates mitophagy and energy expenditure.
PMID: 33758424
Nat Metab · 2021
0.70
5
ROS-induced cytosolic release of mitochondrial PGAM5 promotes colorectal cancer progression by interacting with MST3.
PMID: 39915446
Nat Commun · 2025
0.68