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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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TAS2R8
taste 2 receptor member 8
Chromosome 12 · 12p13.2
NCBI Gene: 50836Ensembl: ENSG00000121314.3HGNC: HGNC:14915UniProt: Q9NYW2
20PubMed Papers
10Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
bitter taste receptor activitydetection of chemical stimulus involved in sensory perception of bitter tasteprotein bindingmembraneovulationneoplasmneuroblastomaNijmegen breakage syndrome
✦AI Summary

TAS2R8 is a G-protein coupled bitter taste receptor that functions beyond gustatory perception in gastrointestinal and systemic homeostasis. In taste signaling, TAS2R8 mediates bitter compound recognition and activates downstream gustducin-dependent calcium mobilization cascades 1. Notably, TAS2R8 responds to diverse ligands including olive oil phenolics 2, anti-HIV protease inhibitors 3, and various pharmaceutical compounds 4. Extraorally, TAS2R8 is expressed in human skin with personalized, sex-dependent expression patterns 5. In gastric tissue, TAS2R8 promotes proton secretion and protects against excessive cadmium accumulation through metal ion transporter regulation, suggesting a role in gastric physiology and xenobiotic homeostasis 6. In neuroblastoma, TAS2R8 exhibits anti-cancer properties by suppressing cancer stem cell markers (DLK1, CD133, Notch1, Sox2), inhibiting cell invasion and migration, and reducing hypoxia-inducible factor-1α signaling 7. TAS2R8 expression is zinc-dependent, regulated through CTCF transcription factor binding in response to intracellular zinc availability 8. These findings establish TAS2R8 as a chemosensory receptor with pleiotropic functions in taste perception, gastrointestinal physiology, metal homeostasis, and cancer biology.

Sources cited
1
TAS2R8 promotes proton secretion and protects against cadmium accumulation in gastric cells through metal ion transporter regulation
PMID: 41009725
2
TAS2R8 suppresses cancer stem cell markers and inhibits neuroblastoma cell invasion and tumorigenicity
PMID: 28467517
3
S6821 and S7958 are approved selective TAS2R8 antagonists that block TAS2R8-mediated bitterness
PMID: 32330040
4
Ritonavir activates TAS2R8 among other bitter taste receptors
PMID: 37625013
5
TAS2R8 promoter activity is zinc-dependent and regulated by CTCF transcription factor binding
PMID: 33071257
6
TAS2R8 activates calcium mobilization cascades and can be screened using genetically encoded calcium sensors
PMID: 31278864
7
TAS2R8 is expressed in human skin with sex-dependent expression patterns
PMID: 30332676
8
Seven out of twelve olive oil phenolic compounds activate TAS2R8, with oleuropein and ligstroside aglycons as potent activators
PMID: 34785711
Disease Associationsⓘ10
ovulationOpen Targets
0.02Suggestive
neoplasmOpen Targets
0.02Suggestive
neuroblastomaOpen Targets
0.01Suggestive
Nijmegen breakage syndromeOpen Targets
0.01Suggestive
cancerOpen Targets
0.01Suggestive
papillary thyroid carcinomaOpen Targets
0.00Suggestive
gliomaOpen Targets
0.00Suggestive
oral squamous cell carcinomaOpen Targets
0.00Suggestive
asthmaOpen Targets
0.00Suggestive
Parkinson diseaseOpen Targets
0.00Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
TAS2R60Shared pathway100%TAS2R36Shared pathway100%TAS2R33Shared pathway100%TAS2R50Shared pathway100%TAS2R20Shared pathway100%TAS2R19Shared pathway100%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
0%
Ovary
0%
Heart
0%
Liver
0%
Lung
0%
Gene Interaction Network
Click a node to explore
TAS2R8TAS2R60TAS2R36TAS2R33TAS2R50TAS2R20TAS2R19
PROTEIN STRUCTURE
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AlphaFoldAI-predicted · UniProt Q9NYW2
View on AlphaFold ↗
RankingsWhere TAS2R8 stands among ~20K protein-coding genes
  • #14,284of 20,598
    Most Researched20
Genes detectedTAS2R8
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Bitter Taste Receptors TAS2R8 and TAS2R10 Reduce Proton Secretion and Differentially Modulate Cadmium Uptake in Immortalized Human Gastric Cells.
PMID: 41009725
Int J Mol Sci · 2025
1.00
2
Anti-cancer stemness and anti-invasive activity of bitter taste receptors, TAS2R8 and TAS2R10, in human neuroblastoma cells.
PMID: 28467517
PLoS One · 2017
0.90
3
Discovery and Development of S6821 and S7958 as Potent TAS2R8 Antagonists.
PMID: 32330040
J Med Chem · 2020
0.80
4
Anti-HIV drugs lopinavir/ritonavir activate bitter taste receptors.
PMID: 37625013
Chem Senses · 2023
0.70
5
Intracellular zinc-dependent TAS2R8 gene expression through CTCF activation.
PMID: 33071257
Biomed Res · 2020
0.60