HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
TIGAR
TP53 induced glycolysis regulatory phosphatase
Chromosome 12 · 12p13.32
NCBI Gene: 57103Ensembl: ENSG00000078237.8HGNC: HGNC:1185UniProt: Q9NQ88
97PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
positive regulation of hexokinase activitycytosolnucleuscytoplasmdiabetes mellitustype 2 diabetes mellitusdiabetic eye diseasecellulitis
✦AI Summary

TIGAR (TP53 induced glycolysis regulatory phosphatase) is a p53-inducible enzyme that functions as a fructose-2,6-bisphosphatase, playing a dual role in metabolic regulation and cellular protection. Its primary function involves inhibiting glycolysis by hydrolyzing fructose-2,6-bisphosphate, thereby redirecting glucose flux toward the pentose phosphate pathway (PPP) to generate NADPH and ribose 1. This metabolic reprogramming reduces intracellular reactive oxygen species and enhances DNA repair capacity 2. TIGAR expression is transcriptionally regulated by p53 family members and various transcription factors, with its activity being stress-responsive 1. Beyond its enzymatic function, TIGAR exhibits non-canonical roles through protein-protein interactions, including binding to TAK1 to promote inflammatory responses in sepsis 3 and regulating autophagy pathways through LRRK2-mediated mechanisms in adipocytes 4. In disease contexts, TIGAR demonstrates complex roles: it can be protective by reducing oxidative stress in cardiovascular and neurological conditions 2, yet promotes tumor survival and chemoresistance by enhancing PPP flux and DNA repair in cancer cells 5. TIGAR's involvement in metabolic reprogramming makes it a potential therapeutic target for obesity, cancer, and inflammatory diseases, though its dual protective and pathogenic functions require careful consideration in therapeutic applications.

Sources cited
1
TIGAR functions as fructose-2,6-bisphosphatase, inhibits glycolysis, promotes PPP flux, and is regulated by p53 family members
PMID: 33510458
2
TIGAR is part of PPARγ-p53 transcriptional complex involved in DNA repair and vascular protection
PMID: 33322916
3
TIGAR binds TAK1 to promote inflammatory responses in sepsis through non-enzymatic function
PMID: 38773142
4
TIGAR regulates autophagy through LRRK2-mediated mechanisms in adipocytes and contributes to obesity
PMID: 38686804
5
TIGAR promotes cancer cell survival and chemoresistance by enhancing PPP flux and providing metabolic advantages
PMID: 30284488
Disease Associationsⓘ20
diabetes mellitusOpen Targets
0.53Moderate
type 2 diabetes mellitusOpen Targets
0.40Weak
diabetic eye diseaseOpen Targets
0.36Weak
cellulitisOpen Targets
0.27Weak
cervical carcinomaOpen Targets
0.27Weak
neoplasmOpen Targets
0.11Weak
cancerOpen Targets
0.11Weak
hepatocellular carcinomaOpen Targets
0.10Weak
gliomaOpen Targets
0.10Suggestive
nasopharyngeal carcinomaOpen Targets
0.09Suggestive
acute myeloid leukemiaOpen Targets
0.09Suggestive
colorectal carcinomaOpen Targets
0.09Suggestive
esophageal squamous cell carcinomaOpen Targets
0.09Suggestive
leukemiaOpen Targets
0.09Suggestive
colorectal cancerOpen Targets
0.09Suggestive
non-small cell lung carcinomaOpen Targets
0.09Suggestive
cervical cancerOpen Targets
0.08Suggestive
lung cancerOpen Targets
0.08Suggestive
gastric cancerOpen Targets
0.08Suggestive
carcinomaOpen Targets
0.08Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
TP53Protein interaction98%PFKMProtein interaction98%HK2Protein interaction98%PFKFB3Protein interaction97%PFKFB2Protein interaction97%PFKFB4Protein interaction97%
Tissue Expression6 tissues
Brain
100%
Lung
69%
Liver
38%
Ovary
11%
Heart
10%
Bone Marrow
2%
Gene Interaction Network
Click a node to explore
TIGARTP53PFKMHK2PFKFB3PFKFB2PFKFB4
PROTEIN STRUCTURE
Preparing viewer…
PDB3DCY · 1.75 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.19LoF Tolerant
pLIⓘ
0.13Tolerant
Observed/Expected LoF0.52 [0.26–1.19]
RankingsWhere TIGAR stands among ~20K protein-coding genes
  • #4,970of 20,598
    Most Researched97 · top quartile
  • #12,533of 17,882
    Most Constrained (LOEUF)1.19
Genes detectedTIGAR
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
ROS and Autophagy: Interactions and Molecular Regulatory Mechanisms.
PMID: 25722131
Cell Mol Neurobiol · 2015
1.00
2
Disruption of TIGAR-TAK1 alleviates immunopathology in a murine model of sepsis.
PMID: 38773142
Nat Commun · 2024
0.90
3
IDH2 stabilizes HIF-1α-induced metabolic reprogramming and promotes chemoresistance in urothelial cancer.
PMID: 36637036
EMBO J · 2023
0.80
4
TIGAR exacerbates obesity by triggering LRRK2-mediated defects in macroautophagy and chaperone-mediated autophagy in adipocytes.
PMID: 38686804
Autophagy · 2024
0.70
5
A systematic review of p53 regulation of oxidative stress in skeletal muscle.
PMID: 29298131
Redox Rep · 2018
0.60