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GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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TIPARP
TCDD inducible poly(ADP-ribose) polymerase
Chromosome 3 · 3q25.31
NCBI Gene: 25976Ensembl: ENSG00000163659.14HGNC: HGNC:23696UniProt: Q05BQ2
45PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Highly Constrained
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
cis-regulatory region sequence-specific DNA bindingNAD+-protein mono-ADP-ribosyltransferase activityNAD+ poly-ADP-ribosyltransferase activitynucleusovarian carcinomaneurodegenerative diseaseovarian cancerovarian serous carcinoma
✦AI Summary

TIPARP (TCDD inducible poly(ADP-ribose) polymerase) is a mono-ADP-ribosyltransferase that catalyzes the transfer of single ADP-ribose units onto target proteins, specifically modifying glutamate, aspartate, and cysteine residues 1. The enzyme functions as a negative regulator of the aryl hydrocarbon receptor (AHR) through mono-ADP-ribosylation, inhibiting AHR's transcriptional activity 2. TIPARP also targets transcription factors like FRA1, where ADP-ribosylation prevents protein degradation and suppresses IRF1- and IRF3-dependent apoptotic pathways 1. The protein negatively regulates type I interferon signaling in cancer cells, and its inhibition restores nucleic acid sensing responses that can trigger antitumor immunity 3. TIPARP demonstrates antiviral properties against alphaviruses by promoting viral protein degradation through ubiquitination 4. Clinically, TIPARP expression is elevated in various pathological conditions including ischemic stroke, where it contributes to mitochondrial dysfunction and brain injury 5, and in glaucoma patients, where it regulates intraocular pressure through modulation of extracellular matrix proteins 6. These diverse functions make TIPARP a potential therapeutic target for stroke, cancer, and ocular diseases.

Sources cited
1
TIPARP is a cysteine-specific mono-ADP-ribosyltransferase that modifies FRA1 and regulates apoptotic pathways
PMID: 38011562
2
TIPARP negatively regulates type I interferon signaling and its inhibition triggers antitumor immunity
PMID: 34375612
3
TIPARP exhibits antiviral properties against alphaviruses through viral protein degradation
PMID: 37768084
4
TIPARP expression is elevated in ischemic stroke and contributes to mitochondrial dysfunction
PMID: 39547463
5
TIPARP regulates intraocular pressure and is upregulated in glaucoma patients
PMID: 36536086
Disease Associationsⓘ20
ovarian carcinomaOpen Targets
0.44Moderate
neurodegenerative diseaseOpen Targets
0.38Weak
ovarian cancerOpen Targets
0.36Weak
ovarian serous carcinomaOpen Targets
0.36Weak
urinary bladder cancerOpen Targets
0.35Weak
alcohol drinkingOpen Targets
0.32Weak
high grade ovarian serous adenocarcinomaOpen Targets
0.31Weak
Abruptio PlacentaeOpen Targets
0.30Weak
malignant epithelial tumor of ovaryOpen Targets
0.30Weak
breast cancerOpen Targets
0.29Weak
seborrheic keratosisOpen Targets
0.17Weak
skin neoplasmOpen Targets
0.16Weak
lysosomal storage diseaseOpen Targets
0.14Weak
Testicular Germ Cell TumorOpen Targets
0.13Weak
actinic keratosisOpen Targets
0.13Weak
neoplasmOpen Targets
0.09Suggestive
cancerOpen Targets
0.08Suggestive
infectionOpen Targets
0.08Suggestive
primary ovarian insufficiencyOpen Targets
0.08Suggestive
46,XX gonadal dysgenesisOpen Targets
0.08Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
PARP16Protein interaction74%DAOAShared pathway25%ZNF410Shared pathway25%SFMBT2Shared pathway25%PARP11Shared pathway25%CNPY2Shared pathway25%
Tissue Expression6 tissues
Bone Marrow
100%
Brain
49%
Ovary
44%
Lung
37%
Heart
29%
Liver
21%
Gene Interaction Network
Click a node to explore
TIPARPPARP16DAOAZNF410SFMBT2PARP11CNPY2
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q05BQ2
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.35Highly Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.21 [0.14–0.35]
RankingsWhere TIPARP stands among ~20K protein-coding genes
  • #9,535of 20,598
    Most Researched45
  • #1,509of 17,882
    Most Constrained (LOEUF)0.35 · top 10%
Genes detectedTIPARP
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
New TIPARP inhibitor rescues mitochondrial function and brain injury in ischemic stroke.
PMID: 39547463
Pharmacol Res · 2024
1.00
2
Glucocorticoids, genes and brain function.
PMID: 29180230
Prog Neuropsychopharmacol Biol Psychiatry · 2018
0.90
3
PARP7-mediated ADP-ribosylation of FRA1 promotes cancer cell growth by repressing IRF1- and IRF3-dependent apoptosis.
PMID: 38011562
Proc Natl Acad Sci U S A · 2023
0.80
4
Integrative RNA profiling of TBEV-infected neurons and astrocytes reveals potential pathogenic effectors.
PMID: 35685361
Comput Struct Biotechnol J · 2022
0.70
5
Identification and characterization of human TIPARP gene within the CCNL amplicon at human chromosome 3q25.31.
PMID: 12851707
Int J Oncol · 2003
0.60