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25 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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TREM1
triggering receptor expressed on myeloid cells 1
Chromosome 6 · 6p21.1
NCBI Gene: 54210Ensembl: ENSG00000124731.14HGNC: HGNC:17760UniProt: K7EKM5
264PubMed Papers
20Diseases
1Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
RESEARCH IMPACT
Trending
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
transmembrane signaling receptor activitycell surfacescaffold protein bindingneutrophil-mediated killing of gram-negative bacteriumneurodegenerative diseaseneoplasmSepsiscancer
✦AI Summary

TREM1 (triggering receptor expressed on myeloid cells 1) is a cell surface immunoregulatory receptor expressed on neutrophils, monocytes, and tissue macrophages 1. TREM1 functions as an inflammatory amplifier that, upon activation by damage- and pathogen-associated molecular patterns, initiates downstream signaling cascades resulting in pro-inflammatory cytokine and chemokine production 1. In the brain, TREM1 becomes upregulated in microglia following injurious stimuli and synergistically amplifies inflammatory responses, contributing to neurocognitive disorders including diabetes-associated cognitive impairment 2. In diabetes-associated cognitive impairment, impaired microglial lipophagy causes lipid droplet accumulation that colocalizes with TREM1, promoting neuroinflammatory cascades via NLRP3 inflammasome activation 3. Pharmacological TREM1 blockade reduces neuroinflammation and improves cognitive function 3. In cancer, TREM1 overactivation in tumor-infiltrating myeloid cells promotes tumor progression and immunosuppression by expanding immunosuppressive myeloid-derived suppressor cells and driving T cell exhaustion 4. TREM1 inhibition enhances anti-PD-1 immunotherapy efficacy 4. Genetically, rs2062323 polymorphism in TREM1 associates with reduced Alzheimer's disease risk 5. These findings establish TREM1 as a promising therapeutic target for inflammation-associated diseases including cancer and neurodegeneration.

Sources cited
1
TREM1 is a cell surface receptor on myeloid cells functioning as an immunoregulator and inflammatory amplifier activated by DAMPs/PAMPs
PMID: 38749377
2
TREM1 is upregulated in microglia upon injury and amplifies inflammatory responses contributing to neurocognitive disorders
PMID: 39645047
3
In diabetes-associated cognitive impairment, impaired lipophagy causes TREM1 accumulation in microglia promoting neuroinflammation; TREM1 blockade improves cognition
PMID: 37204119
4
TREM1 promotes tumor progression through myeloid-derived suppressor cell expansion and T cell exhaustion; TREM1 inhibition enhances anti-PD-1 therapy
PMID: 37651197
5
TREM1 rs2062323 SNP associates with reduced Alzheimer's disease risk and elevated cerebrospinal fluid sTREM2
PMID: 36815315
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.24Weak
neoplasmOpen Targets
0.12Weak
SepsisOpen Targets
0.11Weak
cancerOpen Targets
0.11Weak
rheumatoid arthritisOpen Targets
0.11Weak
hepatocellular carcinomaOpen Targets
0.11Weak
liver diseaseOpen Targets
0.11Weak
glioblastoma multiformeOpen Targets
0.11Weak
gliomaOpen Targets
0.10Weak
Parkinson diseaseOpen Targets
0.10Weak
subarachnoid hemorrhageOpen Targets
0.10Suggestive
septic shockOpen Targets
0.10Suggestive
colitisOpen Targets
0.09Suggestive
Crohn's diseaseOpen Targets
0.09Suggestive
acute kidney injuryOpen Targets
0.09Suggestive
COVID-19Open Targets
0.08Suggestive
gastric cancerOpen Targets
0.08Suggestive
infectionOpen Targets
0.08Suggestive
papillary thyroid carcinomaOpen Targets
0.08Suggestive
psoriasisOpen Targets
0.08Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets1
NANGIBOTIDEPhase II
Triggering receptor expressed on myeloid cells 1 inhibitor
septic shock
Related Genes
TYROBPProtein interaction100%TREM2Protein interaction99%TREML1Protein interaction97%HMGB1Protein interaction96%TREML2Protein interaction95%PGLYRP1Protein interaction92%
Tissue Expression6 tissues
Lung
100%
Bone Marrow
89%
Brain
3%
Liver
3%
Heart
1%
Ovary
1%
Gene Interaction Network
Click a node to explore
TREM1TYROBPTREM2TREML1HMGB1TREML2PGLYRP1
PROTEIN STRUCTURE
Preparing viewer…
PDB1SMO · 1.47 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.02LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.67 [0.46–1.02]
RankingsWhere TREM1 stands among ~20K protein-coding genes
  • #1,428of 20,598
    Most Researched264 · top 10%
  • #10,099of 17,882
    Most Constrained (LOEUF)1.02
Genes detectedTREM1
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
Impaired lipophagy induced-microglial lipid droplets accumulation contributes to the buildup of TREM1 in diabetes-associated cognitive impairment.
PMID: 37204119
Autophagy · 2023
1.00
2
TREM1: Activation, signaling, cancer and therapy.
PMID: 38749377
Pharmacol Res · 2024
0.90
3
Alveolar macrophages: plasticity in a tissue-specific context.
PMID: 24445666
Nat Rev Immunol · 2014
0.80
4
Association of rs2062323 in the TREM1 gene with Alzheimer's disease and cerebrospinal fluid-soluble TREM2.
PMID: 36815315
CNS Neurosci Ther · 2023
0.70
5
Age-Associated Modulation of TREM1/2-Expressing Macrophages Promotes Melanoma Progression and Metastasis.
PMID: 40126543
Cancer Res · 2025
0.64