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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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UGT2A2
UDP glucuronosyltransferase family 2 member A2
Chromosome 4 · 4q13.3
NCBI Gene: 574537Ensembl: ENSG00000271271.6HGNC: HGNC:28183UniProt: P0DTE5
11PubMed Papers
13Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
bile acid metabolic processglucuronosyltransferase activityxenobiotic metabolic processresponse to symbionttricuspid valve diseaseAgeusiaAbnormality of the sense of smellplacental retention
✦AI Summary

UGT2A2 is a UDP-glucuronosyltransferase that catalyzes phase II biotransformation through glucuronidation, conjugating lipophilic substrates with glucuronic acid to enhance water solubility and facilitate excretion 1234. The enzyme is essential for eliminating and detoxifying drugs, xenobiotics, and endogenous compounds 24. UGT2A2 demonstrates high activity in bile acid glucuronidation, particularly for cholic acid-24G and chenodeoxycholic acid-24G formation with low micromolar affinity 4. It catalyzes estradiol glucuronidation 13 and contributes to detoxification of polycyclic aromatic hydrocarbons and other tobacco carcinogens 5. Notably, UGT2A2 is predominantly expressed in nasal mucosa 6, linking it to olfactory dysfunction. Genetic variants near UGT2A2 associate with anosmia in COVID-19 patients 78, while UGT2A2 expression is significantly downregulated in meningiomas of current smokers, suggesting altered xenobiotic metabolism in smoking-related cancers 9. The enzyme participates in glucuronidation of hydroxypropranolol metabolites alongside other UGTs 10, highlighting its broader role in drug metabolism.

Sources cited
1
UGT2A2 is a UDP-glucuronosyltransferase that catalyzes phase II biotransformation through glucuronidation, conjugating lipophilic substrates with glucuronic acid to enhance water solubility and facilitate excretion , , , .
PMID: 23756265
2
It catalyzes estradiol glucuronidation , and contributes to detoxification of polycyclic aromatic hydrocarbons and other tobacco carcinogens .
PMID: 23086198
3
Notably, UGT2A2 is predominantly expressed in nasal mucosa , linking it to olfactory dysfunction.
PMID: 30836059
4
Genetic variants near UGT2A2 associate with anosmia in COVID-19 patients , , while UGT2A2 expression is significantly downregulated in meningiomas of current smokers, suggesting altered xenobiotic metabolism in smoking-related cancers .
PMID: 37318677
5
The enzyme participates in glucuronidation of hydroxypropranolol metabolites alongside other UGTs , highlighting its broader role in drug metabolism.
PMID: 38067513
Disease Associationsⓘ13
tricuspid valve diseaseOpen Targets
0.32Weak
AgeusiaOpen Targets
0.32Weak
Abnormality of the sense of smellOpen Targets
0.31Weak
placental retentionOpen Targets
0.27Weak
response to statinOpen Targets
0.15Weak
smoking initiationOpen Targets
0.12Weak
Uterine leiomyomaOpen Targets
0.07Suggestive
uterine fibroidOpen Targets
0.07Suggestive
COVID-19Open Targets
0.01Suggestive
AnosmiaOpen Targets
0.01Suggestive
cancerOpen Targets
0.00Suggestive
hepatocellular carcinomaOpen Targets
0.00Suggestive
ovarian cancerOpen Targets
0.00Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
UGT2A3Shared pathway100%CYP1A1Protein interaction95%CYP2A13Protein interaction95%CYP3A4Protein interaction95%CYP19A1Protein interaction95%SULT1E1Protein interaction95%
Tissue Expression6 tissues
Lung
0%
Bone Marrow
0%
Ovary
0%
Heart
0%
Liver
0%
Brain
0%
Gene Interaction Network
Click a node to explore
UGT2A2UGT2A3CYP1A1CYP2A13CYP3A4CYP19A1SULT1E1
PROTEIN STRUCTURE
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AlphaFoldAI-predicted · UniProt P0DTE5
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.43LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF1.15 [0.93–1.43]
RankingsWhere UGT2A2 stands among ~20K protein-coding genes
  • #16,936of 20,598
    Most Researched11
  • #14,685of 17,882
    Most Constrained (LOEUF)1.43
Genes detectedUGT2A2
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
The Human UDP-glucuronosyltransferase UGT2A1 and UGT2A2 enzymes are highly active in bile acid glucuronidation.
PMID: 23756265
Drug Metab Dispos · 2013
1.00
2
Integrated clinical genomic analysis reveals xenobiotic metabolic genes are downregulated in meningiomas of current smokers.
PMID: 37318677
J Neurooncol · 2023
0.90
3
The Molecular Basis of Olfactory Dysfunction in COVID-19 and Long COVID.
PMID: 38749402
Lifestyle Genom · 2024
0.80
4
Functional and molecular characterization of UDP-glucuronosyltransferase 2 family in cynomolgus macaques.
PMID: 30836059
Biochem Pharmacol · 2019
0.70
5
Nomenclature update for the mammalian UDP glycosyltransferase (UGT) gene superfamily.
PMID: 16141793
Pharmacogenet Genomics · 2005
0.60