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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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ASGR1
asialoglycoprotein receptor 1
Chromosome 17 · 17p13.1
NCBI Gene: 432Ensembl: ENSG00000141505.13HGNC: HGNC:742UniProt: P07306
80PubMed Papers
20Diseases
2Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingimmune responseD-mannose bindingpattern recognition receptor activityHypercholesterolemiametabolic diseaseresponse to statinDisorder of lipid metabolism
✦AI Summary

ASGR1 (asialoglycoprotein receptor 1) is a hepatocyte-specific C-type lectin that primarily functions as a pattern recognition receptor mediating endocytosis and lysosomal degradation of asialoglycoproteins 12. The receptor binds specifically to N-acetylgalactosamine (GalNAc) residues in a calcium-dependent manner 2. ASGR1 plays a crucial role in cholesterol metabolism by regulating LXRα stability through mTORC1 and AMPK signaling pathways, ultimately promoting cholesterol excretion via ABCA1 and ABCG5/G8 transporters while inhibiting lipogenesis through SREBP1 suppression 1. The receptor also maintains liver homeostasis by facilitating lysosomal degradation of GP73, an endoplasmic reticulum stress mediator, with deficiency leading to increased hepatic injury 3. Beyond its hepatic functions, ASGR1 serves as an alternative SARS-CoV-2 receptor, enabling ACE2-independent viral entry 4. Disease relevance includes cardiovascular protection through cholesterol regulation, liver injury susceptibility, and potential roles in cancer progression 135. Therapeutically, ASGR1 represents a promising target for hypocholesterolemic drugs and cardiovascular disease prevention, with neutralizing antibodies showing efficacy in preclinical models 16.

Sources cited
1
ASGR1 mediates endocytosis and lysosomal degradation of asialoglycoproteins and regulates cholesterol metabolism through LXRα/AMPK/mTORC1 pathways
PMID: 35922515
2
ASGR1 is a hepatocyte-specific C-type lectin that binds N-acetylgalactosamine in a calcium-dependent manner
PMID: 32650396
3
ASGR1 maintains liver homeostasis by facilitating GP73 degradation and preventing endoplasmic reticulum stress-induced liver injury
PMID: 38459023
4
ASGR1 serves as an alternative functional receptor for SARS-CoV-2, enabling ACE2-independent viral entry
PMID: 34837059
5
ASGR1 shows abnormal expression patterns in multiple human cancers and correlates with prognosis
PMID: 36628237
6
ASGR1 represents a potential therapeutic target for heart failure prevention in chronic kidney disease patients
PMID: 38757788
Disease Associationsⓘ20
HypercholesterolemiaOpen Targets
0.50Moderate
metabolic diseaseOpen Targets
0.42Moderate
response to statinOpen Targets
0.35Weak
Disorder of lipid metabolismOpen Targets
0.34Weak
hyperlipidemiaOpen Targets
0.33Weak
familial hyperlipidemiaOpen Targets
0.32Weak
Insulin resistanceOpen Targets
0.11Weak
hepatocellular carcinomaOpen Targets
0.10Weak
atherosclerosisOpen Targets
0.08Suggestive
cardiovascular diseaseOpen Targets
0.08Suggestive
type 2 diabetes mellitusOpen Targets
0.08Suggestive
non-alcoholic fatty liver diseaseOpen Targets
0.08Suggestive
homozygous familial hypercholesterolemiaOpen Targets
0.07Suggestive
familial partial lipodystrophyOpen Targets
0.07Suggestive
HypertriglyceridemiaOpen Targets
0.07Suggestive
neoplasmOpen Targets
0.07Suggestive
isolated asymptomatic elevation of creatine phosphokinaseOpen Targets
0.06Suggestive
Immunodeficiency due to a late component of complements deficiencyOpen Targets
0.06Suggestive
Autoimmune HepatitisOpen Targets
0.05Suggestive
maleylacetoacetate isomerase deficiencyOpen Targets
0.05Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets2
VUPANORSENPhase II
Asialoglycoprotein receptor 1 binding agent
cardiovascular disease
VUPANORSEN SODIUMUNKNOWN
Angiopoietin like 3 (ANGPTL3) mRNA antisense inhibitor
hyperlipidemia
Related Genes
TGProtein interaction95%ALBProtein interaction91%ASGR2Protein interaction90%CERS2Protein interaction86%CLEC1BProtein interaction85%VWFProtein interaction84%
Tissue Expression6 tissues
Liver
100%
Bone Marrow
0%
Lung
0%
Brain
0%
Ovary
0%
Heart
0%
Gene Interaction Network
Click a node to explore
ASGR1TGALBASGR2CERS2CLEC1BVWF
PROTEIN STRUCTURE
Preparing viewer…
PDB9G76 · 1.20 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.32LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF1.00 [0.76–1.32]
RankingsWhere ASGR1 stands among ~20K protein-coding genes
  • #5,923of 20,598
    Most Researched80
  • #13,891of 17,882
    Most Constrained (LOEUF)1.32
Genes detectedASGR1
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Inhibition of ASGR1 decreases lipid levels by promoting cholesterol excretion.
PMID: 35922515
Nature · 2022
1.00
2
Deficiency of ASGR1 promotes liver injury by increasing GP73-mediated hepatic endoplasmic reticulum stress.
PMID: 38459023
Nat Commun · 2024
0.90
3
Plasma proteomic signatures of social isolation and loneliness associated with morbidity and mortality.
PMID: 39753750
Nat Hum Behav · 2025
0.80
4
Cholesterol metabolism: molecular mechanisms, biological functions, diseases, and therapeutic targets.
PMID: 41062796
Mol Biomed · 2025
0.70
5
Receptome profiling identifies KREMEN1 and ASGR1 as alternative functional receptors of SARS-CoV-2.
PMID: 34837059
Cell Res · 2022
0.60