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25 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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CDK5
cyclin dependent kinase 5
Chromosome 7 · 7q36.1
NCBI Gene: 1020Ensembl: ENSG00000164885.14HGNC: HGNC:1774UniProt: A0A090N7W4
463PubMed Papers
21Diseases
7Drugs
2Pathogenic Variants
FUNCTIONAL ROLE
Hub GeneKinase
RESEARCH IMPACT
Highly StudiedTrending
CLINICAL
Clinical TrialsOMIM Disease Gene
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
oligodendrocyte differentiationprotein serine/threonine kinase activitysignaling receptor inhibitor activityplasma membraneAlzheimer diseaseneurodegenerative diseaselissencephaly 7 with cerebellar hypoplasiaParkinson disease
✦AI Summary

CDK5 is a proline-directed serine/threonine kinase essential for neuronal development and function, activated uniquely by non-cyclin proteins p35 and p39 rather than classical cyclins 1. However, CDK5 also partners with cyclin B1 to maintain mitotic fidelity in dividing cells 2. In neurons, CDK5 regulates survival, migration, differentiation, axonal growth, synaptogenesis, and synaptic plasticity by phosphorylating key substrates including tau, MAP proteins, and small GTPases 3. CDK5 promotes cell survival through anti-apoptotic pathways and p53 stabilization, while protecting against DNA damage and oxidative stress 4. Dysregulation of CDK5 activity contributes to multiple neurodegenerative diseases. Pathological cleavage of p35 into p25 causes prolonged, aberrant CDK5 activation associated with tau hyperphosphorylation, cytoskeletal disruption, and neuronal death in Alzheimer's disease 5. Reduced CDK5 expression occurs in AD brain tissue, particularly in hippocampus and entorhinal cortex 6. Beyond neurodegeneration, astrocyte-induced CDK5 overexpression in brain metastases suppresses MHC-I expression, enabling immune evasion of cancer cells; CDK5 inhibition with roscovitine enhances checkpoint immunotherapy efficacy 7. Understanding CDK5 regulation and developing selective inhibitors represents a promising therapeutic strategy for neurodegenerative and cancer-related conditions.

Sources cited
1
CDK5 is active during mitosis and partners with cyclin B1 to maintain mitotic fidelity
PMID: 39232161
2
CDK5 governs neuronal/synaptic functions, circadian clocks, DNA damage responses, and cell cycle reentry; aberrant CDK5 activity is common in neurodegenerative diseases
PMID: 34814918
3
CDK5 is activated by p35 and p39 rather than classical cyclins; recent evidence shows CDK5 can interact with certain cyclins
PMID: 28077789
4
CDK5 regulates synaptic plasticity, neurotransmitter release, neuron migration, and neurite outgrowth; CDK5 overactivation mediates neuronal cell death through tau hyperphosphorylation and cytoskeletal disruption
PMID: 26601962
5
CDK5 expression is decreased in Alzheimer's disease brain samples, particularly in hippocampus and entorhinal cortex
PMID: 28714390
6
Astrocyte-induced CDK5 overexpression in brain metastases suppresses MHC-I expression to evade immune recognition; CDK5 inhibition enhances checkpoint immunotherapy efficacy
PMID: 39304713
7
Pathological cleavage of p35 into p25 causes prolonged CDK5 activation associated with neurodegeneration; CDK5 peptide inhibitors disrupt Cdk5/p25 interaction and protect against neurodegenerative phenotypes
PMID: 37043533
Disease Associationsⓘ21
Alzheimer diseaseOpen Targets
0.68Moderate
neurodegenerative diseaseOpen Targets
0.48Moderate
lissencephaly 7 with cerebellar hypoplasiaOpen Targets
0.40Weak
Parkinson diseaseOpen Targets
0.38Weak
neuroinflammatory disorderOpen Targets
0.37Weak
multiple sclerosisOpen Targets
0.35Weak
lysosomal storage diseaseOpen Targets
0.35Weak
chronic lymphocytic leukemiaOpen Targets
0.28Weak
lissencephaly with cerebellar hypoplasiaOpen Targets
0.19Weak
neoplasmOpen Targets
0.14Weak
non-small cell lung carcinomaOpen Targets
0.12Weak
small cell lung carcinomaOpen Targets
0.12Weak
hepatocellular carcinomaOpen Targets
0.11Weak
gastric cancerOpen Targets
0.11Weak
melanomaOpen Targets
0.11Weak
cancerOpen Targets
0.11Weak
breast cancerOpen Targets
0.11Weak
colorectal carcinomaOpen Targets
0.10Weak
lung cancerOpen Targets
0.10Weak
medullary thyroid gland carcinomaOpen Targets
0.10Weak
Lissencephaly 7, with cerebellar hypoplasiaUniProt
Pathogenic Variants2
NM_004935.4(CDK5):c.149G>A (p.Arg50Gln)Likely pathogenic
Lissencephaly 7 with cerebellar hypoplasia|Colon adenocarcinoma
★☆☆☆2023→ Residue 50
NM_004935.4(CDK5):c.580+1G>APathogenic
Lissencephaly 7 with cerebellar hypoplasia
☆☆☆☆2015
View on ClinVar ↗
Drug Targets7
AT-7519Phase II
Cyclin-dependent kinase inhibitor
chronic lymphocytic leukemia
AZD-5438Phase I
Cyclin-dependent kinase inhibitor
DINACICLIBPhase III
Cyclin-dependent kinase 2 inhibitor
PHA-793887Phase I
Cyclin-dependent kinase inhibitor
RGB-286638Phase I
Cyclin-dependent kinase 1 inhibitor
RONICICLIBPhase II
Cyclin-dependent kinase inhibitor
small cell lung carcinoma
SELICICLIBPhase II
Cyclin-dependent kinase 2 inhibitor
non-small cell lung carcinoma
Related Genes
CDK2Protein interaction100%CDKN1BProtein interaction100%CDKN1AProtein interaction100%CCNA1Protein interaction100%CCNA2Protein interaction100%BACE1Protein interaction100%
Tissue Expression6 tissues
Brain
100%
Liver
41%
Bone Marrow
37%
Heart
25%
Lung
22%
Ovary
12%
Gene Interaction Network
Click a node to explore
CDK5CDK2CDKN1BCDKN1ACCNA1CCNA2BACE1
PROTEIN STRUCTURE
Preparing viewer…
PDB4AU8 · 1.90 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.58Moderately Constrained
pLIⓘ
0.56Intermediate
Observed/Expected LoF0.39 [0.27–0.58]
RankingsWhere CDK5 stands among ~20K protein-coding genes
  • #582of 20,598
    Most Researched463 · top 5%
  • #4,198of 5,498
    Most Pathogenic Variants2
  • #3,919of 17,882
    Most Constrained (LOEUF)0.58 · top quartile
Genes detectedCDK5
Sources retrieved25 papers
Response time—
📄 Sources
25â–¼
1
CDK5-cyclin B1 regulates mitotic fidelity.
PMID: 39232161
Nature · 2024
1.00
2
Astrocyte-induced Cdk5 expedites breast cancer brain metastasis by suppressing MHC-I expression to evade immune recognition.
PMID: 39304713
Nat Cell Biol · 2024
0.90
3
Three decades of Cdk5.
PMID: 34814918
J Biomed Sci · 2021
0.80
4
Phosphorylation of USP32 by CDK5 regulates Rap1 stability and therapeutic resistance in pancreatic ductal adenocarcinoma.
PMID: 40379759
Oncogene · 2025
0.72
5
CDK5 and MAPT Gene Expression in Alzheimer's Disease Brain Samples.
PMID: 28714390
Curr Alzheimer Res · 2018
0.70