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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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CHRNA10
cholinergic receptor nicotinic alpha 10 subunit
Chromosome 11 · 11p15.4
NCBI Gene: 57053Ensembl: ENSG00000129749.3HGNC: HGNC:13800UniProt: C4IXS7
19PubMed Papers
20Diseases
2Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Ion ChannelReceptorTransporter
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
positive regulation of cytosolic calcium ion concentrationacetylcholine receptor signaling pathwayplasma membraneacetylcholine-gated monoatomic cation-selective channel activityTinnitusneurodegenerative diseasenephrotic syndromeAbnormal nasolacrimal system morphology
✦AI Summary

CHR11 encodes the cholinergic receptor nicotinic alpha-10 subunit, a component of neuronal acetylcholine receptors (nAChRs) that function as pentameric, ligand-gated cation channels with high calcium permeability 1. CHR11 forms heteropentameric channels with CHR11, particularly in the inner ear where these receptors mediate synaptic transmission between efferent olivocochlear fibers and cochlear hair cells, thereby modulating auditory stimuli and potentially protecting against acoustic trauma 12. Beyond the auditory system, CHR11 is expressed in immune cells including T-lymphocytes and B-lymphocytes, where it may regulate immune responses 2. In macrophages, unconventional α9* nAChRs containing CHR11 suppress ATP-mediated interleukin-1β release, suggesting anti-inflammatory functions 3. Age-related decline in CHR11 expression correlates with reduced nicotinic receptor conductance in vestibular hair cells and impaired balance in aged mice 4. Clinically, CHR11 variants associate with heroin addiction phenotypes, including duration of transition to dependence 5. Chr11 nicotine exposure downregulates CHR11 expression in human and rodent prefrontal cortex in a sex-dependent manner 6. These findings position CHR11 as a multifunctional receptor subunit relevant to auditory processing, immune regulation, vestibular function, and susceptibility to substance use disorders.

Sources cited
1
CHRNA10 molecular characterization, localization to chromosome 11p15.5, expression in inner ear and lymphoid tissues
PMID: 11350119
2
CHRNA10 expression in T-cells and B-cells; alpha9/10 nAChR involvement in auditory modulation
PMID: 15531379
3
CHRNA10-containing nAChRs suppress ATP-mediated IL-1β release in macrophages
PMID: 41221292
4
Age-related reduction in CHRNA10 expression and reduced nicotinic receptor conductance in vestibular hair cells
PMID: 36840917
5
CHRNA10 SNP variants associated with heroin addiction phenotypes
PMID: 35176404
6
Chronic nicotine exposure downregulates CHRNA10 expression in prefrontal cortex in sex-dependent manner
PMID: 36846236
Disease Associationsⓘ20
TinnitusOpen Targets
0.37Weak
neurodegenerative diseaseOpen Targets
0.32Weak
nephrotic syndromeOpen Targets
0.32Weak
Abnormal nasolacrimal system morphologyOpen Targets
0.27Weak
Alzheimer diseaseOpen Targets
0.26Weak
cancer painOpen Targets
0.07Suggestive
osteoarthritis, hipOpen Targets
0.02Suggestive
osteoarthritis, kneeOpen Targets
0.02Suggestive
hearing lossOpen Targets
0.01Suggestive
neoplasmOpen Targets
0.01Suggestive
experimental autoimmune encephalomyelitisOpen Targets
0.01Suggestive
AutoimmunityOpen Targets
0.00Suggestive
head and neck squamous cell carcinomaOpen Targets
0.00Suggestive
post-traumatic stress disorderOpen Targets
0.00Suggestive
nicotine dependenceOpen Targets
0.00Suggestive
Schnyder corneal dystrophyOpen Targets
0.00Suggestive
complete androgen insensitivity syndromeOpen Targets
0.00Suggestive
gastric cancerOpen Targets
0.00Suggestive
ovarian serous cystadenocarcinomaOpen Targets
0.00Suggestive
thyroid cancer, nonmedullary, 1Open Targets
0.00Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets2
NERAMEXANEPhase III
Neuronal acetylcholine receptor; alpha9/alpha10 antagonist
Alzheimer disease
NERAMEXANE MESYLATEPhase III
Neuronal acetylcholine receptor; alpha9/alpha10 antagonist
Tinnitus
Related Genes
CHRNA9Protein interaction89%CHATProtein interaction77%CHRNA1Protein interaction73%CHRNA5Protein interaction64%CHRNEShared pathway53%CHRNGShared pathway50%
Tissue Expression6 tissues
Liver
100%
Lung
94%
Ovary
66%
Heart
24%
Bone Marrow
19%
Brain
7%
Gene Interaction Network
Click a node to explore
CHRNA10CHRNA9CHATCHRNA1CHRNA5CHRNECHRNG
PROTEIN STRUCTURE
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AlphaFoldAI-predicted · UniProt Q9GZZ6
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.31LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.96 [0.72–1.31]
RankingsWhere CHRNA10 stands among ~20K protein-coding genes
  • #14,385of 20,598
    Most Researched19
  • #13,768of 17,882
    Most Constrained (LOEUF)1.31
Genes detectedCHRNA10
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Sex and diet-dependent gene alterations in human and rat brains with a history of nicotine exposure.
PMID: 36846236
Front Psychiatry · 2023
1.00
2
Molecular cloning and mapping of the human nicotinic acetylcholine receptor alpha10 (CHRNA10).
PMID: 11350119
Genomics · 2001
0.90
3
Characterization of the human nicotinic acetylcholine receptor subunit alpha (alpha) 9 (CHRNA9) and alpha (alpha) 10 (CHRNA10) in lymphocytes.
PMID: 15531379
Life Sci · 2004
0.80
4
Several nAChRs gene variants are associated with phenotypes of heroin addiction in Chinese Han population.
PMID: 35176404
Neurosci Lett · 2022
0.70
5
Dizziness genes.
PMID: 20552679
Am J Med Genet B Neuropsychiatr Genet · 2010
0.60