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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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GALR3
galanin receptor 3
Chromosome 22 · 22q13.1
NCBI Gene: 8484Ensembl: ENSG00000128310.4HGNC: HGNC:4134UniProt: O60755
25PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
positive regulation of transcription by RNA polymerase IIciliumprotein bindingpeptide hormone bindingcolitisneoplasmopen-angle glaucomahypertriglyceridemia 2
✦AI Summary

GALR3 is a G protein-coupled receptor that functions as a receptor for the neuropeptide galanin 1 and the novel peptide spexin-1 2. The receptor is widely distributed across tissues with highest expression in the hypothalamus and pituitary 1, as well as testis, adrenal gland, and pancreas 3. GALR3 couples to G-protein signaling pathways, specifically activating inward rectifying potassium (GIRK) channels 1, and signals predominantly through inhibition of adenylate cyclase 3, distinguishing it from GALR2 which activates phospholipase C. In the atrial context, spexin-GALR2 (not GALR3) signaling reduces atrial fibrillation susceptibility by suppressing CREB phosphorylation and downstream potassium channel regulation 4. GALR3 exhibits disease relevance in colorectal cancer, where elevated GALR3 immunoexpression in cancer tissue correlates with improved patient prognosis and longer overall survival 5. Additionally, GALR3 genetic variation associates with alcoholism risk 6, and GALR3 expression changes occur in polycystic ovary syndrome 7. These findings suggest GALR3 mediates diverse physiological processes including feeding behavior, nociception, and reproductive function.

Sources cited
1
GALR3 cloning, expression pattern in hypothalamus/pituitary, and coupling to GIRK channels
PMID: 9722565
2
Spexin as cognate ligand for GalR2 and GalR3 with pleotropic neuroendocrine functions
PMID: 29355530
3
Human GALR3 cloning, pharmacology, signaling through adenylate cyclase inhibition, tissue distribution
PMID: 9832121
4
GALR2 (not GALR3) mediates spexin effects on atrial fibrillation via CREB signaling
PMID: 38726666
5
Elevated GALR3 in colorectal cancer correlates with better prognosis and longer survival
PMID: 35409094
6
GALR3 genetic variation associates with alcoholism risk
PMID: 17083333
7
GALR3 expression changes in hypothalamus and ovary in polycystic ovary syndrome model
PMID: 36055012
Disease Associationsⓘ20
colitisOpen Targets
0.08Suggestive
neoplasmOpen Targets
0.05Suggestive
open-angle glaucomaOpen Targets
0.05Suggestive
hypertriglyceridemia 2Open Targets
0.05Suggestive
autism spectrum disorderOpen Targets
0.05Suggestive
colorectal carcinomaOpen Targets
0.04Suggestive
thyroid hormone metabolism, abnormal, 2Open Targets
0.04Suggestive
15q11q13 microduplication syndromeOpen Targets
0.04Suggestive
autismOpen Targets
0.04Suggestive
familial hypercholesterolemiaOpen Targets
0.04Suggestive
homozygous familial hypercholesterolemiaOpen Targets
0.04Suggestive
sitosterolemia 2Open Targets
0.03Suggestive
inflammatory bowel diseaseOpen Targets
0.03Suggestive
cancerOpen Targets
0.02Suggestive
gliomaOpen Targets
0.02Suggestive
polycystic ovary syndromeOpen Targets
0.01Suggestive
psoriasisOpen Targets
0.01Suggestive
colorectal cancerOpen Targets
0.01Suggestive
AnxietyOpen Targets
0.01Suggestive
diffuse large B-cell lymphomaOpen Targets
0.01Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
GALProtein interaction100%GALR1Protein interaction91%GCATProtein interaction90%SPXProtein interaction88%GALPProtein interaction82%UTS2RProtein interaction79%
Tissue Expression6 tissues
Liver
100%
Brain
29%
Ovary
29%
Bone Marrow
14%
Heart
0%
Lung
0%
Gene Interaction Network
Click a node to explore
GALR3GALGALR1GCATSPXGALPUTS2R
PROTEIN STRUCTURE
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AlphaFoldAI-predicted · UniProt O60755
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.82LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF1.07 [0.57–1.82]
RankingsWhere GALR3 stands among ~20K protein-coding genes
  • #12,982of 20,598
    Most Researched25
  • #16,679of 17,882
    Most Constrained (LOEUF)1.82
Genes detectedGALR3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Spexin Diminishes Atrial Fibrillation Vulnerability by Acting on Galanin Receptor 2.
PMID: 38726666
Circulation · 2024
1.00
2
Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels.
PMID: 9722565
J Biol Chem · 1998
0.90
3
Molecular characterization and expression of cloned human galanin receptors GALR2 and GALR3.
PMID: 9832121
J Neurochem · 1998
0.80
4
Galanin Receptors (GalR1, GalR2, and GalR3) Expression in Colorectal Cancer Tissue and Correlations to the Overall Survival and Poor Prognosis of CRC Patients.
PMID: 35409094
Int J Mol Sci · 2022
0.70
5
Levels of spexin and its receptors GALR2 and GALR3 in the hypothalamus and ovary of letrozole-induced polycystic ovary syndrome in rats.
PMID: 36055012
Biochem Biophys Res Commun · 2022
0.60