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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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GPR85
G protein-coupled receptor 85
Chromosome 7 · 7q31.1
NCBI Gene: 54329Ensembl: ENSG00000164604.15HGNC: HGNC:4536UniProt: A4D0T8
23PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
plasma membraneprotein bindingendoplasmic reticulumG protein-coupled receptor activitynervous system benign neoplasmmalunion fractureplacenta praeviaAbnormality of the skeletal system
✦AI Summary

GPR85 (SREB2) is a brain-enriched orphan G protein-coupled receptor located on human chromosome 7 1 that functions as a negative regulator of hippocampal adult neurogenesis and associated cognitive processes 2. The receptor is highly evolutionarily conserved across vertebrates 3 and shows predominant expression in the hippocampal dentate gyrus and other brain structures characterized by high neuroplasticity 3. GPR85 interacts with the postsynaptic density protein PSD-95 through its C-terminal PDZ-binding motif, positioning it within synaptic scaffolding complexes 4. Phylogenetic analysis suggests GPR85 may bind ATP, ADP, and UDP glucose 5. Functionally, GPR85 negatively regulates new neuron proliferation and survival in the dentate gyrus, with transgenic overexpression reducing cognitive performance in spatial discrimination and working memory tasks 2. GPR85 dysfunction is implicated in multiple CNS disorders, particularly schizophrenia 6 and autism spectrum disorder, where missense mutations cause aberrant receptor accumulation, endoplasmic reticulum stress, and impaired dendrite formation 4. Recent evidence also associates GPR85 with pain mechanisms 7. The receptor represents a promising therapeutic target for treating cognitive symptoms in psychiatric disorders through modulation of hippocampal neurogenesis.

Sources cited
1
GPR85 is a brain-enriched, evolutionarily conserved GPCR located on human chromosome 7q31
PMID: 10978537
2
GPR85 (SREB2) mRNA is highly conserved across mammalian species with abundant expression in hippocampal dentate gyrus and other plastic brain regions
PMID: 15893849
3
GPR85 negatively regulates hippocampal adult neurogenesis and associated cognitive functions including spatial discrimination and working memory
PMID: 22697179
4
GPR85 interacts with PSD-95 through its C-terminal PDZ-binding motif; mutations in ASD patients cause ER stress and impaired dendrite formation
PMID: 25780553
5
Phylogenetic analysis suggests GPR85 may bind ATP, ADP, and UDP glucose
PMID: 24503482
6
GPR85 is an orphan GPCR relevant to schizophrenia pathophysiology with potential for novel drug development
PMID: 37605621
7
GPR85 is implicated in pain mechanisms in both central and peripheral nervous systems
PMID: 38590871
8
GPR85 is among orphan GPCRs with important roles in CNS pathophysiology including schizophrenia, depression, and other major disorders
PMID: 29268243
Disease Associationsⓘ20
nervous system benign neoplasmOpen Targets
0.30Weak
malunion fractureOpen Targets
0.17Weak
placenta praeviaOpen Targets
0.15Weak
Abnormality of the skeletal systemOpen Targets
0.10Suggestive
atrial fibrillationOpen Targets
0.09Suggestive
obesityOpen Targets
0.08Suggestive
smoking initiationOpen Targets
0.08Suggestive
ovarian neoplasmOpen Targets
0.07Suggestive
joint diseaseOpen Targets
0.06Suggestive
overnutritionOpen Targets
0.06Suggestive
schizophreniaOpen Targets
0.03Suggestive
pyogenic granulomaOpen Targets
0.02Suggestive
glioblastoma multiformeOpen Targets
0.01Suggestive
psychiatric disorderOpen Targets
0.01Suggestive
autism spectrum disorderOpen Targets
0.01Suggestive
lung cancerOpen Targets
0.01Suggestive
neoplasmOpen Targets
0.01Suggestive
pituitary cancerOpen Targets
0.01Suggestive
chronic interstitial cystitisOpen Targets
0.01Suggestive
nervous system diseaseOpen Targets
0.01Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
CXCL14Protein interaction84%INSIG2Protein interaction78%GPR6Co-mentioned in literature20%GPR88Co-mentioned in literature20%GPR151Co-mentioned in literature20%GPR171Co-mentioned in literature20%
Tissue Expression6 tissues
Brain
100%
Heart
50%
Lung
10%
Liver
5%
Ovary
4%
Bone Marrow
1%
Gene Interaction Network
Click a node to explore
GPR85CXCL14INSIG2GPR6GPR88GPR151GPR171
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt P60893
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.59Moderately Constrained
pLIⓘ
0.85Intermediate
Observed/Expected LoF0.32 [0.18–0.59]
RankingsWhere GPR85 stands among ~20K protein-coding genes
  • #13,427of 20,598
    Most Researched23
  • #4,046of 17,882
    Most Constrained (LOEUF)0.59 · top quartile
Genes detectedGPR85
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Orphan G protein-coupled receptors: The role in CNS disorders.
PMID: 29268243
Biomed Pharmacother · 2018
1.00
2
Molecular insights into orphan G protein-coupled receptors relevant to schizophrenia.
PMID: 37605621
Br J Pharmacol · 2024
0.90
3
Sequence-structure based phylogeny of GPCR Class A Rhodopsin receptors.
PMID: 24503482
Mol Phylogenet Evol · 2014
0.80
4
The role of orphan G protein-coupled receptors in pain.
PMID: 38590871
Heliyon · 2024
0.70
5
A conserved mRNA expression profile of SREB2 (GPR85) in adult human, monkey, and rat forebrain.
PMID: 15893849
Brain Res Mol Brain Res · 2005
0.60