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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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GPRIN1
G protein regulated inducer of neurite outgrowth 1
Chromosome 5 · 5q35.2
NCBI Gene: 114787Ensembl: ENSG00000169258.8HGNC: HGNC:24835UniProt: Q7Z2K8
50PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingplasma membraneneuron projection developmentphosphoprotein bindinggastric cancerlung adenocarcinomaFTH1-related iron overloadhemochromatosis type 5
✦AI Summary

GPRIN1 (G protein regulated inducer of neurite outgrowth 1) functions as a multifaceted regulatory protein with significant roles in cancer progression and neuronal signaling. In cancer contexts, GPRIN1 acts as an oncogene that promotes tumor cell proliferation and survival through dual regulatory mechanisms 1. It functions as a transcriptional co-activator by scaffolding and stabilizing E2F1 to drive CDK1 expression, while simultaneously promoting CDK1 activation at the post-translational level by directing the kinase away from its inhibitor MYT1 toward its activator Cdc25C 1. This dual control of CDK1 triggers PI3K-Akt signaling cascades that couple cell cycle progression with mitochondrial homeostasis 1. GPRIN1 overexpression is associated with poor prognosis in multiple cancers, including lung cancer, breast cancer, and gallbladder cancer 231. In lung cancer, GPRIN1 facilitates proliferation and migration possibly through epithelial-mesenchymal transition pathways 2. Additionally, GPRIN1 interacts with 5-HT6 receptors independently of agonists, enhancing receptor activity in neuronal contexts 4. GPRIN1 also contributes to drug resistance mechanisms, as demonstrated in Taxol-resistant non-small cell lung cancer through the circ_0002360/miR-585-3p/GPRIN1 axis 5.

Sources cited
1
GPRIN1 functions as dual transcriptional co-activator and post-translational regulator of CDK1, controlling cell cycle and mitochondrial homeostasis
PMID: 41862463
2
GPRIN1 is overexpressed in lung cancer and promotes proliferation, migration, and epithelial-mesenchymal transition
PMID: 32755106
3
High GPRIN1 expression predicts poor prognosis in breast cancer
PMID: 36807044
4
GPRIN1 interacts with 5-HT6 receptors independently of agonists, enhancing receptor activity
PMID: 40347153
5
GPRIN1 contributes to Taxol resistance in non-small cell lung cancer through circ_0002360/miR-585-3p/GPRIN1 axis
PMID: 35293280
Disease Associationsⓘ20
gastric cancerOpen Targets
0.08Suggestive
lung adenocarcinomaOpen Targets
0.07Suggestive
FTH1-related iron overloadOpen Targets
0.04Suggestive
hemochromatosis type 5Open Targets
0.04Suggestive
isolated hyperferritinemiaOpen Targets
0.04Suggestive
hypoparathyroidism, familial isolated, 2Open Targets
0.04Suggestive
intracranial hemorrhageOpen Targets
0.04Suggestive
non-small cell lung carcinomaOpen Targets
0.04Suggestive
kidney diseaseOpen Targets
0.03Suggestive
familial isolated hyperparathyroidismOpen Targets
0.03Suggestive
hyperparathyroidismOpen Targets
0.03Suggestive
neoplasmOpen Targets
0.03Suggestive
hepatocellular carcinomaOpen Targets
0.03Suggestive
lung cancerOpen Targets
0.02Suggestive
ataxia telangiectasiaOpen Targets
0.02Suggestive
breast cancerOpen Targets
0.02Suggestive
esophageal squamous cell carcinomaOpen Targets
0.02Suggestive
cancerOpen Targets
0.01Suggestive
Colon Sessile Serrated Adenoma/PolypOpen Targets
0.01Suggestive
renal cell carcinomaOpen Targets
0.01Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
GPRIN2Shared pathway100%GPRIN3Shared pathway100%MECP2Protein interaction86%GNAZProtein interaction78%FRYShared pathway50%FRYLShared pathway50%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
2%
Lung
1%
Liver
1%
Heart
1%
Ovary
0%
Gene Interaction Network
Click a node to explore
GPRIN1GPRIN2GPRIN3MECP2GNAZFRYFRYL
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q7Z2K8
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.96LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF2.66 [0.83–1.96]
RankingsWhere GPRIN1 stands among ~20K protein-coding genes
  • #8,818of 20,598
    Most Researched50
  • #17,751of 17,882
    Most Constrained (LOEUF)1.96
Genes detectedGPRIN1
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Structural basis of ketamine action on human NMDA receptors.
PMID: 34321660
Nature · 2021
1.00
2
Dynamic network biomarker to determine the critical point of breast cancer stage progression.
PMID: 36807044
Breast Cancer · 2023
0.90
3
5-HT6 receptors: Contemporary views on their neurobiological and pharmacological relevance in neuropsychiatric disorders.
PMID: 40347153
Dialogues Clin Neurosci · 2025
0.80
4
Circular RNA circ_0002360 regulates the Taxol resistance and malignant behaviors of Taxol-resistant non-small cell lung cancer cells by microRNA-585-3p-dependent modulation of G protein regulated inducer of neurite outgrowth 1.
PMID: 35293280
Bioengineered · 2022
0.70
5
Disrupted callosal connectivity underlies long-lasting sensory-motor deficits in an NMDA receptor antibody encephalitis mouse model.
PMID: 39739422
J Clin Invest · 2024
0.60