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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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LPAR5
lysophosphatidic acid receptor 5
Chromosome 12 · 12p13.31
NCBI Gene: 57121Ensembl: ENSG00000184574.11HGNC: HGNC:13307UniProt: Q5KU18
40PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
behavioral response to painplasma membraneG protein-coupled receptor activityG protein-coupled receptor signaling pathwaytype 2 diabetes mellitusdiabetes mellituspapillary thyroid carcinomaneoplasm
✦AI Summary

LPAR5 (lysophosphatidic acid receptor 5) is a G protein-coupled receptor that mediates diverse cellular responses to lysophosphatidic acid (LPA) signaling 1. The receptor plays crucial roles in skin barrier function, where it promotes keratinocyte differentiation and filaggrin expression through the LPAR1/LPAR5-RHO-ROCK-SRF pathway, contributing to skin homeostasis and protection against allergens and pathogens 2. In nociception, LPAR5 is expressed in dorsal root ganglion neurons and skin keratinocytes, where it mediates itch responses, particularly non-histaminergic itch induced by compounds like hydroxychloroquine 3. LPAR5 has significant implications in cancer biology, where it promotes epithelial-to-mesenchymal transition (EMT) and radioresistance through ERK/Snail pathway activation 4. The receptor's expression is regulated by epigenetic mechanisms, including PARP1-mediated chr12 accessibility control of METTL3, which affects LPAR5 mRNA m6A methylation and stability 5. In the tumor microenvironment, LPAR5 expression in macrophages correlates with better prognosis in osteosarcoma and serves as a potential therapeutic target 6. Additionally, LPAR5 modulates neuroinflammation, as its suppression by PARP14 inhibits microglial activation and promotes post-stroke recovery 7.

Sources cited
1
LPAR5 is a G protein-coupled receptor that mediates diverse cellular responses to LPA signaling
PMID: 37061203
2
LPAR5 promotes keratinocyte differentiation and skin barrier function through RHO-ROCK-SRF pathway
PMID: 30447238
3
LPAR5 is expressed in dorsal root ganglion neurons and keratinocytes and mediates itch responses
PMID: 39125747
4
LPAR5 promotes EMT and radioresistance through ERK/Snail pathway
PMID: 36199069
5
LPAR5 expression is regulated by PARP1-mediated chromatin accessibility and METTL3-dependent m6A methylation
PMID: 37482682
6
LPAR5 expression in tumor-associated macrophages correlates with prognosis in osteosarcoma
PMID: 36591220
7
PARP14 suppresses LPAR5 to inhibit microglial activation and promote post-stroke recovery
PMID: 33317392
Disease Associationsⓘ20
type 2 diabetes mellitusOpen Targets
0.13Weak
diabetes mellitusOpen Targets
0.13Weak
papillary thyroid carcinomaOpen Targets
0.10Weak
neoplasmOpen Targets
0.09Suggestive
cancerOpen Targets
0.08Suggestive
psoriasisOpen Targets
0.08Suggestive
thyroid cancerOpen Targets
0.08Suggestive
osteosarcomaOpen Targets
0.06Suggestive
non-small cell lung carcinomaOpen Targets
0.04Suggestive
spinocerebellar ataxia type 14Open Targets
0.04Suggestive
Cerebral ischemiaOpen Targets
0.04Suggestive
attention deficit hyperactivity disorderOpen Targets
0.04Suggestive
childhood disintegrative disorderOpen Targets
0.04Suggestive
epilepsy, progressive myoclonic, 12Open Targets
0.04Suggestive
Potocki-Lupski syndromeOpen Targets
0.04Suggestive
hereditary attention deficit-hyperactivity disorderOpen Targets
0.04Suggestive
GM2-gangliosidosis, AB variantOpen Targets
0.03Suggestive
joint diseaseOpen Targets
0.03Suggestive
early-onset autosomal dominant Alzheimer diseaseOpen Targets
0.03Suggestive
15q11q13 microduplication syndromeOpen Targets
0.03Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
AGTProtein interaction99%CHRM1Protein interaction99%GNAQProtein interaction99%F2RProtein interaction98%GNA12Protein interaction98%GNA13Protein interaction98%
Tissue Expression6 tissues
Heart
100%
Bone Marrow
40%
Brain
38%
Lung
25%
Liver
13%
Ovary
12%
Gene Interaction Network
Click a node to explore
LPAR5AGTCHRM1GNAQF2RGNA12GNA13
PROTEIN STRUCTURE
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AlphaFoldAI-predicted · UniProt Q5KU18
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.74LoF Tolerant
pLIⓘ
0.40Tolerant
Observed/Expected LoF0.00 [0.00–1.74]
RankingsWhere LPAR5 stands among ~20K protein-coding genes
  • #10,196of 20,598
    Most Researched40
  • #16,278of 17,882
    Most Constrained (LOEUF)1.74
Genes detectedLPAR5
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
PARP14 inhibits microglial activation via LPAR5 to promote post-stroke functional recovery.
PMID: 33317392
Autophagy · 2021
1.00
2
Potential role of LPAR5 gene in prognosis and immunity of thyroid papillary carcinoma and pan-cancer.
PMID: 37037831
Sci Rep · 2023
0.90
3
Emerging roles of lysophosphatidic acid receptor subtype 5 (LPAR5) in inflammatory diseases and cancer.
PMID: 37061203
Pharmacol Ther · 2023
0.80
4
LPA Induces Keratinocyte Differentiation and Promotes Skin Barrier Function through the LPAR1/LPAR5-RHO-ROCK-SRF Axis.
PMID: 30447238
J Invest Dermatol · 2019
0.70
5
Lysophosphatidic Acid Receptors LPAR5 and LPAR2 Inversely Control Hydroxychloroquine-Evoked Itch and Scratching in Mice.
PMID: 39125747
Int J Mol Sci · 2024
0.60