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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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MAP3K9
mitogen-activated protein kinase kinase kinase 9
Chromosome 14 · 14q24.2
NCBI Gene: 4293Ensembl: ENSG00000006432.16HGNC: HGNC:6861UniProt: B4DZC4
38PubMed Papers
20Diseases
1Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
KinaseTranscription Factor
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
molecular function activator activityprotein phosphorylationprotein bindingprotein autophosphorylationneurodegenerative diseasemajor depressive disorderinsomniadepressive disorder
✦AI Summary

MAP3K9 is a serine/threonine kinase that functions as an upstream activator of the MKK/JNK signal transduction cascade, phosphorylating MAP2K4/MKK4 and MAP2K7/MKK7 to activate JNK signaling and regulate stress responses through transcription factors like AP-1 and GATA4. The protein also participates in mitochondrial death signaling pathways leading to apoptosis. MAP3K9 expression is tightly regulated by microRNA-mediated mechanisms. miR-148b, miR-23, miR-125b-5p, and miR-361-5p directly target MAP3K9 mRNA to suppress its protein levels 1 2 3 4. Additionally, circUGGT2 acts as a competing endogenous RNA, sponging miR-186-3p to upregulate MAP3K9 5. Post-translational regulation occurs via CBLB-mediated K48-K63-linked polyubiquitination at Lys193, targeting MAP3K9 for proteasomal degradation and suppressing MAPK-P38 pathway activation 6. Dysregulated MAP3K9 expression contributes to multiple pathologies. Elevated MAP3K9 promotes gastric cancer chemoresistance and progression through JNK signaling 5 2, enhances renal cancer proliferation and impairs apoptosis 1, increases glioblastoma invasion 6, and exacerbates shoulder arthritis progression by activating MMP expression 4. Conversely, MAP3K9 suppression by microRNA elevation correlates with improved survival and reduced malignancy in laryngeal squamous cell carcinoma 3. These findings establish MAP3K9 as a critical oncogenic hub amenable to therapeutic targeting.

Sources cited
1
circUGGT2 sponges miR-186-3p to upregulate MAP3K9 and promote gastric cancer progression and chemoresistance
PMID: 38729588
2
miR-148b directly targets MAP3K9, suppressing MAPK/JNK signaling; MAP3K9 overexpression in renal cell carcinoma tissues promotes proliferation
PMID: 26573018
3
miR-23 targets MAP3K9 to inhibit gastric cancer growth, migration, invasion and enhance chemosensitivity to cisplatin
PMID: 33277851
4
CBLB E3 ubiquitin ligase mediates K48-K63-linked polyubiquitination of MAP3K9 at Lys193, promoting degradation and suppressing MAPK-P38 pathway in glioblastoma
PMID: 40254893
5
IL-21 suppresses miR-361-5p, leading to MAP3K9 upregulation and increased MMP expression via ERK1/2/NF-κB pathway in shoulder arthritis
PMID: 38728237
6
miR-125b-5p directly targets MAP3K9; elevated miR-125b-5p correlates with improved survival and reduced proliferation/glycolysis in laryngeal squamous cell carcinoma
PMID: 35188403
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.50Moderate
major depressive disorderOpen Targets
0.41Moderate
insomniaOpen Targets
0.37Weak
depressive disorderOpen Targets
0.33Weak
mood disorderOpen Targets
0.32Weak
dysthymic disorderOpen Targets
0.32Weak
subarachnoid hemorrhageOpen Targets
0.27Weak
Febrile seizure (within the age range of 3 months to 6 years)Open Targets
0.22Weak
asthmaOpen Targets
0.18Weak
Parkinson diseaseOpen Targets
0.09Suggestive
pachyonychia congenitaOpen Targets
0.05Suggestive
neoplasmOpen Targets
0.05Suggestive
gliomaOpen Targets
0.05Suggestive
experimental autoimmune encephalomyelitisOpen Targets
0.05Suggestive
hepatocellular carcinomaOpen Targets
0.05Suggestive
prostate cancerOpen Targets
0.04Suggestive
Testicular regression syndromeOpen Targets
0.04Suggestive
melanomaOpen Targets
0.04Suggestive
X-linked intellectual disability - macrocephaly - macroorchidismOpen Targets
0.03Suggestive
X-linked intellectual disability-macrocephaly-macroorchidism syndromeOpen Targets
0.03Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets1
CEP-1347Phase II/III
Mitogen-activated protein kinase kinase kinase 10 inhibitor
asthma
Related Genes
MAP3K21Shared pathway50%MEX3BShared pathway50%TNK1Shared pathway50%CAMKK2Shared pathway43%MAPK6Shared pathway40%MAPK4Shared pathway40%
Tissue Expression6 tissues
Brain
100%
Liver
37%
Bone Marrow
22%
Lung
21%
Ovary
12%
Heart
11%
Gene Interaction Network
Click a node to explore
MAP3K9MAP3K21MEX3BTNK1CAMKK2MAPK6MAPK4
PROTEIN STRUCTURE
Preparing viewer…
PDB3DTC · 2.60 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.67LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.53 [0.41–0.67]
RankingsWhere MAP3K9 stands among ~20K protein-coding genes
  • #10,512of 20,598
    Most Researched38
  • #4,989of 17,882
    Most Constrained (LOEUF)0.67
Genes detectedMAP3K9
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
CircUGGT2 downregulation by METTL14-dependent m
PMID: 38729588
Pharmacol Res · 2024
1.00
2
MicroRNA-148b enhances proliferation and apoptosis in human renal cancer cells via directly targeting MAP3K9.
PMID: 26573018
Mol Med Rep · 2016
0.90
3
MicroRNA-23 regulates the growth, metastasis and chemosensitivity of human gastric cancer cells by targeting MAP3K9.
PMID: 33277851
J BUON · 2020
0.80
4
Mutations that prevent caspase cleavage of RIPK1 cause autoinflammatory disease.
PMID: 31827281
Nature · 2020
0.70
5
DNA-dependent protein kinase regulates lysosomal AMP-dependent protein kinase activation and autophagy.
PMID: 31983282
Autophagy · 2020
0.60