HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
MAPK4
mitogen-activated protein kinase 4
Chromosome 18 · 18q21.1-q21.2
NCBI Gene: 5596Ensembl: ENSG00000141639.12HGNC: HGNC:6878UniProt: B4DEW2
36PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingnucleuscytoplasmintracellular signal transductionhypertensionessential hypertensionresponse to xenobiotic stimulussquamous cell carcinoma
✦AI Summary

MAPK4 is an atypical mitogen-activated protein kinase that plays crucial roles in cellular proliferation, survival, and immune regulation. The protein exhibits oncogenic properties, being overexpressed in various cancers including glioma, triple-negative breast cancer, and prostate cancer, where it predicts poor prognosis 12. MAPK4 promotes tumor growth through multiple mechanisms: it activates AKT signaling independently of PI3K, enhances PDK1 protein synthesis, and stimulates the AKT/mTOR pathway to facilitate cell cycle progression and migration 231. This dual activation of AKT and PDK1 pathways contributes to cancer cell resistance against PI3K blockade therapy 3. In immune regulation, MAPK4 appears to have protective functions, as its deficiency leads to aberrant B cell activation in rheumatoid arthritis through disruption of the IRF4-SHIP1 signaling pathway, resulting in enhanced PI3K-AKT-mTOR signaling and increased IL-6 production 4. Clinically, MAPK4's role in cancer progression and therapy resistance makes it an attractive therapeutic target, with studies suggesting that co-targeting AKT and PDK1 could effectively treat MAPK4-high cancers 35.

Sources cited
1
MAPK4 is overexpressed in glioma, predicts poor prognosis, and promotes proliferation/migration via AKT/mTOR pathway
PMID: 36999945
2
MAPK4 enhances PDK1 protein synthesis and cooperatively activates PDK1 and AKT to promote cancer growth and therapy resistance
PMID: 37531320
3
MAPK4 promotes triple-negative breast cancer growth by activating AKT independent of PI3K and reduces tumor sensitivity to PI3K blockade
PMID: 35017531
4
MAPK4 deficiency leads to aberrant B cell activation in rheumatoid arthritis through disruption of IRF4-SHIP1 signaling pathway
PMID: 39863600
5
MAPK4 is a non-classical MAPK frequently overexpressed in various malignancies and orchestrates cellular processes via AKT/mTOR and PDK1 pathways
PMID: 38801852
Disease Associationsⓘ20
hypertensionOpen Targets
0.49Moderate
essential hypertensionOpen Targets
0.45Moderate
response to xenobiotic stimulusOpen Targets
0.31Weak
squamous cell carcinomaOpen Targets
0.30Weak
diabetes mellitusOpen Targets
0.30Weak
type 2 diabetes mellitusOpen Targets
0.30Weak
male infertilityOpen Targets
0.28Weak
azoospermiaOpen Targets
0.25Weak
protozoa infectious diseaseOpen Targets
0.21Weak
neoplasmOpen Targets
0.10Weak
gliomaOpen Targets
0.09Suggestive
triple-negative breast cancerOpen Targets
0.09Suggestive
cancerOpen Targets
0.09Suggestive
acute lung injuryOpen Targets
0.08Suggestive
gastric cancerOpen Targets
0.08Suggestive
cervical cancerOpen Targets
0.08Suggestive
infectionOpen Targets
0.07Suggestive
rheumatoid arthritisOpen Targets
0.07Suggestive
non-small cell lung carcinomaOpen Targets
0.07Suggestive
Miyoshi myopathyOpen Targets
0.07Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
MAPKAPK5Protein interaction100%MAPK6Protein interaction90%IGF2BP1Protein interaction82%XPO1Protein interaction80%MAP3K21Shared pathway67%MAP3K19Shared pathway67%
Tissue Expression6 tissues
Heart
100%
Brain
60%
Ovary
6%
Liver
5%
Lung
3%
Bone Marrow
0%
Gene Interaction Network
Click a node to explore
MAPK4MAPKAPK5MAPK6IGF2BP1XPO1MAP3K21MAP3K19
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt P31152
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.75LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.53 [0.38–0.75]
RankingsWhere MAPK4 stands among ~20K protein-coding genes
  • #10,812of 20,598
    Most Researched36
  • #5,972of 17,882
    Most Constrained (LOEUF)0.75
Genes detectedMAPK4
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
MAPK4 predicts poor prognosis and facilitates the proliferation and migration of glioma through the AKT/mTOR pathway.
PMID: 36999945
Cancer Med · 2023
1.00
2
Cooperative activation of PDK1 and AKT by MAPK4 enhances cancer growth and resistance to therapy.
PMID: 37531320
PLoS Biol · 2023
0.90
3
Polystyrene microspheres could inhibit the ferroptosis of prostate cancer cells via USP39/IGF2BP3/MAPK4 axis.
PMID: 40790750
J Transl Med · 2025
0.80
4
Atypical MAPKs in cancer.
PMID: 39348153
FEBS J · 2025
0.70
5
A review of non-classical MAPK family member, MAPK4: A pivotal player in cancer development and therapeutic intervention.
PMID: 38801852
Int J Biol Macromol · 2024
0.60