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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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MKNK1
MAPK interacting serine/threonine kinase 1
Chromosome 1 · 1p33
NCBI Gene: 8569Ensembl: ENSG00000079277.22HGNC: HGNC:7110UniProt: A0A499FJN1
103PubMed Papers
20Diseases
1Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
CLINICAL
Clinical Trials
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingprotein serine/threonine kinase activityprotein phosphorylationintracellular signal transductionneurodegenerative diseaseMyocardial Ischemianeoplasmhepatocellular carcinoma
✦AI Summary

MKNK1 is a serine/threonine kinase that regulates translation initiation by phosphorylating eIF4E, the 5' mRNA cap-binding protein, thereby controlling mRNA translation efficiency 1. As a downstream target of MAPK signaling pathways (ERK and p38), MKNK1 integrates stress responses and growth signals to modulate protein synthesis 1. Mechanistically, MKNK1 participates in the MNK/eIF4E axis that controls translation of specific mRNAs, including c-MYC in KRAS-mutant cancers 2. Beyond translation, MKNK1 regulates acinar cell secretion and proliferation in pancreatic tissue and influences nociceptor excitability in sensory ganglia 3, 1. Clinically, MKNK1 dysregulation contributes to multiple diseases. In aging-associated pancreatitis, miR-503-322 from senescent β-cells targets MKNK1 in acinar cells, impairing secretion and promoting autodigestion 3. MKNK1 overexpression mediates trastuzumab resistance in HER2-positive breast cancers through YB-1 activation and RSK-dependent phosphorylation 4. In KRAS-mutant colorectal cancer, MNK/eIF4E inhibition sensitizes tumors to mTORC1 inhibition by suppressing c-MYC expression, with implications for patient stratification 2. Additionally, MKNK1 regulates cancer stem cell properties and metabolic adaptation in breast and pancreatic cancers 5, while miR-370-3p-mediated MKNK1 inhibition suppresses adipogenesis and lipid accumulation 6. These findings establish MKNK1 as a therapeutic target across multiple cancer types and metabolic disorders.

Sources cited
1
miR-503-322 targets MKNK1 in pancreatic acinar cells to inhibit secretion and proliferation, driving aging-associated pancreatitis
PMID: 40097383
2
MKNK1 is a serine/threonine kinase that phosphorylates eIF4E and is downstream of ERK and p38 MAPK signaling; expressed in human nociceptors
PMID: 36764601
3
KRAS mutations rewire translation via MNK/eIF4E pathway to sustain c-MYC expression; MNK inhibition sensitizes KRAS-mutant colorectal cancers to rapamycin
PMID: 33328217
4
MKNK1 regulates cancer stem cell properties and metabolic adaptation (glycolysis vs. oxidative phosphorylation) in breast and pancreatic cancers; MNK1 loss suppresses liver metastasis
PMID: 39270021
5
MKNK1 is a YB-1 target gene that mediates trastuzumab resistance in HER2-positive breast cancer through RSK-dependent phosphorylation
PMID: 22249268
6
miR-370-3p targets MKNK1 to suppress adipogenesis, lipid accumulation, and regulate fatty acid metabolism
PMID: 34834018
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.37Weak
Myocardial IschemiaOpen Targets
0.26Weak
neoplasmOpen Targets
0.12Weak
hepatocellular carcinomaOpen Targets
0.11Weak
non-small cell lung carcinomaOpen Targets
0.10Suggestive
breast cancerOpen Targets
0.10Suggestive
triple-negative breast cancerOpen Targets
0.09Suggestive
colorectal carcinomaOpen Targets
0.09Suggestive
nasopharyngeal carcinomaOpen Targets
0.08Suggestive
colorectal cancerOpen Targets
0.08Suggestive
lymphomaOpen Targets
0.07Suggestive
cancerOpen Targets
0.06Suggestive
SepsisOpen Targets
0.05Suggestive
pancreatitisOpen Targets
0.05Suggestive
diffuse large B-cell lymphomaOpen Targets
0.04Suggestive
sinusitisOpen Targets
0.04Suggestive
prostate cancerOpen Targets
0.04Suggestive
acute myeloid leukemiaOpen Targets
0.04Suggestive
telomere syndromeOpen Targets
0.04Suggestive
melanomaOpen Targets
0.03Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets1
TOMIVOSERTIBPhase II
MAP kinase-interacting serine/threonine-protein kinase 1/2 inhibitor
colorectal cancer
Related Genes
SGK2Shared pathway100%MAPK1Protein interaction100%PABPC1Protein interaction100%MAPK14Protein interaction100%EIF4G3Protein interaction100%MAPK3Protein interaction99%
Tissue Expression6 tissues
Lung
100%
Ovary
56%
Liver
53%
Heart
42%
Bone Marrow
39%
Brain
24%
Gene Interaction Network
Click a node to explore
MKNK1SGK2MAPK1PABPC1MAPK14EIF4G3MAPK3
PROTEIN STRUCTURE
Preparing viewer…
PDB2Y9Q · 1.55 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.89LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.65 [0.48–0.89]
RankingsWhere MKNK1 stands among ~20K protein-coding genes
  • #4,652of 20,598
    Most Researched103 · top quartile
  • #7,896of 17,882
    Most Constrained (LOEUF)0.89
Genes detectedMKNK1
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Endocrine-exocrine miR-503-322 drives aging-associated pancreatitis via targeting MKNK1 in acinar cells.
PMID: 40097383
Nat Commun · 2025
1.00
2
Splicing factor YBX1 mediates persistence of JAK2-mutated neoplasms.
PMID: 33239784
Nature · 2020
0.90
3
MNK1 and MNK2 Expression in the Human Dorsal Root and Trigeminal Ganglion.
PMID: 36764601
Neuroscience · 2023
0.80
4
MNK1 and MNK2 expression in the human dorsal root and trigeminal ganglion.
PMID: 36711529
bioRxiv · 2023
0.70
5
Blocking tumor-intrinsic MNK1 kinase restricts metabolic adaptation and diminishes liver metastasis.
PMID: 39270021
Sci Adv · 2024
0.60