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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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MAPK6
mitogen-activated protein kinase 6
Chromosome 15 · 15q21.2
NCBI Gene: 5597Ensembl: ENSG00000069956.15HGNC: HGNC:6879UniProt: Q16659
84PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingMAP kinase activityprotein phosphorylationprotein serine/threonine kinase activityliver diseaseneurodegenerative diseaseosteoarthritis, kneeneuroinflammatory disorder
✦AI Summary

MAPK6 (ERK3) is an atypical mitogen-activated protein kinase that plays distinct roles in cancer progression and cellular signaling. Unlike conventional MAPKs, MAPK6 functions as an atypical kinase with unique regulatory mechanisms 1. The protein directly phosphorylates and activates AKT at serine 473 independently of mTORC2, promoting oncogenic signaling and tumor growth 2. This MAPK6-AKT axis contributes to resistance against mTOR kinase inhibitors, suggesting a major therapeutic resistance pathway 2. MAPK6 expression is elevated in multiple cancer types including breast cancer, lung adenocarcinoma, and clear cell renal cell carcinoma, where it correlates with poor patient survival 234. In lung adenocarcinoma, HNF4G transcriptionally upregulates MAPK6, enhancing cisplatin resistance through MAPK6/Akt pathway activation 4. MAPK6 also regulates endothelial inflammation in atherosclerosis via the EGR1/CXCL12 axis, where disturbed shear stress promotes TRIM21-mediated MAPK6 degradation 5. Additionally, MAPK6 contributes to diabetic nephropathy progression through podocyte injury mechanisms 6. These findings establish MAPK6 as a promising therapeutic target, with siRNA-loaded nanoparticles showing anticancer efficacy in breast cancer models 3.

Sources cited
1
MAPK6 is an atypical MAPK with distinctive features different from conventional family members
PMID: 39348153
2
MAPK6 directly phosphorylates AKT at S473 independent of mTORC2 and promotes tumor growth and mTOR inhibitor resistance
PMID: 34767444
3
MAPK6 is upregulated in breast cancer and siRNA-loaded nanoparticles targeting MAPK6 show anticancer effects
PMID: 39823246
4
HNF4G increases cisplatin resistance in lung adenocarcinoma via transcriptional regulation of MAPK6
PMID: 36923501
5
MAPK6 regulates endothelial inflammation in atherosclerosis and is degraded by TRIM21 under disturbed shear stress
PMID: 39763069
6
MAPK6 contributes to podocyte injury and diabetic nephropathy progression
PMID: 37440116
Disease Associationsⓘ20
liver diseaseOpen Targets
0.29Weak
neurodegenerative diseaseOpen Targets
0.29Weak
osteoarthritis, kneeOpen Targets
0.25Weak
neuroinflammatory disorderOpen Targets
0.24Weak
Alzheimer diseaseOpen Targets
0.20Weak
osteoarthritisOpen Targets
0.18Weak
adolescent idiopathic scoliosisOpen Targets
0.15Weak
cancerOpen Targets
0.11Weak
breast cancerOpen Targets
0.09Suggestive
total knee arthroplastyOpen Targets
0.09Suggestive
neoplasmOpen Targets
0.08Suggestive
triple-negative breast cancerOpen Targets
0.08Suggestive
head and neck malignant neoplasiaOpen Targets
0.08Suggestive
intrahepatic cholangiocarcinomaOpen Targets
0.07Suggestive
lung adenocarcinomaOpen Targets
0.07Suggestive
azoospermiaOpen Targets
0.07Suggestive
lung cancerOpen Targets
0.06Suggestive
pneumoniaOpen Targets
0.06Suggestive
Congenital pulmonary alveolar proteinosisOpen Targets
0.06Suggestive
Neonatal acute respiratory distress with surfactant metabolism deficiencyOpen Targets
0.05Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
NEURL4Protein interaction94%CCND3Protein interaction93%UBE3AProtein interaction91%SEPTIN7Protein interaction91%MAPK4Protein interaction90%HERC2Protein interaction89%
Tissue Expression6 tissues
Bone Marrow
100%
Brain
60%
Liver
49%
Heart
22%
Lung
21%
Ovary
15%
Gene Interaction Network
Click a node to explore
MAPK6NEURL4CCND3UBE3ASEPTIN7MAPK4HERC2
PROTEIN STRUCTURE
Preparing viewer…
PDB7AQB · 2.25 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.47Moderately Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.31 [0.22–0.47]
RankingsWhere MAPK6 stands among ~20K protein-coding genes
  • #5,679of 20,598
    Most Researched84
  • #2,643of 17,882
    Most Constrained (LOEUF)0.47 · top quartile
Genes detectedMAPK6
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Aberrant activation of m6A demethylase FTO renders HIF2α
PMID: 34586831
Sci Transl Med · 2021
1.00
2
Disturbed shear stress promotes atherosclerosis through TRIM21-regulated MAPK6 degradation and consequent endothelial inflammation.
PMID: 39763069
Clin Transl Med · 2025
0.90
3
Atypical MAPKs in cancer.
PMID: 39348153
FEBS J · 2025
0.80
4
Transcriptome analysis of the cytokine storm-related genes among the subtypes of idiopathic multicentric Castleman disease.
PMID: 39462545
J Clin Exp Hematop · 2024
0.70
5
CircGAB1 Facilitates Podocyte Injury Through Sponging miR-346 and Activating MAPK6 in Diabetic Nephropathy.
PMID: 37440116
Appl Biochem Biotechnol · 2024
0.60