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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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PHLPP2
PH domain and leucine rich repeat protein phosphatase 2
Chromosome 16 · 16q22.2
NCBI Gene: 23035Ensembl: ENSG00000040199.19HGNC: HGNC:29149UniProt: Q6ZVD8
89PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Tumor Suppressor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
cytosolcytoplasmprotein bindingintercellular bridgeAbnormality of the skeletal systemneurodegenerative diseasebreast cancerneoplasm
✦AI Summary

PHLPP2 is a member of the metal-dependent protein phosphatase (PPM) family involved in regulating Akt and PKC signaling 1. However, recent structural analysis reveals that PHLPP2 is a pseudophosphatase that lost catalytic activity in the metazoan ancestor, containing a single zinc ion in its catalytic center but lacking enzymatic activity in vitro 2. Despite this surprising finding, PHLPP2 retains functional importance through noncatalytic mechanisms, potentially serving a scaffolding role on membranes 2. In disease contexts, PHLPP2 functions as a tumor suppressor through the PI3K-AKT pathway regulation. CircANAPC7 suppresses pancreatic cancer growth and cachexia by acting as a miR-373 sponge to maintain PHLPP2 expression, which dephosphorylates AKT and inhibits proliferation 3. In hepatocellular carcinoma, TRIM22-mediated PHLPP2 degradation activates AKT-p53-p21 signaling and induces cellular senescence 4. Conversely, downregulation of PHLPP2 by exosomal miR-25-3p in gliomas and miR-188-3p in colorectal cancer promotes tumor progression by activating PI3K-AKT-mTOR signaling 56. In cardiac tissue, METTL14-mediated suppression of Phlpp2 m6A modification activates AKT-S473, promoting physiological hypertrophy and protecting against ischemia-reperfusion injury 7. Genetic polymorphisms in PHLPP2 (rs61733127) are associated with increased colon cancer susceptibility 8.

Sources cited
1
PHLPP2 is a member of the metal-dependent protein phosphatase (PPM) family with conserved catalytic core region
PMID: 32650009
2
PHLPP2 is a pseudophosphatase that lost catalytic activity in metazoan ancestors, containing a zinc ion but lacking enzymatic activity in vitro
PMID: 40168118
3
PHLPP2 suppresses pancreatic cancer growth and cachexia through AKT dephosphorylation and downstream effects on cyclin D1 and TGF-β
PMID: 35176309
4
TRIM22-mediated PHLPP2 degradation activates AKT-p53-p21 signaling and induces cellular senescence in hepatocellular carcinoma
PMID: 38199981
5
Exosomal miR-25-3p downregulates PHLPP2 expression in macrophages, activating PI3K-AKT-mTOR signaling and promoting M2 polarization in gliomas
PMID: 39407269
6
Exosomal miR-188-3p from colorectal cancer cells targets PHLPP2 to activate AKT/mTOR pathway and promote liver metastasis
PMID: 40134019
7
METTL14-mediated suppression of Phlpp2 m6A modification activates AKT-S473 in cardiomyocytes, promoting physiological hypertrophy
PMID: 36351918
8
PHLPP2 gene L1016S polymorphism (rs61733127) is associated with increased colon cancer risk
PMID: 34193013
Disease Associationsⓘ20
Abnormality of the skeletal systemOpen Targets
0.39Weak
neurodegenerative diseaseOpen Targets
0.37Weak
breast cancerOpen Targets
0.09Suggestive
neoplasmOpen Targets
0.09Suggestive
lymphatic system diseaseOpen Targets
0.09Suggestive
colorectal carcinomaOpen Targets
0.08Suggestive
hepatocellular carcinomaOpen Targets
0.08Suggestive
urinary bladder carcinomaOpen Targets
0.08Suggestive
ulcerative colitisOpen Targets
0.07Suggestive
depressive disorderOpen Targets
0.06Suggestive
non-small cell lung carcinomaOpen Targets
0.06Suggestive
cancerOpen Targets
0.06Suggestive
glomerulonephritisOpen Targets
0.05Suggestive
head and neck squamous cell carcinomaOpen Targets
0.05Suggestive
goutOpen Targets
0.05Suggestive
triple-negative breast cancerOpen Targets
0.05Suggestive
Neck painOpen Targets
0.04Suggestive
Shoulder painOpen Targets
0.04Suggestive
gliomaOpen Targets
0.04Suggestive
gastric cancerOpen Targets
0.03Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
AKT1Protein interaction100%AKT2Protein interaction99%USP1Protein interaction99%AKT3Protein interaction99%PTENProtein interaction98%USP12Protein interaction94%
Tissue Expression6 tissues
Bone Marrow
100%
Brain
53%
Ovary
51%
Lung
28%
Liver
27%
Heart
26%
Gene Interaction Network
Click a node to explore
PHLPP2AKT1AKT2USP1AKT3PTENUSP12
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q6ZVD8
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.68LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.54 [0.43–0.68]
RankingsWhere PHLPP2 stands among ~20K protein-coding genes
  • #5,374of 20,598
    Most Researched89
  • #5,119of 17,882
    Most Constrained (LOEUF)0.68
Genes detectedPHLPP2
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Metal-dependent Ser/Thr protein phosphatase PPM family: Evolution, structures, diseases and inhibitors.
PMID: 32650009
Pharmacol Ther · 2020
1.00
2
Hypoxic glioma-derived exosomal miR-25-3p promotes macrophage M2 polarization by activating the PI3K-AKT-mTOR signaling pathway.
PMID: 39407269
J Nanobiotechnology · 2024
0.90
3
METTL14 is required for exercise-induced cardiac hypertrophy and protects against myocardial ischemia-reperfusion injury.
PMID: 36351918
Nat Commun · 2022
0.80
4
Circular RNA ANAPC7 Inhibits Tumor Growth and Muscle Wasting via PHLPP2-AKT-TGF-β Signaling Axis in Pancreatic Cancer.
PMID: 35176309
Gastroenterology · 2022
0.70
5
TRIM22 induces cellular senescence by targeting PHLPP2 in hepatocellular carcinoma.
PMID: 38199981
Cell Death Dis · 2024
0.60