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26 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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PRKCQ
protein kinase C theta
Chromosome 10 · 10p15.1
NCBI Gene: 5588Ensembl: ENSG00000065675.17HGNC: HGNC:9410UniProt: Q04759
243PubMed Papers
20Diseases
5Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
RESEARCH IMPACT
Trending
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
negative regulation of insulin receptor signaling pathwaycell chemotaxiscentriolar satellitediacylglycerol-dependent, calcium-independent serine/threonine kinase activityasthmaacute myeloid leukemiaatopic eczemaEczematoid dermatitis
✦AI Summary

PRKCQ (protein kinase C theta) is a calcium-independent serine/threonine kinase localized to chromosome 10 that functions as a critical mediator of T-cell receptor (TCR) signaling and immune responses. In T cells, PRKCQ phosphorylates CARD11 to activate the canonical NF-κB pathway and regulates transcription factors including NF-κB, JUN, NFATC1, and NFATC2, driving IL-2 production and T-cell activation 1. PRKCQ plays essential roles in Th2 cell development and Th17 cell differentiation during inflammatory responses, while having minor involvement in Th1 responses 1. Beyond immune function, PRKCQ mediates phagocytosis by phosphorylating WIP during macrophage antibody-dependent cellular cytotoxicity, enabling tumor cell phagocytosis 2. The kinase also regulates platelet signaling and may suppress insulin signaling by phosphorylating IRS1. Dysregulation of PRKCQ associates with multiple autoimmune diseases, including Vogt-Koyanagi-Harada syndrome, as demonstrated by genetic polymorphism studies 1. In cancer, particularly triple-negative breast cancer, PRKCQ promotes cell survival and chemotherapy resistance through suppression of pro-apoptotic Bim; PRKCQ inhibition enhances chemosensitivity 3. PRKCQ expression is also linked to breast cancer proliferation and inflammation via NF-κB pathway activation 4, while PRKCQ-AS1 lncRNA regulates cancer metabolism and paclitaxel resistance 56.

Sources cited
1
PRKCQ rs4750316 polymorphism is associated with Vogt-Koyanagi-Harada syndrome susceptibility and involvement in TCR signaling pathways
PMID: 31908401
2
PKC-θ phosphorylates WIP during macrophage phagocytosis to enable tumor cell uptake induced by therapeutic antibodies
PMID: 35484420
3
PRKCQ promotes chemotherapy resistance in triple-negative breast cancer by suppressing pro-apoptotic Bim; PRKCQ inhibition enhances chemosensitivity
PMID: 32600444
4
PRKCQ mediates NF-κB-dependent proliferation and inflammation in breast cancer cells
PMID: 35447530
5
lncRNA PRKCQ-AS1 regulates glycolysis and mitochondrial function in papillary thyroid carcinoma via IGF2BPs/PRMT7 signaling
PMID: 38092752
6
lncRNA PRKCQ-AS1 promotes paclitaxel resistance in triple-negative breast cancer through miR-361-5p/PIK3C3-mediated autophagy
PMID: 36732923
Disease Associationsⓘ20
asthmaOpen Targets
0.55Moderate
acute myeloid leukemiaOpen Targets
0.53Moderate
atopic eczemaOpen Targets
0.51Moderate
Eczematoid dermatitisOpen Targets
0.48Moderate
systemic mastocytosisOpen Targets
0.48Moderate
mast-cell leukemiaOpen Targets
0.47Moderate
allergic rhinitisOpen Targets
0.47Moderate
childhood onset asthmaOpen Targets
0.46Moderate
respiratory system diseaseOpen Targets
0.46Moderate
MastocytosisOpen Targets
0.46Moderate
inflammatory bowel disease 1Open Targets
0.43Moderate
hypothyroidismOpen Targets
0.42Moderate
rheumatoid arthritisOpen Targets
0.42Moderate
neoplasmOpen Targets
0.40Weak
myxedemaOpen Targets
0.39Weak
acute myeloid leukemia by FAB classificationOpen Targets
0.37Weak
polymyalgia rheumaticaOpen Targets
0.34Weak
atopic asthmaOpen Targets
0.34Weak
Abnormal thrombosisOpen Targets
0.34Weak
allergic diseaseOpen Targets
0.34Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets5
CEP-2563Phase I
Protein kinase C (PKC) inhibitor
GSK-690693Phase I
Protein kinase C (PKC) inhibitor
MIDOSTAURINApproved
Tyrosine-protein kinase receptor FLT3 inhibitor
mast-cell leukemia
SOTRASTAURINPhase II
Protein kinase C (PKC) inhibitor
kidney transplant
UCN-01Phase II
3-phosphoinositide dependent protein kinase-1 inhibitor
non-small cell lung carcinoma
Related Genes
RELAProtein interaction100%IKBKGProtein interaction100%MAPK8Protein interaction99%LCKProtein interaction97%PLCG1Protein interaction97%PRKCBProtein interaction97%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
85%
Lung
62%
Ovary
15%
Liver
9%
Heart
5%
Gene Interaction Network
Click a node to explore
PRKCQRELAIKBKGMAPK8LCKPLCG1PRKCB
PROTEIN STRUCTURE
Preparing viewer…
PDB1XJD · 2.00 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.57Moderately Constrained
pLIⓘ
0.01Tolerant
Observed/Expected LoF0.44 [0.34–0.57]
RankingsWhere PRKCQ stands among ~20K protein-coding genes
  • #1,606of 20,598
    Most Researched243 · top 10%
  • #832of 1,025
    FDA-Approved Drug Targets1
  • #3,755of 17,882
    Most Constrained (LOEUF)0.57 · top quartile
Genes detectedPRKCQ
Sources retrieved26 papers
Response time—
📄 Sources
26▼
1
Macrophage mitochondrial fission improves cancer cell phagocytosis induced by therapeutic antibodies and is impaired by glutamine competition.
PMID: 35484420
Nat Cancer · 2022
1.00
2
BNIP3L/Nix-induced mitochondrial fission, mitophagy, and impaired myocyte glucose uptake are abrogated by PRKA/PKA phosphorylation.
PMID: 33044904
Autophagy · 2021
0.90
3
Molecular characterization of the human protein kinase C theta gene locus (PRKCQ).
PMID: 9790596
Mol Gen Genet · 1998
0.80
4
Fasting regulates mitochondrial function through lncRNA PRKCQ-AS1-mediated IGF2BPs in papillary thyroid carcinoma.
PMID: 38092752
Cell Death Dis · 2023
0.70
5
Clinical significance and biological function of PRKCQ-AS1/miR-582-3p expression in LUAD.
PMID: 40597380
Hereditas · 2025
0.68